Literature DB >> 35983270

Call for Manuscripts for ACS Pharmacology & Translational Science Review Series on Recommended Tool Compounds.

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Abstract

Entities:  

Year:  2022        PMID: 35983270      PMCID: PMC9379939          DOI: 10.1021/acsptsci.2c00135

Source DB:  PubMed          Journal:  ACS Pharmacol Transl Sci        ISSN: 2575-9108


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  9 in total

1.  The art of the chemical probe.

Authors:  Stephen V Frye
Journal:  Nat Chem Biol       Date:  2010-03       Impact factor: 15.040

2.  Evidence-Based and Quantitative Prioritization of Tool Compounds in Phenotypic Drug Discovery.

Authors:  Yuan Wang; Allen Cornett; Fred J King; Yi Mao; Florian Nigsch; C Gregory Paris; Gregory McAllister; Jeremy L Jenkins
Journal:  Cell Chem Biol       Date:  2016-07-14       Impact factor: 8.116

3.  The promise and peril of chemical probes.

Authors:  Cheryl H Arrowsmith; James E Audia; Christopher Austin; Jonathan Baell; Jonathan Bennett; Julian Blagg; Chas Bountra; Paul E Brennan; Peter J Brown; Mark E Bunnage; Carolyn Buser-Doepner; Robert M Campbell; Adrian J Carter; Philip Cohen; Robert A Copeland; Ben Cravatt; Jayme L Dahlin; Dashyant Dhanak; Aled M Edwards; Mathias Frederiksen; Stephen V Frye; Nathanael Gray; Charles E Grimshaw; David Hepworth; Trevor Howe; Kilian V M Huber; Jian Jin; Stefan Knapp; Joanne D Kotz; Ryan G Kruger; Derek Lowe; Mary M Mader; Brian Marsden; Anke Mueller-Fahrnow; Susanne Müller; Ronan C O'Hagan; John P Overington; Dafydd R Owen; Saul H Rosenberg; Bryan Roth; Brian Roth; Ruth Ross; Matthieu Schapira; Stuart L Schreiber; Brian Shoichet; Michael Sundström; Giulio Superti-Furga; Jack Taunton; Leticia Toledo-Sherman; Chris Walpole; Michael A Walters; Timothy M Willson; Paul Workman; Robert N Young; William J Zuercher
Journal:  Nat Chem Biol       Date:  2015-08       Impact factor: 15.040

Review 4.  Chemical Probes for Understudied Kinases: Challenges and Opportunities.

Authors:  Ricardo A M Serafim; Jonathan M Elkins; William J Zuercher; Stefan A Laufer; Matthias Gehringer
Journal:  J Med Chem       Date:  2021-09-03       Impact factor: 7.446

Review 5.  Choose and Use Your Chemical Probe Wisely to Explore Cancer Biology.

Authors:  Julian Blagg; Paul Workman
Journal:  Cancer Cell       Date:  2017-07-10       Impact factor: 31.743

6.  Report and Application of a Tool Compound Data Set.

Authors:  Kyle V Butler; Ian A MacDonald; Nathaniel A Hathaway; Jian Jin
Journal:  J Chem Inf Model       Date:  2017-11-02       Impact factor: 4.956

7.  Donated chemical probes for open science.

Authors:  Susanne Müller; Suzanne Ackloo; Cheryl H Arrowsmith; Marcus Bauser; Jeremy L Baryza; Julian Blagg; Jark Böttcher; Chas Bountra; Peter J Brown; Mark E Bunnage; Adrian J Carter; David Damerell; Volker Dötsch; David H Drewry; Aled M Edwards; James Edwards; Jon M Elkins; Christian Fischer; Stephen V Frye; Andreas Gollner; Charles E Grimshaw; Adriaan IJzerman; Thomas Hanke; Ingo V Hartung; Steve Hitchcock; Trevor Howe; Terry V Hughes; Stefan Laufer; Volkhart Mj Li; Spiros Liras; Brian D Marsden; Hisanori Matsui; John Mathias; Ronan C O'Hagan; Dafydd R Owen; Vineet Pande; Daniel Rauh; Saul H Rosenberg; Bryan L Roth; Natalie S Schneider; Cora Scholten; Kumar Singh Saikatendu; Anton Simeonov; Masayuki Takizawa; Chris Tse; Paul R Thompson; Daniel K Treiber; Amélia Yi Viana; Carrow I Wells; Timothy M Willson; William J Zuercher; Stefan Knapp; Anke Mueller-Fahrnow
Journal:  Elife       Date:  2018-04-20       Impact factor: 8.140

8.  A chemical toolbox for the study of bromodomains and epigenetic signaling.

Authors:  Qin Wu; David Heidenreich; Stanley Zhou; Suzanne Ackloo; Andreas Krämer; Kiran Nakka; Evelyne Lima-Fernandes; Genevieve Deblois; Shili Duan; Ravi N Vellanki; Fengling Li; Masoud Vedadi; Jeffrey Dilworth; Mathieu Lupien; Paul E Brennan; Cheryl H Arrowsmith; Susanne Müller; Oleg Fedorov; Panagis Filippakopoulos; Stefan Knapp
Journal:  Nat Commun       Date:  2019-04-23       Impact factor: 14.919

Review 9.  Recommended tool compounds and drugs for blocking P2X and P2Y receptors.

Authors:  Christa E Müller; Vigneshwaran Namasivayam
Journal:  Purinergic Signal       Date:  2021-09-02       Impact factor: 3.765

  9 in total

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