Literature DB >> 32999866

Potential of Lenvatinib for an Expanded Indication from the REFLECT Trial in Patients with Advanced Hepatocellular Carcinoma.

Susumu Maruta1, Sadahisa Ogasawara1,2, Yoshihiko Ooka1, Masamichi Obu3, Masanori Inoue4, Norio Itokawa5, Yuki Haga6, Atsuyoshi Seki7, Shinichiro Okabe8, Ryosaku Azemoto3, Ei Itobayashi4, Masanori Atsukawa5,9, Nobuyuki Sugiura6, Hideaki Mizumoto7, Keisuke Koroki1, Kengo Kanayama1, Hiroaki Kanzaki1, Kazufumi Kobayashi1,2, Soichiro Kiyono1, Masato Nakamura1, Naoya Kanogawa1, Tomoko Saito1, Takayuki Kondo1, Eiichiro Suzuki1, Shingo Nakamoto1, Akinobu Tawada1, Tetsuhiro Chiba1, Makoto Arai1,10, Tatsuo Kanda1,11, Hitoshi Maruyama1,12, Naoya Kato1,2.   

Abstract

BACKGROUND: The present study aimed to assess the efficacy and safety of lenvatinib and verify the possibility of lenvatinib for the expanded indication from the REFLECT trial in patients with advanced hepatocellular carcinoma (HCC) in real-world practice, primarily focusing on the population that was excluded in the REFLECT trial.
METHODS: We retrospectively collected data on patients with advanced HCC who were administered lenvatinib in 7 institutions in Japan.
RESULTS: Of 152 advanced HCC patients, 95 and 57 patients received lenvatinib in first-line and second- or later-line systemic therapies, respectively. The median progression-free survival in Child-Pugh class A patients was nearly equal between first- and second- or later-line therapies (5.2 months; 95% CI 3.7-6.9 for first line, 4.8 months; 95% CI 3.8-5.9 for second or later line, p = 0.933). According to the modified Response Evaluation Criteria in Solid Tumors, the objective response rate of 27 patients (18%) who showed a high burden of intrahepatic lesions (i.e., main portal vein and/or bile duct invasion or 50% or higher liver occupation) at baseline radiological assessment was 41% and similar with that of other population. The present study included 20 patients (13%) with Child-Pugh class B. These patients observed high frequency rates of liver function-related adverse events due to lenvatinib. The 8-week dose intensity of lenvatinib had a strong correlation with liver function according to both the Child-Pugh and albumin - bilirubin scores.
CONCLUSION: Lenvatinib had potential benefits for patients with advanced HCC with second- or later-line therapies and a high burden of intrahepatic lesions. Dose modification should be paid increased attention among patients with poor liver function, such as Child-Pugh class B patients.
Copyright © 2020 by S. Karger AG, Basel.

Entities:  

Keywords:  Hepatocellular carcinoma; Lenvatinib; REFLECT trial

Year:  2020        PMID: 32999866      PMCID: PMC7506220          DOI: 10.1159/000507022

Source DB:  PubMed          Journal:  Liver Cancer        ISSN: 1664-5553            Impact factor:   11.740


  37 in total

Review 1.  Chemotherapy for hepatocellular carcinoma: current status and future perspectives.

Authors:  Masafumi Ikeda; Chigusa Morizane; Makoto Ueno; Takuji Okusaka; Hiroshi Ishii; Junji Furuse
Journal:  Jpn J Clin Oncol       Date:  2018-02-01       Impact factor: 3.019

2.  Clinical outcomes of sorafenib treatment failure for advanced hepatocellular carcinoma and candidates for regorafenib treatment in real-world practice.

Authors:  Shinsuke Uchikawa; Tomokazu Kawaoka; Hiroshi Aikata; Kenichiro Kodama; Yuno Nishida; Yuki Inagaki; Masahiro Hatooka; Kei Morio; Takashi Nakahara; Eisuke Murakami; Akira Hiramatsu; Masataka Tsuge; Michio Imamura; Yoshiiku Kawakami; Kazuaki Chayama
Journal:  Hepatol Res       Date:  2018-05-27       Impact factor: 4.288

3.  Pharmacokinetics and excretion of (14)C-lenvatinib in patients with advanced solid tumors or lymphomas.

Authors:  Anne-Charlotte Dubbelman; Hilde Rosing; Cynthia Nijenhuis; Alwin D R Huitema; Marja Mergui-Roelvink; Anubha Gupta; David Verbel; Gary Thompson; Robert Shumaker; Jan H M Schellens; Jos H Beijnen
Journal:  Invest New Drugs       Date:  2014-11-08       Impact factor: 3.850

4.  Efficacy and safety of sorafenib in patients in the Asia-Pacific region with advanced hepatocellular carcinoma: a phase III randomised, double-blind, placebo-controlled trial.

