Literature DB >> 15203133

Biological evaluation of substituted quinolines.

Xavier Franck1, Alain Fournet, Eric Prina, Renaud Mahieux, Reynald Hocquemiller, Bruno Figadère.   

Abstract

Several quinolines were synthesized and evaluated in vitro against several parasites (Trypanosoma brucei, T. cruzi, Leishmania infantum, L. amazonensis, Plasmodium falciparum). Then, they were evaluated in vitro (at 10 microM), against HTLV-1 transformed cells. A few of them displayed interesting activities, comparable to the reference drugs.

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Year:  2004        PMID： 15203133     DOI： 10.1016/j.bmcl.2004.05.026

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  10 in total

1.  Efficacy of orally administered 2-substituted quinolines in experimental murine cutaneous and visceral leishmaniases.

Authors:  Hector Nakayama; Philippe M Loiseau; Christian Bories; Susana Torres de Ortiz; Alicia Schinini; Elsa Serna; Antonieta Rojas de Arias; Mohamed A Fakhfakh; Xavier Franck; Bruno Figadère; Reynald Hocquemiller; Alain Fournet
Journal:  Antimicrob Agents Chemother       Date:  2005-12       Impact factor: 5.191

2.  Chemicals possessing a neurotrophin-like activity on dopaminergic neurons in primary culture.

Authors:  Fanny Schmidt; Pierre Champy; Blandine Séon-Méniel; Xavier Franck; Rita Raisman-Vozari; Bruno Figadère
Journal:  PLoS One       Date:  2009-07-10       Impact factor: 3.240

3.  Quinoline: A versatile heterocyclic.

Authors:  Akranth Marella; Om Prakash Tanwar; Rikta Saha; Mohammad Rahmat Ali; Sandeep Srivastava; Mymoona Akhter; Mohammad Shaquiquzzaman; Mohammad Mumtaz Alam
Journal:  Saudi Pharm J       Date:  2012-03-29       Impact factor: 4.330

4.  Oxyrane derivative of alpha-lapachone is potent growth inhibitor of Trypanosoma cruzi epimastigote forms.

Authors:  Alessandra Jorqueira; Robson M Gouvêa; Vitor F Ferreira; Milton N da Silva; Maria C B V de Souza; Aline A Zuma; Danielle F B Cavalcanti; Humberto P Araújo; Dilvani O Santos; Saulo C Bourguignon
Journal:  Parasitol Res       Date:  2006-04-05       Impact factor: 2.383

5.  8-Nitro-quinoline.

Authors:  Liang Xu; Bao-Li Xu; Shu-Jun Lu; Bing Wang; Ting-Guo Kang
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2011-03-23

6.  4-Chloro-6,7-dimeth-oxy-quinoline.

Authors:  Min Wu
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2011-10-22

7.  2-(4-Methyl-phen-yl)-1-phenyl-sulfonyl-3-nitro-1,2-dihydro-quinoline.

Authors:  J Kanchanadevi; G Anbalagan; V Saravanan; A K Mohanakrishnan; V Manivannan
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2011-08-02

8.  Quantitative Structure-Activity Relationships for Structurally Diverse Chemotypes Having Anti-Trypanosoma cruzi Activity.

Authors:  Anacleto S de Souza; Leonardo L G Ferreira; Aldo S de Oliveira; Adriano D Andricopulo
Journal:  Int J Mol Sci       Date:  2019-06-08       Impact factor: 5.923

Review 9.  The Potential of 2-Substituted Quinolines as Antileishmanial Drug Candidates.

Authors:  Philippe M Loiseau; Kaluvu Balaraman; Gillian Barratt; Sébastien Pomel; Rémy Durand; Frédéric Frézard; Bruno Figadère
Journal:  Molecules       Date:  2022-04-02       Impact factor: 4.411

10.  Intestinal cestodes of chicken are effectively killed by quinoline-rich extract of Spilanthes acmella.

Authors:  Pawi Bawitlung Lalthanpuii; Kholhring Lalchhandama
Journal:  Vet World       Date:  2020-04-30
  10 in total

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