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82 in total

1. The 2011 E. B. Hershberg award for important discoveries in medicinally active substances: (1S,3S)-3-amino-4-difluoromethylenyl-1-cyclopentanoic acid (CPP-115), a GABA aminotransferase inactivator and new treatment for drug addiction and infantile spasms.

Authors: Richard B Silverman
Journal: J Med Chem Date: 2012-01-10 Impact factor: 7.446

2. (1S, 3S)-3-amino-4-difluoromethylenyl-1-cyclopentanoic acid (CPP-115), a potent γ-aminobutyric acid aminotransferase inactivator for the treatment of cocaine addiction.

Authors: Yue Pan; Madina R Gerasimov; Trine Kvist; Petrine Wellendorph; Karsten K Madsen; Elena Pera; Hyunbeom Lee; Arne Schousboe; Mary Chebib; Hans Bräuner-Osborne; Cheryl M Craft; Jonathan D Brodie; Wynne K Schiffer; Stephen L Dewey; Steven R Miller; Richard B Silverman
Journal: J Med Chem Date: 2011-12-30 Impact factor: 7.446

3. An amino acid position at crossroads of evolution of protein function: antibiotic sensor domain of BlaR1 protein from Staphylococcus aureus versus clasS D β-lactamases.

Authors: Malika Kumarasiri; Leticia I Llarrull; Oleg Borbulevych; Jennifer Fishovitz; Elena Lastochkin; Brian M Baker; Shahriar Mobashery
Journal: J Biol Chem Date: 2012-01-18 Impact factor: 5.157

4. Structure-Based Engineering of Irreversible Inhibitors against Histone Lysine Demethylase KDM5A.

Authors: John R Horton; Clayton B Woodcock; Qin Chen; Xu Liu; Xing Zhang; John Shanks; Ganesha Rai; Bryan T Mott; Daniel J Jansen; Stephen C Kales; Mark J Henderson; Matthew Cyr; Katherine Pohida; Xin Hu; Pranav Shah; Xin Xu; Ajit Jadhav; David J Maloney; Matthew D Hall; Anton Simeonov; Haian Fu; Paula M Vertino; Xiaodong Cheng
Journal: J Med Chem Date: 2018-11-15 Impact factor: 7.446

5. Examination of the new alpha-(2'Z-fluoro)vinyl trigger with lysine decarboxylase: the absolute stereochemistry dictates the reaction course.

Authors: Kannan R Karukurichi; Roberto de la Salud-Bea; Wan Jin Jahng; David B Berkowitz
Journal: J Am Chem Soc Date: 2007-01-17 Impact factor: 15.419

Review 6. LSD1 and the chemistry of histone demethylation.

Authors: Jeffrey C Culhane; Philip A Cole
Journal: Curr Opin Chem Biol Date: 2007-09-11 Impact factor: 8.822

7. Pharmacological inhibition of ALDH1A in mice decreases all-trans retinoic acid concentrations in a tissue specific manner.

Authors: Samuel L M Arnold; Travis Kent; Cathryn A Hogarth; Michael D Griswold; John K Amory; Nina Isoherranen
Journal: Biochem Pharmacol Date: 2015-03-09 Impact factor: 5.858

8. An antibiotic-resistance enzyme from a deep-sea bacterium.

Authors: Marta Toth; Clyde Smith; Hilary Frase; Shahriar Mobashery; Sergei Vakulenko
Journal: J Am Chem Soc Date: 2010-01-20 Impact factor: 15.419

9. The pneumotoxin 3-methylindole is a substrate and a mechanism-based inactivator of CYP2A13, a human cytochrome P450 enzyme preferentially expressed in the respiratory tract.

Authors: Jaime D'Agostino; Xiaoliang Zhuo; Mohammad Shadid; Daniel G Morgan; Xiuling Zhang; W Griffith Humphreys; Yue-Zhong Shu; Garold S Yost; Xinxin Ding
Journal: Drug Metab Dispos Date: 2009-07-16 Impact factor: 3.922

10. Understanding the roles of strictly conserved tryptophan residues in O2 producing chlorite dismutases.

Authors: Beatrice Blanc; Kenton R Rodgers; Gudrun S Lukat-Rodgers; Jennifer L DuBois
Journal: Dalton Trans Date: 2012-12-17 Impact factor: 4.390