Authors:  Ann-Lii Cheng; Yoon-Koo Kang; Zhendong Chen; Chao-Jung Tsao; Shukui Qin; Jun Suk Kim; Rongcheng Luo; Jifeng Feng; Shenglong Ye; Tsai-Sheng Yang; Jianming Xu; Yan Sun; Houjie Liang; Jiwei Liu; Jiejun Wang; Won Young Tak; Hongming Pan; Karin Burock; Jessie Zou; Dimitris Voliotis; Zhongzhen Guan
Journal:  Lancet Oncol       Date:  2008-12-16       Impact factor: 41.316

5.  Effect of everolimus on survival in advanced hepatocellular carcinoma after failure of sorafenib: the EVOLVE-1 randomized clinical trial.

Authors:  Andrew X Zhu; Masatoshi Kudo; Eric Assenat; Stéphane Cattan; Yoon-Koo Kang; Ho Yeong Lim; Ronnie T P Poon; Jean-Frederic Blanc; Arndt Vogel; Chao-Long Chen; Etienne Dorval; Markus Peck-Radosavljevic; Armando Santoro; Bruno Daniele; Junji Furuse; Annette Jappe; Kevin Perraud; Oezlem Anak; Dalila B Sellami; Li-Tzong Chen
Journal:  JAMA       Date:  2014-07-02       Impact factor: 56.272

6.  Brivanib in patients with advanced hepatocellular carcinoma who were intolerant to sorafenib or for whom sorafenib failed: results from the randomized phase III BRISK-PS study.

Authors:  Josep M Llovet; Thomas Decaens; Jean-Luc Raoul; Eveline Boucher; Masatoshi Kudo; Charissa Chang; Yoon-Koo Kang; Eric Assenat; Ho-Yeong Lim; Valerie Boige; Philippe Mathurin; Laetitia Fartoux; Deng-Yn Lin; Jordi Bruix; Ronnie T Poon; Morris Sherman; Jean-Frédéric Blanc; Richard S Finn; Won-Young Tak; Yee Chao; Rana Ezzeddine; David Liu; Ian Walters; Joong-Won Park
Journal:  J Clin Oncol       Date:  2013-08-26       Impact factor: 44.544

7.  Brivanib versus sorafenib as first-line therapy in patients with unresectable, advanced hepatocellular carcinoma: results from the randomized phase III BRISK-FL study.

Authors:  Philip J Johnson; Shukui Qin; Joong-Won Park; Ronnie T P Poon; Jean-Luc Raoul; Philip A Philip; Chih-Hung Hsu; Tsung-Hui Hu; Jeong Heo; Jianming Xu; Ligong Lu; Yee Chao; Eveline Boucher; Kwang-Hyub Han; Seung-Woon Paik; Jorge Robles-Aviña; Masatoshi Kudo; Lunan Yan; Abhasnee Sobhonslidsuk; Dmitry Komov; Thomas Decaens; Won-Young Tak; Long-Bin Jeng; David Liu; Rana Ezzeddine; Ian Walters; Ann-Lii Cheng
Journal:  J Clin Oncol       Date:  2013-08-26       Impact factor: 44.544

8.  Sorafenib in advanced hepatocellular carcinoma.

Authors:  Josep M Llovet; Sergio Ricci; Vincenzo Mazzaferro; Philip Hilgard; Edward Gane; Jean-Frédéric Blanc; Andre Cosme de Oliveira; Armando Santoro; Jean-Luc Raoul; Alejandro Forner; Myron Schwartz; Camillo Porta; Stefan Zeuzem; Luigi Bolondi; Tim F Greten; Peter R Galle; Jean-François Seitz; Ivan Borbath; Dieter Häussinger; Tom Giannaris; Minghua Shan; Marius Moscovici; Dimitris Voliotis; Jordi Bruix
Journal:  N Engl J Med       Date:  2008-07-24       Impact factor: 91.245

9.  Complete removal of the tumor-bearing portal territory decreases local tumor recurrence and improves disease-specific survival of patients with hepatocellular carcinoma.

