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Literature DB >> 21898832

Identification and characterization of inhibitors of the aminoglycoside resistance acetyltransferase Eis from Mycobacterium tuberculosis.

Keith D Green¹, Wenjing Chen, Sylvie Garneau-Tsodikova.

Abstract

Entities: Chemical Disease Species

Mesh：

Substances：

Year: 2011 PMID： 21898832 PMCID： PMC3401626 DOI： 10.1002/cmdc.201100332

Source DB: PubMed Journal: ChemMedChem ISSN： 1860-7179 Impact factor: 3.466

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38 in total

1. Domain-domain interactions in the aminoglycoside antibiotic resistance enzyme AAC(6')-APH(2'').

Authors: David D Boehr; Denis M Daigle; Gerard D Wright
Journal: Biochemistry Date: 2004-08-03 Impact factor: 3.162

2. Molecular modeling studies of N-substituted pyrrole derivatives--potential HIV-1 gp41 inhibitors.

Authors: Cátia Teixeira; Florent Barbault; Joseph Rebehmed; Kun Liu; Lan Xie; Hong Lu; Shibo Jiang; BoTao Fan; François Maurel
Journal: Bioorg Med Chem Date: 2008-01-28 Impact factor: 3.641

3. Design, synthesis, and biological evaluation of N-carboxyphenylpyrrole derivatives as potent HIV fusion inhibitors targeting gp41.

Authors: Kun Liu; Hong Lu; Ling Hou; Zhi Qi; Cátia Teixeira; Florent Barbault; Bo-Tao Fan; Shuwen Liu; Shibo Jiang; Lan Xie
Journal: J Med Chem Date: 2008-12-25 Impact factor: 7.446

4. Combinations of antibiotics and nonantibiotic drugs enhance antimicrobial efficacy.

Authors: Linda Ejim; Maya A Farha; Shannon B Falconer; Jan Wildenhain; Brian K Coombes; Mike Tyers; Eric D Brown; Gerard D Wright
Journal: Nat Chem Biol Date: 2011-04-24 Impact factor: 15.040

5. Subcellular localization of the Iitracellular survival-enhancing Eis protein of Mycobacterium tuberculosis.

Authors: J L Dahl; J Wei; J W Moulder; S Laal; R L Friedman
Journal: Infect Immun Date: 2001-07 Impact factor: 3.441

6. The relA homolog of Mycobacterium smegmatis affects cell appearance, viability, and gene expression.

Authors: John L Dahl; Kriti Arora; Helena I Boshoff; Danelle C Whiteford; Sophia A Pacheco; Olaus J Walsh; Dalia Lau-Bonilla; William B Davis; Anthony G Garza
Journal: J Bacteriol Date: 2005-04 Impact factor: 3.490

7. The kinetic mechanism of AAC3-IV aminoglycoside acetyltransferase from Escherichia coli.

Authors: Maria L B Magalhaes; John S Blanchard
Journal: Biochemistry Date: 2005-12-13 Impact factor: 3.162

8. Effects of altering aminoglycoside structures on bacterial resistance enzyme activities.

Authors: Keith D Green; Wenjing Chen; Sylvie Garneau-Tsodikova
Journal: Antimicrob Agents Chemother Date: 2011-05-02 Impact factor: 5.191

9. Molecular characterization of the eis promoter of Mycobacterium tuberculosis.

Authors: Esteban A Roberts; Amanda Clark; Sarah McBeth; Richard L Friedman
Journal: J Bacteriol Date: 2004-08 Impact factor: 3.490

10. Oral hypoglycemic agents. Discovery and structure-activity relationships of phenacylimidazolium halides.

Authors: S J Dominianni; T T Yen
Journal: J Med Chem Date: 1989-10 Impact factor: 7.446

41 in total

1. 6''-Thioether tobramycin analogues: towards selective targeting of bacterial membranes.

Authors: Ido M Herzog; Keith D Green; Yifat Berkov-Zrihen; Mark Feldman; Roee R Vidavski; Anat Eldar-Boock; Ronit Satchi-Fainaro; Avigdor Eldar; Sylvie Garneau-Tsodikova; Micha Fridman
Journal: Angew Chem Int Ed Engl Date: 2012-04-12 Impact factor: 15.336

2. Aminoglycoside multiacetylating activity of the enhanced intracellular survival protein from Mycobacterium smegmatis and its inhibition.

Authors: Wenjing Chen; Keith D Green; Oleg V Tsodikov; Sylvie Garneau-Tsodikova
Journal: Biochemistry Date: 2012-06-05 Impact factor: 3.162

3. Chemical and structural insights into the regioversatility of the aminoglycoside acetyltransferase Eis.

Authors: Jacob L Houghton; Tapan Biswas; Wenjing Chen; Oleg V Tsodikov; Sylvie Garneau-Tsodikova
Journal: Chembiochem Date: 2013-09-17 Impact factor: 3.164

4. Inhibitors of the aminoglycoside 6'-N-acetyltransferase type Ib [AAC(6')-Ib] identified by in silico molecular docking.

Authors: David L Lin; Tung Tran; Christina Adams; Jamal Y Alam; Steven R Herron; Marcelo E Tolmasky
Journal: Bioorg Med Chem Lett Date: 2013-08-12 Impact factor: 2.823

5. Combating Enhanced Intracellular Survival (Eis)-Mediated Kanamycin Resistance of Mycobacterium tuberculosis by Novel Pyrrolo[1,5-a]pyrazine-Based Eis Inhibitors.

Authors: Atefeh Garzan; Melisa J Willby; Huy X Ngo; Chathurada S Gajadeera; Keith D Green; Selina Y L Holbrook; Caixia Hou; James E Posey; Oleg V Tsodikov; Sylvie Garneau-Tsodikova
Journal: ACS Infect Dis Date: 2017-02-17 Impact factor: 5.084

10. Identification of an Inhibitor of the Aminoglycoside 6'-N-Acetyltransferase type Ib [AAC(6')-Ib] by Glide Molecular Docking.

Authors: Kevin Chiem; Saumya Jani; Brooke Fuentes; David L Lin; Madeline E Rasche; Marcelo E Tolmasky
Journal: Medchemcomm Date: 2015-11-03 Impact factor: 3.597