Literature DB >> 33527479

CDK 4/6 inhibitors are associated with a high incidence of thrombotic events in women with breast cancer in real-world practice.

Malinda T West1, Claire E Smith1, Andy Kaempf2, Tia C L Kohs3, Ramin Amirsoltani4, Jessica Ribkoff4, Josh Lee Choung5, Alison Palumbo5, Zahi Mitri1, Joseph J Shatzel1,3.   

Abstract

PURPOSE: Cyclin-dependent kinase (CDK) 4/6 inhibitors are integral treatment for advanced hormone receptor positive breast cancer; however, venous thromboembolic events (VTE) occurred in 1%-5% of clinical trial patients. Thrombosis rates in the real-world setting remain unclear. We aimed to define the rate of thromboembolic events, risk factors for thrombosis on CDK 4/6 inhibitors and evaluate the Khorana VTE risk score as a predictive tool for VTE in patients on CDK 4/6 therapy.
METHODS: Multicenter retrospective analysis of adult breast cancer patients prescribed palbociclib, ribociclib, or abemaciclib. The primary endpoint was thrombosis during treatment or within 30 days of CDK inhibitor discontinuation. Cox regression was used to model time-to-thrombosis, starting from a patient's initiation of CDK 4/6 therapy. The extended Kaplan-Meier method and Cox modeling were used to assess the effect of time-varying thrombosis status on overall survival.
RESULTS: Two hundred and sixty-six patients were included (89% on palbociclib, 14% on abemaciclib, 7% on ribociclib). Twenty-nine thrombotic events occurred in 26 (9.8%) women. Of these events, 72% were venous and 34% were arterial. The 1-year incidence of thrombosis was 10.4% overall, 10.9% on palbociclib, 8.3% on ribociclib, and 4.8% on abemaciclib. Hemoglobin less than 10 g/dL was a statistically significant predictor of thrombosis (HR 3.53, P: .014). Khorana score ranged from 0-3, with the majority between 0 and 1 and was not predictive of VTE. Thrombosis was associated with reduced overall survival (HR 1.28, P: .128, median 7.3 months) compared to not having a CDK-associated clot (median 35.7 months). DISCUSSION: VTE in our analysis is higher than reported in clinical trials and arterial thrombosis comprised over one-third of events. The highest incidence was with palbociclib, followed by ribociclib. Khorana score did not predict VTE risk. Larger, real-world studies are needed. The role for prophylactic anticoagulation is yet to be defined in this patient population.
© 2021 John Wiley & Sons A/S. Published by John Wiley & Sons Ltd.

Entities:  

Keywords:  CDK inhibitor; arterial; breast cancer; thrombosis; venous

Mesh:

Substances:

Year:  2021        PMID: 33527479      PMCID: PMC8087188          DOI: 10.1111/ejh.13590

Source DB:  PubMed          Journal:  Eur J Haematol        ISSN: 0902-4441            Impact factor:   2.997


  26 in total

1.  Apixaban to Prevent Venous Thromboembolism in Patients with Cancer.

Authors:  Marc Carrier; Karim Abou-Nassar; Ranjeeta Mallick; Vicky Tagalakis; Sudeep Shivakumar; Ariah Schattner; Philip Kuruvilla; Danny Hill; Silvana Spadafora; Katerine Marquis; Mateya Trinkaus; Anna Tomiak; Agnes Y Y Lee; Peter L Gross; Alejandro Lazo-Langner; Robert El-Maraghi; Glenwood Goss; Gregoire Le Gal; David Stewart; Timothy Ramsay; Marc Rodger; Debra Witham; Philip S Wells
Journal:  N Engl J Med       Date:  2018-12-04       Impact factor: 91.245

Review 2.  The Role of CDK4/6 Inhibition in Breast Cancer.

Authors:  Conleth G Murphy; Maura N Dickler
Journal:  Oncologist       Date:  2015-04-15

3.  The incidence of thromboembolism for lenalidomide versus thalidomide in older patients with newly diagnosed multiple myeloma.

