Literature DB >> 16650998

Synthesis of 7-chloro-5-trifluoromethyl/7-fluoro/7-trifluoromethyl-4H-1,4-benzothiazines as antimicrobial agents.

Bhawani Singh Rathore1, M Kumar.   

Abstract

7-Chloro-5-trifluoromethyl/7-fluoro/7-trifluoromethyl-4H-1,4-benzothiazines have been synthesized by 2-amino-5-fluoro/5-trifluoromethyl/5-chloro-3-trifluoromethyl benzenethiols condensed with beta-diketone/beta-ketoesters in the presence of DMSO involving oxidative cyclization. Pharmacological activities have also been included.

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Year:  2006        PMID： 16650998     DOI： 10.1016/j.bmc.2006.04.009

Source DB:  PubMed          Journal:  Bioorg Med Chem        ISSN： 0968-0896            Impact factor:   3.641


  12 in total

1.  Base catalyzed multicomponent synthesis of spiroheterocycles with fused heterosystems.

Authors:  Anand Kumar Arya; Mahendra Kumar
Journal:  Mol Divers       Date:  2011-03-20       Impact factor: 2.943

2.  Crystal structure of (E)-2-benzyl-idene-4-[(3-phenyl-4,5-di-hydro-isoxazol-5-yl)meth-yl]-2H-benzo[b][1,4]thia-zin-3(4H)-one.

Authors:  Nada Kheira Sebbar; Mohamed Ellouz; El Mokhtar Essassi; Mohamed Saadi; Lahcen El Ammari
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2015-05-23

3.  Diversity oriented one-pot three-component sequential synthesis of annulated benzothiazoloquinazolines.

Authors:  Mahendra Kumar; Kailash Sharma; Dinesh Kumar Sharma
Journal:  Org Med Chem Lett       Date:  2012-03-02

4.  4-[(1-Benzyl-1H-1,2,3-triazol-4-yl)meth-yl]-2H-1,4-benzo-thia-zin-3(4H)-one.

Authors:  Nada Kheira Sebbar; Abdelfettah Zerzouf; El Mokhtar Essassi; Mohamed Saadi; Lahcen El Ammari
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2014-01-18

5.  Ethyl 2-{5-[(3-oxo-3,4-di-hydro-2H-1,4-benzo-thia-zin-4-yl)meth-yl]-1H-1,2,3-triazol-1-yl}acetate.

Authors:  Nada Kheira Sebbar; Abdelfettah Zerzouf; El Mokhtar Essassi; Mohamed Saadi; Lahcen El Ammari
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2014-01-08

6.  (2Z)-2-Benzyl-idene-4-(prop-2-yn-1-yl)-2H-1,4-benzo-thia-zin-3(4H)-one.

Authors:  Nada Kheira Sebbar; Abdelfettah Zerzouf; El Mokhtar Essassi; Mohamed Saadi; Lahcen El Ammari
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2014-04-26

7.  Antinociceptive properties of new coumarin derivatives bearing substituted 3,4-dihydro-2H-benzothiazines.

Authors:  Masoumeh Alipour; Mehdi Khoobi; Saeed Emami; Saeed Fallah-Benakohal; Seyedeh Farnaz Ghasemi-Niri; Mohammad Abdollahi; Alireza Foroumadi; Abbas Shafiee
Journal:  Daru       Date:  2014-01-07       Impact factor: 3.117

8.  Synthesis and antibacterial activity of new 1,2,3-triazolylmethyl-2H-1,4-benzothiazin-3(4H)-one derivatives.

Authors:  Mohamed Ellouz; Nada Kheira Sebbar; Ismail Fichtali; Younes Ouzidan; Zakaria Mennane; Reda Charof; Joel T Mague; Martine Urrutigoïty; El Mokhtar Essassi
Journal:  Chem Cent J       Date:  2018-11-29       Impact factor: 4.215

9.  Crystal structure, Hirshfeld surface analysis and inter-action energy and DFT studies of 3-{(2Z)-2-[(2,4-di-chloro-phen-yl)methyl-idene]-3-oxo-3,4-di-hydro-2H-1,4-benzo-thia-zin-4-yl}propane-nitrile.

Authors:  Nada Kheira Sebbar; Brahim Hni; Tuncer Hökelek; Abdelhakim Jaouhar; Mohamed Labd Taha; Joel T Mague; El Mokhtar Essassi
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2019-05-03

10.  (2Z)-2-Benzyl-idene-4-n-butyl-3,4-di-hydro-2H-1,4-benzo-thia-zin-3-one.

Authors:  Nada Kheira Sebbar; Mohammed El Fal; El Mokhtar Essassi; Mohamed Saadi; Lahcen El Ammari
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2014-05-21
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