Literature DB >> 8464047

Cyclic sulfolanes as novel and high affinity P2 ligands for HIV-1 protease inhibitors.

A K Ghosh1, W J Thompson, H Y Lee, S P McKee, P M Munson, T T Duong, P L Darke, J A Zugay, E A Emini, W A Schleif.   

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Year:  1993        PMID： 8464047     DOI： 10.1021/jm00059a019

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  6 in total

Review 1.  Antiviral therapy for human immunodeficiency virus infections.

Authors:  E De Clercq
Journal:  Clin Microbiol Rev       Date:  1995-04       Impact factor: 26.132

2.  Asymmetric Aldol Route to Hydroxyethylamine Isostere: Stereoselective Synthesis of the Core Unit of Saquinavir.

Authors:  Arun K Ghosh; Khaja Azhar Hussain; Steve Fidanze
Journal:  J Org Chem       Date:  1997-08-22       Impact factor: 4.354

3.  Chiral Auxiliary Mediated Conjugate Reduction and Asymmetric Protonation: Synthesis of High Affinity Ligands for HIV Protease Inhibitors.

Authors:  Arun K Ghosh; Wenming Liu
Journal:  J Org Chem       Date:  1995-09-01       Impact factor: 4.354

4.  Efficient synthesis of 3-sulfolenes from allylic alcohols and 1,3-dienes enabled by sodium metabisulfite as a sulfur dioxide equivalent.

Authors:  Hang T Dang; Vu T Nguyen; Viet D Nguyen; Hadi D Arman; Oleg V Larionov
Journal:  Org Biomol Chem       Date:  2018-05-15       Impact factor: 3.876

5.  Design, synthesis, and X-ray studies of potent HIV-1 protease inhibitors incorporating aminothiochromane and aminotetrahydronaphthalene carboxamide derivatives as the P2 ligands.

Authors:  Arun K Ghosh; Ravindra D Jadhav; Hannah Simpson; Satish Kovela; Heather Osswald; Johnson Agniswamy; Yuan-Fang Wang; Shin-Ichiro Hattori; Irene T Weber; Hiroaki Mitsuya
Journal:  Eur J Med Chem       Date:  2018-09-18       Impact factor: 6.514

6.  CYCLIC SULFONE-3-CARBOXAMIDES AS NOVEL P2-LIGANDS FOR Ro 31-8959 BASED HIV-1 PROTEASE INHIBITORS.

Authors:  Arun K Ghosh; Wayne J Thompson; Peter M Munson; Wenming Liut; Joel R Huff
Journal:  Bioorg Med Chem Lett       Date:  2000-03-29       Impact factor: 2.823
  6 in total

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