Authors:  Ang Li; Qian Wu; Greg Warnick; Shan Li; Edward N Libby; David A Garcia; Gary H Lyman
Journal:  Ann Hematol       Date:  2019-11-26       Impact factor: 3.673

4.  Venous thromboembolism in breast cancer patients receiving cyclin-dependent kinase inhibitors.

Authors:  Lorenzo Gervaso; Alberto J Montero; Xuefei Jia; Alok A Khorana
Journal:  J Thromb Haemost       Date:  2019-09-18       Impact factor: 5.824

5.  Incidence and predictors of venous thromboembolism (VTE) among ambulatory high-risk cancer patients undergoing chemotherapy in the United States.

Authors:  Alok A Khorana; Mehul Dalal; Jay Lin; Gregory C Connolly
Journal:  Cancer       Date:  2012-08-14       Impact factor: 6.860

Review 6.  The Strange Case of CDK4/6 Inhibitors: Mechanisms, Resistance, and Combination Strategies.

Authors:  Erik S Knudsen; Agnieszka K Witkiewicz
Journal:  Trends Cancer       Date:  2017-01

7.  Development and validation of a predictive model for chemotherapy-associated thrombosis.

Authors:  Alok A Khorana; Nicole M Kuderer; Eva Culakova; Gary H Lyman; Charles W Francis
Journal:  Blood       Date:  2008-01-23       Impact factor: 22.113

Review 8.  Venous thromboembolism and cancer: risks and outcomes.

Authors:  Agnes Y Y Lee; Mark N Levine
Journal:  Circulation       Date:  2003-06-17       Impact factor: 29.690

9.  Palbociclib and Letrozole in Advanced Breast Cancer.

Authors:  Richard S Finn; Miguel Martin; Hope S Rugo; Stephen Jones; Seock-Ah Im; Karen Gelmon; Nadia Harbeck; Oleg N Lipatov; Janice M Walshe; Stacy Moulder; Eric Gauthier; Dongrui R Lu; Sophia Randolph; Véronique Diéras; Dennis J Slamon
Journal:  N Engl J Med       Date:  2016-11-17       Impact factor: 91.245

10.  The Khorana score for prediction of venous thromboembolism in cancer patients: a systematic review and meta-analysis.

Authors:  Frits I Mulder; Matteo Candeloro; Pieter W Kamphuisen; Marcello Di Nisio; Patrick M Bossuyt; Noori Guman; Kirsten Smit; Harry R Büller; Nick van Es
Journal:  Haematologica       Date:  2019-01-03       Impact factor: 11.047

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  4 in total

Review 1.  Thrombotic events in patients using cyclin dependent kinase 4/6 inhibitors, analysis of existing ambulatory risk assessment models and the potential influences of tumor specific risk factors.

Authors:  Malinda T West; Thomas Kartika; Ashley R Paquin; Erik Liederbauer; Tony J Zheng; Lucy Lane; Kyaw Thein; Joseph J Shatzel
Journal:  Curr Probl Cancer       Date:  2022-01-10       Impact factor: 3.187

Review 2.  Assessing the risk of thromboembolism in cancer patients receiving immunotherapy.

Authors:  Abhishek Goel; Arjun Khorana; Thomas Kartika; Sonia Gowda; Derrick L Tao; Rajat Thawani; Joseph J Shatzel
Journal:  Eur J Haematol       Date:  2022-01-13       Impact factor: 2.997

Review 3.  Cancer-associated venous thromboembolism.

Authors:  Alok A Khorana; Nigel Mackman; Anna Falanga; Ingrid Pabinger; Simon Noble; Walter Ageno; Florian Moik; Agnes Y Y Lee
Journal:  Nat Rev Dis Primers       Date:  2022-02-17       Impact factor: 65.038

Review 4.  Risk factors associated with venous thromboembolism in breast cancer: a narrative review.

Authors:  Zayd Adnan Razouki; Nadeen T Ali; Vinh Q Nguyen; Carmen P Escalante
Journal:  Support Care Cancer       Date:  2022-05-05       Impact factor: 3.359

  4 in total

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