Literature DB >> 33862496

Poly (ADP-ribose) polymerase inhibitors in solid tumours: Systematic review and meta-analysis.

Francesco Schettini1, Fabiola Giudici2, Ottavia Bernocchi3, Marianna Sirico4, Silvia P Corona3, Mario Giuliano5, Mariavittoria Locci6, Ida Paris7, Giovanni Scambia8, Sabino De Placido5, Pasquale Rescigno9, Aleix Prat10, Giuseppe Curigliano11, Daniele Generali12.   

Abstract

BACKGROUND: Poly (ADP-ribose) polymerase-inhibitors (PARPis) showed antitumour activity in BRCA1/2-mutated cancers, with more heterogeneous outcomes in tumours harbouring mutations that impair other genes involved in the DNA homologous recombination repair (HRR) or wild-type (wt).
METHODS: We conducted a systematic review and meta-analysis to better assess the role of PARPis in the treatment of metastatic solid tumours, with and without BRCA1/2 mutations. The primary end-point was progression-free survival (PFS). The secondary end-points were overall response rate (ORR) and overall survival (OS). A random-effects model was applied.
RESULTS: Twenty-nine studies (8,839 patients) were included. PFS was significantly improved (hazard ratio [HR]: 0.59, 95% confidence interval [CI]: 0.51-0.68, p < 0.001), without being affected by BRCA mutational status (p = 0.65). Significant subgroup differences were observed with regard to the tumour site (p = 0.001), line of therapy (p = 0.002), control arm (p < 0.001), type of PARPi (p < 0.001) and trials' phase (p = 0.006). PARPis were associated with ORR (relative risk: 1.35, 95% CI: 1.16-1.56, p < 0.001), with significant subgroup differences observed with regard to treatment line (p = 0.03), control arm (p = 0.04) and PARPis (p < 0.001) and independent of mutational status (p = 0.44), tumour site (p = 0.86) and trials' phase (p = 0.09). OS was significantly improved by PARPis (HR: 0.86, 95% CI: 0.80-0.92, p < 0.001), regardless of mutational status (p = 0.57), tumour site (p = 0.82), treatment line (p = 0.22), control arm (p = 0.21), PARPis (p = 0.30) and trials' phase (p = 0.26). Finally, an exploratory subgroup analysis showed a significant PFS improvement (HR: 0.51, 95% CI: 0.43-0.60, p < 0.001) with PARPis in BRCA-wt/HRR-deficient tumours.
CONCLUSION: Our results confirm the efficacy of already approved PARPi-based treatments in BRCA1/2-mutant solid tumours, support their role also in BRCA-independent HRR-deficient tumours and suggest a potentially broader efficacy in some wt tumours, perhaps with appropriate therapeutic partners. Prospective studies are warranted.
Copyright © 2021 Elsevier Ltd. All rights reserved.

Entities:  

Keywords:  Breast cancer; Meta-analysis; Niraparib; Olaparib; Ovarian cancer; PARP inhibitor; Prostate cancer; Rucaparib; Talazoparib; Veliparib

Year:  2021        PMID: 33862496     DOI: 10.1016/j.ejca.2021.02.035

Source DB:  PubMed          Journal:  Eur J Cancer        ISSN: 0959-8049            Impact factor:   9.162


  7 in total

Review 1.  Addressing the routine failure to clinically identify monogenic cases of common disease.

Authors:  Michael F Murray; Muin J Khoury; Noura S Abul-Husn
Journal:  Genome Med       Date:  2022-06-07       Impact factor: 15.266

2.  Care of men with cancer-predisposing BRCA variants.

Authors:  Rachel Horton; Paul Pharoah; Judith Hayward; Anneke Lucassen
Journal:  BMJ       Date:  2021-10-14

Review 3.  Updated Neoadjuvant Treatment Landscape for Early Triple Negative Breast Cancer: Immunotherapy, Potential Predictive Biomarkers, and Novel Agents.

Authors:  Giovanna Garufi; Luisa Carbognin; Francesco Schettini; Elia Seguí; Alba Di Leone; Antonio Franco; Ida Paris; Giovanni Scambia; Giampaolo Tortora; Alessandra Fabi
Journal:  Cancers (Basel)       Date:  2022-08-23       Impact factor: 6.575

4.  Clinical, Radiometabolic and Immunologic Effects of Olaparib in Locally Advanced Triple Negative Breast Cancer: The OLTRE Window of Opportunity Trial.

Authors:  Francesco Schettini; Silvia Paola Corona; Fabiola Giudici; Carla Strina; Marianna Sirico; Ottavia Bernocchi; Manuela Milani; Nicoletta Ziglioli; Sergio Aguggini; Carlo Azzini; Giuseppina Barbieri; Valeria Cervoni; Maria Rosa Cappelletti; Alfredo Molteni; Maria Chiara Lazzari; Giuseppina Ferrero; Marco Ungari; Elena Marasco; Alice Bruson; Luciano Xumerle; Elisa Zago; Davide Cerra; Marco Loddo; Gareth H Williams; Ida Paris; Giovanni Scambia; Daniele Generali
Journal:  Front Oncol       Date:  2021-06-28       Impact factor: 6.244

Review 5.  OB-Folds and Genome Maintenance: Targeting Protein-DNA Interactions for Cancer Therapy.

Authors:  Sui Par; Sofia Vaides; Pamela S VanderVere-Carozza; Katherine S Pawelczak; Jason Stewart; John J Turchi
Journal:  Cancers (Basel)       Date:  2021-07-03       Impact factor: 6.639

6.  Redefining and expanding the sphere of influence of BRCA in breast and colorectal cancers and beyond.

Authors:  Emil Lou
Journal:  Oncotarget       Date:  2022-01-14

Review 7.  Anthracyclines Strike Back: Rediscovering Non-Pegylated Liposomal Doxorubicin in Current Therapeutic Scenarios of Breast Cancer.

Authors:  Francesco Schettini; Mario Giuliano; Matteo Lambertini; Rupert Bartsch; David James Pinato; Concetta Elisa Onesti; Nadia Harbeck; Diana Lüftner; Sylvie Rottey; Peter A van Dam; Khalil Zaman; Giorgio Mustacchi; Joseph Gligorov; Ahmad Awada; Mario Campone; Hans Wildiers; Alessandra Gennari; Vivianne C G Tjan-Heijnen; Javier Cortes; Mariavittoria Locci; Ida Paris; Lucia Del Mastro; Sabino De Placido; Miguel Martín; Guy Jerusalem; Sergio Venturini; Giuseppe Curigliano; Daniele Generali
Journal:  Cancers (Basel)       Date:  2021-09-01       Impact factor: 6.639

  7 in total

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