Literature DB >> 19835352

Rapid discovery of triazolobenzylidene-thiazolopyrimidines (TBTP) as CDC25 phosphatase inhibitors by parallel click chemistry and in situ screening.

Romain Duval1, Stéphanie Kolb, Emmanuelle Braud, David Genest, Christiane Garbay.   

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Year:  2009        PMID: 19835352     DOI: 10.1021/cc900140f

Source DB:  PubMed          Journal:  J Comb Chem        ISSN: 1520-4766


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  9 in total

Review 1.  Comprehensive survey of chemical libraries for drug discovery and chemical biology: 2009.

Authors:  Roland E Dolle; Bertrand Le Bourdonnec; Karin Worm; Guillermo A Morales; Craig J Thomas; Wei Zhang
Journal:  J Comb Chem       Date:  2010-10-05

2.  Efficient and green synthesis of novel hexahydro-5H-thiazolo[2',3':2,3]pyrimido[4,5-b]quinoline derivatives.

Authors:  Tooba Tabibi; Abbas Ali Esmaeili
Journal:  Mol Divers       Date:  2022-05-08       Impact factor: 2.943

Review 3.  A Comprehensive Overview of the Developments of Cdc25 Phosphatase Inhibitors.

Authors:  Ahmed Bakr Abdelwahab; Eslam Reda El-Sawy; Atef G Hanna; Denyse Bagrel; Gilbert Kirsch
Journal:  Molecules       Date:  2022-04-07       Impact factor: 4.927

Review 4.  CuAAC click chemistry accelerates the discovery of novel chemical scaffolds as promising protein tyrosine phosphatases inhibitors.

Authors:  X-P He; J Xie; Y Tang; J Li; G-R Chen
Journal:  Curr Med Chem       Date:  2012       Impact factor: 4.530

5.  Microwave assisted synthesis of some new thiazolopyrimidine, thiazolodipyrimidine and thiazolopyrimidothiazolopyrimidine derivatives with potential antioxidant and antimicrobial activity.

Authors:  Mohamed M Youssef; Mahmoud A Amin
Journal:  Molecules       Date:  2012-08-13       Impact factor: 4.411

6.  Synthesis and Anticancer Activity of New 1-Thia-4-azaspiro[4.5]decane, Their Derived Thiazolopyrimidine and 1,3,4-Thiadiazole Thioglycosides.

Authors:  Eman M Flefel; Wael A El-Sayed; Ashraf M Mohamed; Walaa I El-Sofany; Hanem M Awad
Journal:  Molecules       Date:  2017-01-20       Impact factor: 4.411

7.  Visible-light driven regioselective synthesis, characterization and binding studies of 2-aroyl-3-methyl-6,7-dihydro-5H-thiazolo[3,2-a]pyrimidines with DNA and BSA using biophysical and computational techniques.

Authors:  Ranjana Aggarwal; Naman Jain; Shilpa Sharma; Prince Kumar; Gyan Prakash Dubey; Heerak Chugh; Ramesh Chandra
Journal:  Sci Rep       Date:  2021-11-11       Impact factor: 4.379

8.  Microwave assisted synthesis of some new thiazolopyrimidine and pyrimidothiazolopyrimidopyrimidine derivatives with potential antimicrobial activity.

Authors:  Ayman M S Youssef; Ahmed M Fouda; Rasha M Faty
Journal:  Chem Cent J       Date:  2018-05-05       Impact factor: 4.215

9.  Synthesis and Cytotoxic Activity of New Thiazolopyrimidine Sugar Hydrazones and Their Derived Acyclic Nucleoside Analogues.

Authors:  Ebtesam A Basiony; Allam A Hassan; Zahra M Al-Amshany; Ahmed A Abd-Rabou; Adel A-H Abdel-Rahman; Nasser A Hassan; Wael A El-Sayed
Journal:  Molecules       Date:  2020-01-18       Impact factor: 4.411

  9 in total

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