Literature DB >> 22968839

Efficient assembly of iminodicarboxamides by a "truly" four-component reaction.

Kareem Khoury1, Mantosh K Sinha, Tadamichi Nagashima, Eberhardt Herdtweck, Alexander Dömling.   

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Year:  2012        PMID: 22968839      PMCID: PMC3874142          DOI: 10.1002/anie.201205366

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN: 1433-7851            Impact factor:   15.336


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  24 in total

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4.  Multicomponent synthesis of 2-imidazolines.

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5.  Short and novel stereospecific synthesis of trisubstituted 2,5-diketopiperazines.

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6.  An efficient synthesis of morpholin-2-one derivatives using glycolaldehyde dimer by the Ugi multicomponent reaction.

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  13 in total

1.  Isocyanide-Based Multicomponent Reactions of Free Phenylboronic Acids.

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2.  Synthesis of isoindolin-1-one derivatives via multicomponent reactions of methyl 2-formylbenzoate and intramolecular amidation.

Authors:  Jie Lei; Zhi-Gang Xu; Shi-Qiang Li; Jia Xu; Jin Zhu; Zhong-Zhu Chen
Journal:  Mol Divers       Date:  2016-06-07       Impact factor: 2.943

3.  With unprotected amino acids to tetrazolo peptidomimetics.

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4.  MCR synthesis of a tetracyclic tetrazole scaffold.

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5.  Towards a facile and convenient synthesis of highly functionalized indole derivatives based on multi-component reactions.

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6.  Efficient isocyanide-less isocyanide-based multicomponent reactions.

Authors:  Constantinos G Neochoritis; Silvia Stotani; Bhupendra Mishra; Alexander Dömling
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7.  Expanding the substrate scope of Ugi five-center, four-component reaction U-5C-4CR): ketones as coupling partners for secondary amino acids.

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8.  Multicomponent synthesis of diverse 1,4-benzodiazepine scaffolds.

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9.  Various cyclization scaffolds by a truly Ugi 4-CR.

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10.  Tricycles by a new Ugi variation and Pictet-Spengler reaction in one pot.

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