Literature DB >> 30393403

cis-1-Aminoindan-2-ol in Asymmetric Syntheses.

Arun K Ghosh1, Steve Fidanze1, Chris H Senanayake2.   

Abstract

A review on cis-1-aminoindan-2-ol derived asymmetric syntheses is described.

Entities:  

Keywords:  1-aminoindan-2-ol; asymmetric synthesis; inhibitor; protease

Year:  1998        PMID: 30393403      PMCID: PMC6214626          DOI: 10.1055/s-1998-2092

Source DB:  PubMed          Journal:  Synthesis (Stuttg)        ISSN: 0039-7881            Impact factor:   3.157


  27 in total

1.  Toward the Development of a General Chiral Auxiliary. 5. High Diastereofacial Selectivity in Cycloadditions with Trienol Silyl Ethers: An Application to an Enantioselective Synthesis of (-)-Cassioside.

Authors:  Robert K Boeckman; Yugang Liu
Journal:  J Org Chem       Date:  1996-11-15       Impact factor: 4.354

2.  Highly Enantioselective Aldol Reaction: Development of a New Chiral Auxiliary from cis-1-Amino-2-hydroxyindan.

Authors:  Arun K Ghosh; Tien T Duong; Sean P McKee
Journal:  J Chem Soc Chem Commun       Date:  1992

3.  SYNTHESIS AND OPTICAL RESOLUTION OF HIGH AFFINITY P2-LIGANDS FOR HIV-1 PROTEASE INHIBITORS.

Authors:  Arun K Ghosh; Yan Chen
Journal:  Tetrahedron Lett       Date:  2000-06-14       Impact factor: 2.415

4.  Control of Metal-Catalyzed Reactions by Organic Ligands: From Corrinoid and Porphinoid Metal Complexes to Tailor-Made Catalysts for Asymmetric Synthesis.

Authors:  Andreas Pfaltz
Journal:  Chimia (Aarau)       Date:  2006-06-01       Impact factor: 1.509

5.  HIV-1 protease inhibitors based on hydroxyethylene dipeptide isosteres: an investigation into the role of the P1' side chain on structure-activity.

Authors:  S D Young; L S Payne; W J Thompson; N Gaffin; T A Lyle; S F Britcher; S L Graham; T H Schultz; A A Deana; P L Darke
Journal:  J Med Chem       Date:  1992-05-15       Impact factor: 7.446

6.  Potent HIV-1 Protease Inhibitors: Stereoselective Synthesis of a Dipeptide Mimic.

Authors:  Arun K Ghosh; Sean P McKee; Wayne J Thompson; Paul L Darke; Joan C Zugay
Journal:  J Org Chem       Date:  1993-02       Impact factor: 4.354

7.  Rational design of peptide-based HIV proteinase inhibitors.

Authors:  N A Roberts; J A Martin; D Kinchington; A V Broadhurst; J C Craig; I B Duncan; S A Galpin; B K Handa; J Kay; A Kröhn
Journal:  Science       Date:  1990-04-20       Impact factor: 47.728

8.  Inhibitors of human immunodeficiency virus type 1 protease containing 2-aminobenzyl-substituted 4-amino-3-hydroxy-5-phenylpentanoic acid: synthesis, activity, and oral bioavailability.

Authors:  P Lehr; A Billich; B Charpiot; P Ettmayer; D Scholz; B Rosenwirth; H Gstach
Journal:  J Med Chem       Date:  1996-05-10       Impact factor: 7.446

9.  L-735,524: the design of a potent and orally bioavailable HIV protease inhibitor.

Authors:  B D Dorsey; R B Levin; S L McDaniel; J P Vacca; J P Guare; P L Darke; J A Zugay; E A Emini; W A Schleif; J C Quintero
Journal:  J Med Chem       Date:  1994-10-14       Impact factor: 7.446

10.  SYNTHETIC STUDIES OF ANTITUMOR MACROLIDE LAULIMALIDE: ENANTIOSELECTIVE SYNTHESIS OF THE C3-C14 SEGMENT BY A CATALYTIC HETERO DIELS-ALDER STRATEGY.

Authors:  Arun K Ghosh; Packiarajan Mathivanan; John Cappiello
Journal:  Tetrahedron Lett       Date:  2000-03-17       Impact factor: 2.415

View more
  1 in total

1.  Asymmetric Syntheses of Potent Antitumor Macrolides Cryptophycin B and Arenastatin A.

Authors:  Arun K Ghosh; A Bischoff
Journal:  European J Org Chem       Date:  2004-04-27
  1 in total

北京卡尤迪生物科技股份有限公司 © 2022-2023.