Literature DB >> 20923157

Comprehensive survey of chemical libraries for drug discovery and chemical biology: 2009.

Roland E Dolle1, Bertrand Le Bourdonnec, Karin Worm, Guillermo A Morales, Craig J Thomas, Wei Zhang.   

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Year:  2010        PMID： 20923157      PMCID： PMC4140011          DOI： 10.1021/cc100128w

Source DB:  PubMed          Journal:  J Comb Chem        ISSN： 1520-4766


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  325 in total

1.  Normal-phase automated mass-directed HPLC purification of a pyrrolobenzodiazepine library with vasopressin agonist activity.

Authors:  Michael Kagan; Michael Chlenov; Sergey Melnikov; Oliver McConnell; Alvin C Bach; Guy Carter; Amedeo Failli; Thomas J Caggiano; Jay S Shumsky; Dieter Lubda
Journal:  J Comb Chem       Date:  2009 Jul-Aug

2.  Access to flavones via a microwave-assisted, one-pot Sonogashira-carbonylation-annulation reaction.

Authors:  Emelia Awuah; Alfredo Capretta
Journal:  Org Lett       Date:  2009-08-06       Impact factor: 6.005

3.  Discovery of small molecule human C5a receptor antagonists.

Authors:  Hitesh J Sanganee; Andrew Baxter; Simon Barber; Alastair J H Brown; Denise Grice; Fraser Hunt; Sarah King; David Laughton; Garry Pairaudeau; Bob Thong; Richard Weaver; John Unitt
Journal:  Bioorg Med Chem Lett       Date:  2008-12-31       Impact factor: 2.823

4.  Design, synthesis and biological evaluation of novel pyridine derivatives as anticancer agents and phosphodiesterase 3 inhibitors.

Authors:  Ashraf H Abadi; Tamer M Ibrahim; Khaled M Abouzid; Jochen Lehmann; Heather N Tinsley; Bernard D Gary; Gary A Piazza
Journal:  Bioorg Med Chem       Date:  2009-07-03       Impact factor: 3.641

5.  Efficient three-component Strecker reaction of aldehydes/ketones via NHC-amidate palladium(II) complex catalysis.

Authors:  Jamie Jarusiewicz; Yvonne Choe; Kyung Soo Yoo; Chan Pil Park; Kyung Woon Jung
Journal:  J Org Chem       Date:  2009-04-03       Impact factor: 4.354

6.  A new entry of copper-catalyzed four-component reaction: facile access to alpha-aryl beta-hydroxy imidates.

Authors:  Eun Jeong Yoo; Sae Hume Park; Sang Hyup Lee; Sukbok Chang
Journal:  Org Lett       Date:  2009-03-05       Impact factor: 6.005

7.  Small molecule inhibitors of Myc/Max dimerization and Myc-induced cell transformation.

Authors:  Jin Shi; James S Stover; Landon R Whitby; Peter K Vogt; Dale L Boger
Journal:  Bioorg Med Chem Lett       Date:  2009-09-17       Impact factor: 2.823

8.  Traceless solid-phase synthesis of heteroannulated 1,3-oxazin-6-ones.

Authors:  Jun Che; Makam S Raghavendra; Yulin Lam
Journal:  J Comb Chem       Date:  2009 May-Jun

9.  Fluorous parallel synthesis of a piperazinedione-fused tricyclic compound library.

Authors:  Stefan Werner; Simon D Nielsen; Peter Wipf; David M Turner; Peter G Chambers; Steven J Geib; Dennis P Curran; Wei Zhang
Journal:  J Comb Chem       Date:  2009 May-Jun

10.  Syntheses of aminoalcohol-derived macrocycles leading to a small-molecule binder to and inhibitor of Sonic Hedgehog.

Authors:  Lee F Peng; Benjamin Z Stanton; Nicole Maloof; Xiang Wang; Stuart L Schreiber
Journal:  Bioorg Med Chem Lett       Date:  2009-09-25       Impact factor: 2.823
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  16 in total

1.  Synthesis of a unique isoindoline/tetrahydroisoquinoline-based tricyclic sultam library utilizing a Heck-aza-Michael strategy.

