Literature DB >> 4145013

Measurement of hydrophobicity, surface activity, local anaesthesia, and myocardial conduction velocity as quantitative parameters of the non-specific membrane affinity of nine -adrenergic blocking agents.

D Hellenbrecht, B Lemmer, G Wiethold, H Grobecker.   

Abstract

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Substances：

Year:  1973        PMID： 4145013     DOI： 10.1007/bf00501161

Source DB:  PubMed          Journal:  Naunyn Schmiedebergs Arch Pharmacol        ISSN： 0028-1298            Impact factor:   3.000


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  18 in total

Review 1.  Linear relationships between lipophilic character and biological activity of drugs.

Authors:  C Hansch; W J Dunn
Journal:  J Pharm Sci       Date:  1972-01       Impact factor: 3.534

2.  A comparison of the local anaesthetic-, "quinidine-like"- and adrenergic beta-blocking-activities of five beta-receptor antagonists.

Authors:  W G Davis
Journal:  J Pharm Pharmacol       Date:  1970-04       Impact factor: 3.765

3.  Myocardial and local anesthetic actions of beta-adrenergic receptor blocking drugs: relationship to physicochemical properties.

Authors:  J V Levy
Journal:  Eur J Pharmacol       Date:  1968-02       Impact factor: 4.432

4.  Surface tension effects of beta-adrenergic blocking drugs.

Authors:  J V Levy
Journal:  J Pharm Pharmacol       Date:  1968-10       Impact factor: 3.765

Review 5.  [Mechanism of action of local anesthetics].

Authors:  H F Zipf
Journal:  Pharm Acta Helv       Date:  1967 Aug-Oct

Review 6.  [Change relations between the active substance and receptor in local anesthetics of the N-aminoacylephedrine type].

Authors:  H Schönenberger; A Petter; W Zwez
Journal:  Pharm Acta Helv       Date:  1967 Aug-Oct

Review 7.  [Chemical constitution, chemical reactivity and effect of various homologues of the local anesthetic series].

Authors:  J Büchi
Journal:  Pharm Acta Helv       Date:  1967 Aug-Oct

Review 8.  [Chemical constitution, physical chemical properties and the effect of various homologues of the local anesthetic series].

Authors:  X Perlia
Journal:  Pharm Acta Helv       Date:  1967 Aug-Oct

9.  A nerve chamber bioassay of local anesthetic activity.

Authors:  J G Paterson; J T Hamilton
Journal:  Arch Int Pharmacodyn Ther       Date:  1970-02

Review 10.  Principles and practice of Hansch analysis: a guide to structure-activity correlation for the medicinal chemist.

Authors:  M S Tute
Journal:  Adv Drug Res       Date:  1971
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  37 in total

1.  Beta-Adrenoceptor studies. 4. Influence of albumin on in vitro beta-adrenoceptor blocking and antiarrhythmic properties of propranolol, pindolol, practolol and metoprolol.

Authors:  J Zaagsma; L Meems; M Boorsma
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1977-05       Impact factor: 3.000

2.  Influence of isoprenaline and salbutamol on the threshold of electrically induced ventricular fibrillation in anaesthetized guinea pigs.

Authors:  D Hellenbrecht; L Gortner
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1975       Impact factor: 3.000

3.  [3H]-tetracaine binding on rat synaptosomes and sodium channels.

Authors:  M Grima; J Schwartz; M O Spach; J Velly
Journal:  Br J Pharmacol       Date:  1985-09       Impact factor: 8.739

4.  Change of mitochondrial buffering capacity induced by propranolol.

Authors:  J O Järvisalo
Journal:  J Bioenerg       Date:  1975-03

5.  The beta 1- and beta 2-adrenoceptor affinity and beta 1-blocking potency of S- and R-metoprolol.

Authors:  G Wahlund; V Nerme; T Abrahamsson; P O Sjöquist
Journal:  Br J Pharmacol       Date:  1990-03       Impact factor: 8.739

6.  Chronopharmacokinetics of beta-receptor blocking drugs of different lipophilicity (propranolol, metoprolol, sotalol, atenolol) in plasma and tissues after single and multiple dosing in the rat.

Authors:  B Lemmer; H Winkler; T Ohm; M Fink
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1985-07       Impact factor: 3.000

7.  Direct labelling of myocardial beta 1-adrenoceptors. Comparison of binding affinity of 3H-(-)-bisoprolol with its blocking potency.

Authors:  A J Kaumann; H Lemoine
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1985-10       Impact factor: 3.000

8.  beta 2-Adrenoceptors regulate induction of myocardial ornithine decarboxylase in mice in vivo.

Authors:  J G Copeland; D F Larson; W R Roeske; D H Russell; J R Womble
Journal:  Br J Pharmacol       Date:  1982-03       Impact factor: 8.739

9.  Effects of various structurally related beta-adrenoceptor blocking agents on maximum upstroke velocity of action potential in guinea-pig papillary muscles.

Authors:  H Sada; T Ban
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1981-11       Impact factor: 3.000

10.  Quantitative correlation between histamine and 35S release from isolated rat mast cells due to the beta-adrenergic blocking drug Kö 1124.

Authors:  R Nosál; J Pecivová; K Drábiková
Journal:  Agents Actions       Date:  1981-07
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