Authors:  Junichi Shindoh; Masatoshi Makuuchi; Yutaka Matsuyama; Yoshihiro Mise; Junichi Arita; Yoshihiro Sakamoto; Kiyoshi Hasegawa; Norihiro Kokudo
Journal:  J Hepatol       Date:  2015-10-24       Impact factor: 25.083

10.  Ramucirumab after sorafenib in patients with advanced hepatocellular carcinoma and increased α-fetoprotein concentrations (REACH-2): a randomised, double-blind, placebo-controlled, phase 3 trial.

Authors:  Andrew X Zhu; Yoon-Koo Kang; Chia-Jui Yen; Richard S Finn; Peter R Galle; Josep M Llovet; Eric Assenat; Giovanni Brandi; Marc Pracht; Ho Yeong Lim; Kun-Ming Rau; Kenta Motomura; Izumi Ohno; Philippe Merle; Bruno Daniele; Dong Bok Shin; Guido Gerken; Christophe Borg; Jean-Baptiste Hiriart; Takuji Okusaka; Manabu Morimoto; Yanzhi Hsu; Paolo B Abada; Masatoshi Kudo
Journal:  Lancet Oncol       Date:  2019-01-18       Impact factor: 41.316

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  20 in total

1.  Real-World Efficacy and Safety of Lenvatinib in Korean Patients with Advanced Hepatocellular Carcinoma: A Multicenter Retrospective Analysis.

Authors:  Jaekyung Cheon; Hong Jae Chon; Yeonghak Bang; Neung Hwa Park; Jung Woo Shin; Kang Mo Kim; Han Chu Lee; Jooho Lee; Changhoon Yoo; Baek-Yeol Ryoo
Journal:  Liver Cancer       Date:  2020-07-29       Impact factor: 11.740

2.  Hepatic Arterial Infusion Chemotherapy versus Sorafenib in Patients with Advanced Hepatocellular Carcinoma.

Authors:  Kazuomi Ueshima; Sadahisa Ogasawara; Masafumi Ikeda; Yutaka Yasui; Takeshi Terashima; Tatsuya Yamashita; Shuntaro Obi; Shinpei Sato; Hiroshi Aikata; Takumi Ohmura; Hidekatsu Kuroda; Takamasa Ohki; Kengo Nagashima; Yoshihiko Ooka; Masahiro Takita; Masayuki Kurosaki; Kazuaki Chayama; Shuichi Kaneko; Namiki Izumi; Naoya Kato; Masatoshi Kudo; Masao Omata
Journal:  Liver Cancer       Date:  2020-07-24       Impact factor: 11.740

3.  Posttreatment after Lenvatinib in Patients with Advanced Hepatocellular Carcinoma.

Authors:  Keisuke Koroki; Naoya Kanogawa; Susumu Maruta; Sadahisa Ogasawara; Yotaro Iino; Masamichi Obu; Tomomi Okubo; Norio Itokawa; Takahiro Maeda; Masanori Inoue; Yuki Haga; Atsuyoshi Seki; Shinichiro Okabe; Yoshihiro Koma; Ryosaku Azemoto; Masanori Atsukawa; Ei Itobayashi; Kenji Ito; Nobuyuki Sugiura; Hideaki Mizumoto; Hidemi Unozawa; Terunao Iwanaga; Takafumi Sakuma; Naoto Fujita; Hiroaki Kanzaki; Kazufumi Kobayashi; Soichiro Kiyono; Masato Nakamura; Tomoko Saito; Takayuki Kondo; Eiichiro Suzuki; Yoshihiko Ooka; Shingo Nakamoto; Akinobu Tawada; Tetsuhiro Chiba; Makoto Arai; Tatsuo Kanda; Hitoshi Maruyama; Jun Kato; Naoya Kato
Journal:  Liver Cancer       Date:  2021-04-20       Impact factor: 11.740

4.  Real-World Data on Ramucirumab Therapy including Patients Who Experienced Two or More Systemic Treatments: A Multicenter Study.