Authors:  Qin Zang; Salim Javed; Patrick Porubsky; Farman Ullah; Benjamin Neuenswander; Gerald H Lushington; Fatima Z Basha; Michael G Organ; Paul R Hanson
Journal:  ACS Comb Sci       Date:  2012-02-06       Impact factor: 3.784

2.  Facile (triazolyl)methylation of MACOS-derived benzofused sultams utilizing ROMP-derived OTP reagents.

Authors:  Saqib Faisal; Farman Ullah; Pradip K Maity; Alan Rolfe; Thiwanka B Samarakoon; Patrick Porubsky; Benjamin Neuenswander; Gerald H Lushington; Fatima Z Basha; Michael G Organ; Paul R Hanson
Journal:  ACS Comb Sci       Date:  2012-03-05       Impact factor: 3.784

3.  Recent progress on fluorous synthesis of biologically interesting compounds.

Authors:  Zhong-Xing Jiang; Sanjun Zhi; Wei Zhang
Journal:  Mol Divers       Date:  2014-01-20       Impact factor: 2.943

4.  Silica-Supported Oligomeric Benzyl Phosphate (Si-OBP) and Triazole Phosphate (Si-OTP) Alkylating Reagents.

Authors:  Pradip K Maity; Saqib Faisal; Alan Rolfe; Diana Stoianova; Paul R Hanson
Journal:  J Org Chem       Date:  2015-10-02       Impact factor: 4.354

5.  Triazole-containing isothiazolidine 1,1-dioxide library synthesis: one-pot, multi-component protocols for small molecular probe discovery.

Authors:  Alan Rolfe; Thomas O Painter; Naeem Asad; Moon Young Hur; Kyu Ok Jeon; Marek Brzozowski; Sarra V Klimberg; Patrick Porubsky; Benjamin Neuenswander; Gerald H Lushington; Conrad Santini; Paul R Hanson
Journal:  ACS Comb Sci       Date:  2011-08-25       Impact factor: 3.784

6.  Synthesis of novel 4H-pyrimido[1,6-a]pyrimidines via a one-pot three-component condensation.

Authors:  Jinbao Xiang; Hanghang Li; Kai Yang; Lang Yi; Yongnan Xu; Qun Dang; Xu Bai
Journal:  Mol Divers       Date:  2011-12-04       Impact factor: 2.943

7.  Synthesis of amino-benzothiaoxazepine-1,1-dioxides utilizing a microwave-assisted, S(N)Ar protocol.

Authors:  Alan Rolfe; Farman Ullah; Thiwanka B Samarakoon; Ryan D Kurtz; Patrick Porubsky; Benjamin Neuenswander; Gerald H Lushington; Conrad Santini; Michael G Organ; Paul R Hanson
Journal:  ACS Comb Sci       Date:  2011-09-08       Impact factor: 3.784

8.  Diversity through phosphine catalysis identifies octahydro-1,6-naphthyridin-4-ones as activators of endothelium-driven immunity.

Authors:  Daniel Cruz; Zhiming Wang; Jon Kibbie; Robert Modlin; Ohyun Kwon
Journal:  Proc Natl Acad Sci U S A       Date:  2011-03-07       Impact factor: 11.205

9.  A novel method for the determination of isokinetic ratios and its application in the synthesis of two new positional scanning libraries.

Authors:  Marc A Giulianotti; Ginamarie Debevec; Radleigh G Santos; Laura E Maida; Wenteng Chen; Lili Ou; Yongping Yu; Colette T Dooley; Richard A Houghten
Journal:  ACS Comb Sci       Date:  2012-08-28       Impact factor: 3.784

10.  Parallel synthesis of 7-heteroaryl-pyrazolo[1,5-a]pyrimidine-3-carboxamides.

Authors:  Sizana Ahmetaj; Nina Velikanje; Uroš Grošelj; Ines Šterbal; Benjamin Prek; Amalija Golobič; Drago Kočar; Georg Dahmann; Branko Stanovnik; Jurij Svete
Journal:  Mol Divers       Date:  2013-08-22       Impact factor: 2.943
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