Literature DB >> 2002466

Benzocycloalkyl amines as novel C-termini for HIV protease inhibitors.

T A Lyle1, C M Wiscount, J P Guare, W J Thompson, P S Anderson, P L Darke, Z A Zugay, E A Emini, W A Schleif, J C Qunitero.   

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Year:  1991        PMID： 2002466     DOI： 10.1021/jm00107a051

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  10 in total

1.  An Efficient Synthesis of Hydroxyethylene Dipeptide Isosteres: The Core Unit of Potent HIV-1 Protease Inhibitors.

Authors:  Arun K Ghosh; Sean P McKee; Wayne J Thompson
Journal:  J Org Chem       Date:  1991-11       Impact factor: 4.354

Review 2.  Antiviral therapy for human immunodeficiency virus infections.

Authors:  E De Clercq
Journal:  Clin Microbiol Rev       Date:  1995-04       Impact factor: 26.132

3.  Highly Enantioselective Aldol Reaction: Development of a New Chiral Auxiliary from cis-1-Amino-2-hydroxyindan.

Authors:  Arun K Ghosh; Tien T Duong; Sean P McKee
Journal:  J Chem Soc Chem Commun       Date:  1992

4.  STEREOCONTROLLED SYNTHESIS OF HIV-l PROTEASE INHIBITORS WITH C2-AXIS OF SYMMETRY.

Authors:  Arun K Ghosh; Sean P McKee; Wayne J Thompson
Journal:  Tetrahedron Lett       Date:  2001-03-26       Impact factor: 2.415

5.  cis-1-Aminoindan-2-ol in Asymmetric Syntheses.

Authors:  Arun K Ghosh; Steve Fidanze; Chris H Senanayake
Journal:  Synthesis (Stuttg)       Date:  1998-07       Impact factor: 3.157

6.  A Facile and Enantiospecific Synthesis of 2(S)- and 2(R)-[1'(S)-Azido-2-phenylethyl]oxirane.

Authors:  Arun K Ghosh; Sean P McKee; Hee Yoon Lee; Wayne J Thompson
Journal:  J Chem Soc Chem Commun       Date:  1992

7.  Pyrrolinone-based peptidomimetics. "Let the enzyme or receptor be the judge".

Authors:  Amos B Smith; Adam K Charnley; Ralph Hirschmann
Journal:  Acc Chem Res       Date:  2010-12-22       Impact factor: 22.384

8.  Calculation of solvation and binding free energy differences between VX-478 and its analogs by free energy perturbation and AMSOL methods.

Authors:  B G Rao; E E Kim; M A Murcko
Journal:  J Comput Aided Mol Des       Date:  1996-02       Impact factor: 3.686

9.  L-735,524: an orally bioavailable human immunodeficiency virus type 1 protease inhibitor.

Authors:  J P Vacca; B D Dorsey; W A Schleif; R B Levin; S L McDaniel; P L Darke; J Zugay; J C Quintero; O M Blahy; E Roth
Journal:  Proc Natl Acad Sci U S A       Date:  1994-04-26       Impact factor: 11.205

Review 10.  Viral proteases as targets for chemotherapeutic intervention.

Authors:  C U Hellen; E Wimmer
Journal:  Curr Opin Biotechnol       Date:  1992-12       Impact factor: 9.740
  10 in total

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