Literature DB >> 24312840

Synthesis and antimicrobial evaluation of certain novel thiazoles.

Meesaraganda Sreedevi1, Aluru Raghavendra Guru Prasad, Yadati Narasimha Spoorthy, Lakshmana Rao Krishna Rao Ravindranath.   

Abstract

PURPOSE: This article makes an attempt to synthesize certain compounds containing thiazole and imidazole moieties and screen for the antimicrobial properties.
METHODS: The novel compounds synthesized were characterized by elemental analysis, IR and (1)HNMR spectral data. The antimicrobial activity of novel compounds was evaluated by cup plate method.
RESULTS: The compound p-t showed more antibacterial activity than that of the standard. p-hp and p-as showed considerable antibacterial activity. p-t demonstrated higher antifungal activity than that of the standard while p-hp and p-as showed considerable antifungal activity.
CONCLUSION: The antimicrobial activity studies were conducted on certain selected bacteria and fungi. In each case antimicrobial activity of the compounds was compared with that of standards. p-t, p-hp, p-np, p-cp, p-ts and p-as showed considerable antimicrobial activity.

Entities:  

Keywords:  Antimicrobial activity; Characterization; Imidazole moiety; Synthesis; Thiazole moiety

Year:  2013        PMID: 24312840      PMCID: PMC3846066          DOI: 10.5681/apb.2013.037

Source DB:  PubMed          Journal:  Adv Pharm Bull        ISSN: 2228-5881


  8 in total

1.  Synthesis and biological activities of 2-amino-1-arylidenamino imidazoles as orally active anticancer agents.

Authors:  Wen-Tai Li; Der-Ren Hwang; Jen-Shin Song; Ching-Ping Chen; Jiunn-Jye Chuu; Chih-Bo Hu; Heng-Liang Lin; Chen-Lung Huang; Chiung-Yi Huang; Huan-Yi Tseng; Chu-Chung Lin; Tung-Wei Chen; Chi-Hung Lin; Hsin-Sheng Wang; Chien-Chang Shen; Chung-Ming Chang; Yu-Sheng Chao; Chiung-Tong Chen
Journal:  J Med Chem       Date:  2010-03-25       Impact factor: 7.446

2.  Synthesis, characterization and antimicrobial activity of certain novel aryl hydrazone pyrazoline-5-ones containing thiazole moiety.

Authors:  Maliki Reddy Dastagiri Reddy; Aluru Raghavendra Guru Prasad; Yadati Narasimha Spoorthy; Lakshmana Rao Krishna Rao Ravindranath
Journal:  Adv Pharm Bull       Date:  2013-02-07

3.  Design, synthesis, and evaluation of 2-aryl-3-heteroaryl-1,3-thiazolidin-4-ones as anti-HIV agents.

Authors:  Ravindra K Rawal; Rajkamal Tripathi; S B Katti; Christophe Pannecouque; Erik De Clercq
Journal:  Bioorg Med Chem       Date:  2006-12-06       Impact factor: 3.641

4.  Synthesis, antibacterial and potential anti-HIV activity of some novel imidazole analogs.

Authors:  Swastika Ganguly; Vatsal Vijay Vithlani; Anup Kumar Kesharwani; Ritu Kuhu; Lakshmanan Baskar; Papiya Mitramazumder; Ashok Sharon; Abhimanyu Dev
Journal:  Acta Pharm       Date:  2011-06       Impact factor: 2.230

5.  Synthesis, antimicrobial and antiviral evaluation of substituted imidazole derivatives.

Authors:  Deepika Sharma; Balasubramanian Narasimhan; Pradeep Kumar; Vikramjeet Judge; Rakesh Narang; Erik De Clercq; Jan Balzarini
Journal:  Eur J Med Chem       Date:  2008-09-11       Impact factor: 6.514

6.  Synthesis, anti-bacterial and anti-fungal activities of some novel Schiff bases containing 2,4-disubstituted thiazole ring.

Authors:  S K Bharti; G Nath; R Tilak; S K Singh
Journal:  Eur J Med Chem       Date:  2009-11-06       Impact factor: 6.514

7.  Poly(ethylene glycol) (PEG-400) as an alternative reaction solvent for the synthesis of some new 1-(4-(4'-chlorophenyl)-2-thiazolyl)-3-aryl-5-(2-butyl-4-chloro-1H-imidazol-5yl)-2-pyrazolines and their in vitro antimicrobial evaluation.

Authors:  Bhaskar S Dawane; Shankaraiah G Konda; Gajanan G Mandawad; Baseer M Shaikh
Journal:  Eur J Med Chem       Date:  2009-10-14       Impact factor: 6.514

8.  Synthesis and anticancer activity of N-bis(trifluoromethyl)alkyl-N'-thiazolyl and N-bis(trifluoromethyl)alkyl-N'-benzothiazolyl ureas.

Authors:  Elena L Luzina; Anatoliy V Popov
Journal:  Eur J Med Chem       Date:  2009-08-28       Impact factor: 6.514

  8 in total
  1 in total

1.  (Z)-1-[(2E)-3,4-Diphenyl-2,3-di-hydro-1,3-thia-zol-2-yl-idene]-2-[1-(4-hy-droxy-phen-yl)ethyl-idene]hydrazinium bromide including an unknown solvate.

Authors:  Joel T Mague; Shaaban K Mohamed; Mehmet Akkurt; Alaa A Hassan; Mustafa R Albayati
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2014-05-10
  1 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.