Authors:  Yutaka Yasui; Masayuki Kurosaki; Kaoru Tsuchiya; Yuka Hayakawa; Chitomi Hasebe; Masami Abe; Chikara Ogawa; Kouji Joko; Hironori Ochi; Toshifumi Tada; Shinichiro Nakamura; Koichiro Furuta; Hiroyuki Kimura; Keiji Tsuji; Yuji Kojima; Takehiro Akahane; Takashi Tamada; Yasushi Uchida; Masahiko Kondo; Akeri Mitsuda; Namiki Izumi
Journal:  Cancers (Basel)       Date:  2022-06-16       Impact factor: 6.575

5.  Lenvatinib with or without Concurrent Drug-Eluting Beads Transarterial Chemoembolization in Patients with Unresectable, Advanced Hepatocellular Carcinoma: A Real-World, Multicenter, Retrospective Study.

Authors:  Dongdong Xia; Wei Bai; Enxin Wang; Jiaping Li; Xiaoming Chen; Zhexuan Wang; Mingsheng Huang; Ming Huang; Junhui Sun; Weizhu Yang; Zhengyu Lin; Jianbing Wu; Zixiang Li; Shufa Yang; Xu Zhu; Zaizhong Chen; Yanfang Zhang; Wenzhe Fan; Qicong Mai; Rong Ding; Chunhui Nie; Long Feng; Xueda Li; Wukui Huang; Jun Sun; Qiuhe Wang; Yong Lv; Xiaomei Li; Bohan Luo; Zhengyu Wang; Jie Yuan; Wengang Guo; Kai Li; Bing Li; Ruijun Li; Zhanxin Yin; Jielai Xia; Guohong Han
Journal:  Liver Cancer       Date:  2022-03-09       Impact factor: 12.430

Review 6.  Systemic Treatment for Older Patients with Unresectable Hepatocellular Carcinoma.

Authors:  Antonella Cammarota; Antonio D'Alessio; Tiziana Pressiani; Lorenza Rimassa; Nicola Personeni
Journal:  Drugs Aging       Date:  2021-06-21       Impact factor: 3.923

7.  Identification of the Response-Related Biomarker of Bimonthly Hepatic Arterial Infusion Chemotherapy.

Authors:  Kei Moriya; Tadashi Namisaki; Hiroaki Takaya; Kosuke Kaji; Hideto Kawaratani; Naotaka Shimozato; Yasuhiko Sawada; Akitoshi Douhara; Shinya Sato; Masanori Furukawa; Koh Kitagawa; Takemi Akahane; Hitoshi Yoshiji
Journal:  J Clin Med       Date:  2021-02-07       Impact factor: 4.241

Review 8.  Lenvatinib for Hepatocellular Carcinoma: A Literature Review.

Authors:  Takeshi Hatanaka; Atsushi Naganuma; Satoru Kakizaki
Journal:  Pharmaceuticals (Basel)       Date:  2021-01-06

9.  Baseline serum angiopoietin-2 and VEGF levels predict the deterioration of the liver functional reserve during lenvatinib treatment for hepatocellular carcinoma.

Authors:  Taku Shigesawa; Goki Suda; Megumi Kimura; Osamu Maehara; Yoshimasa Tokuchi; Akinori Kubo; Ren Yamada; Ken Furuya; Masaru Baba; Takashi Kitagataya; Kazuharu Suzuki; Masatsugu Ohara; Naoki Kawagishi; Masato Nakai; Takuya Sho; Mitsuteru Natsuizaka; Kenichi Morikawa; Koji Ogawa; Naoya Sakamoto
Journal:  PLoS One       Date:  2021-03-01       Impact factor: 3.240

10.  Antitumor Effect of Lenvatinib Combined with Alisertib in Hepatocellular Carcinoma by Targeting the DNA Damage Pathway.

Authors:  Jianwen Hao; Qizhen Peng; Keruo Wang; Ge Yu; Yi Pan; Xiaoling Du; Na Hu; Xuening Zhang; Yu Qin; Huikai Li
Journal:  Biomed Res Int       Date:  2021-07-22       Impact factor: 3.411

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