Literature DB >> 32534646

Atezolizumab, vemurafenib, and cobimetinib as first-line treatment for unresectable advanced BRAFV600 mutation-positive melanoma (IMspire150): primary analysis of the randomised, double-blind, placebo-controlled, phase 3 trial.

Ralf Gutzmer1, Daniil Stroyakovskiy2, Helen Gogas3, Caroline Robert4, Karl Lewis5, Svetlana Protsenko6, Rodrigo P Pereira7, Thomas Eigentler8, Piotr Rutkowski9, Lev Demidov10, Georgy Moiseevich Manikhas11, Yibing Yan12, Kuan-Chieh Huang12, Anne Uyei12, Virginia McNally13, Grant A McArthur14, Paolo A Ascierto15.   

Abstract

BACKGROUND: IMspire150 aimed to evaluate first-line combination treatment with BRAF plus MEK inhibitors and immune checkpoint therapy in BRAFV600 mutation-positive advanced or metastatic melanoma.
METHODS: IMspire150 was a randomised, double-blind, placebo-controlled phase 3 study done at 112 institutes in 20 countries. Patients with unresectable stage IIIc-IV, BRAFV600 mutation-positive melanoma were randomly assigned 1:1 to 28-day cycles of atezolizumab, vemurafenib, and cobimetinib (atezolizumab group) or atezolizumab placebo, vemurafenib, and cobimetinib (control group). In cycle 1, all patients received vemurafenib and cobimetinib only; atezolizumab placebo was added from cycle 2 onward. Randomisation was stratified by lactate dehydrogenase concentration and geographical region. Blinding for atezolizumab was achieved by means of an identical intravenous placebo, and blinding for vemurafenib was achieved by means of a placebo tablet. The primary outcome was investigator-assessed progression-free survival. This trial (ClinicalTrials.gov, NCT02908672) is ongoing but no longer recruiting patients.
FINDINGS: Between Jan 13, 2017, and April 26, 2018, 777 patients were screened and 514 were enrolled and randomly assigned to the atezolizumab group (n=256) or control group (n=258). At a median follow-up of 18·9 months (IQR 10·4-23·8), progression-free survival as assessed by the study investigator was significantly prolonged with atezolizumab versus control (15·1 vs 10·6 months; hazard ratio [HR] 0·78; 95% CI 0·63-0·97; p=0·025). Common treatment-related adverse events (>30%) in the atezolizumab and control groups were blood creatinine phosphokinase increased (51·3% vs 44·8%), diarrhoea (42·2% vs 46·6%), rash (40·9%, both groups), arthralgia (39·1% vs 28·1%), pyrexia (38·7% vs 26·0%), alanine aminotransferase increased (33·9% vs 22·8%), and lipase increased (32·2% vs 27·4%); 13% of patients in the atezolizumab group and 16% in the control group stopped all treatment because of adverse events.
INTERPRETATION: The addition of atezolizumab to targeted therapy with vemurafenib and cobimetinib was safe and tolerable and significantly increased progression-free survival in patients with BRAFV600 mutation-positive advanced melanoma. FUNDING: F Hoffmann-La Roche and Genentech.
Copyright © 2020 Elsevier Ltd. All rights reserved.

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Year:  2020        PMID: 32534646     DOI: 10.1016/S0140-6736(20)30934-X

Source DB:  PubMed          Journal:  Lancet        ISSN: 0140-6736            Impact factor:   79.321


  134 in total

1.  Mechanisms of Resistance to BRAF-Targeted Melanoma Therapies.

Authors:  Ozgecan Dulgar; Tugce Kutuk; Zeynep Eroglu
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2.  Combining BRAF/MEK Inhibitors with Immunotherapy in the Treatment of Metastatic Melanoma.

Authors:  Dimitrios C Ziogas; Frosso Konstantinou; Spyros Bouros; Maria Theochari; Helen Gogas
Journal:  Am J Clin Dermatol       Date:  2021-03-25       Impact factor: 7.403

3.  Melanoma: An immunotherapy journey from bench to bedside.

Authors:  Vishal Navani; Moira C Graves; Hiren Mandaliya; Martin Hong; Andre van der Westhuizen; Jennifer Martin; Nikola A Bowden
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Review 4.  Therapeutic Advancements Across Clinical Stages in Melanoma, With a Focus on Targeted Immunotherapy.

Authors:  Claudia Trojaniello; Jason J Luke; Paolo A Ascierto
Journal:  Front Oncol       Date:  2021-06-10       Impact factor: 6.244

5.  Real-world analysis of clinicopathological characteristics, survival rates, and prognostic factors in patients with melanoma brain metastases in China.

Authors:  Yang Wang; Bin Lian; Lu Si; ZhiHong Chi; XiNan Sheng; Xuan Wang; LiLi Mao; BiXia Tang; SiMing Li; XieQiao Yan; Xue Bai; Li Zhou; ChuanLiang Cui; Jun Guo
Journal:  J Cancer Res Clin Oncol       Date:  2021-02-21       Impact factor: 4.553

6.  Triple therapy for BRAFV600-mutated melanoma.

Authors:  Antoni Ribas
Journal:  Lancet       Date:  2020-06-13       Impact factor: 79.321

Review 7.  Development of Immunotherapy Combination Strategies in Cancer.

Authors:  Timothy A Yap; Eileen E Parkes; Weiyi Peng; Justin T Moyers; Michael A Curran; Hussein A Tawbi
Journal:  Cancer Discov       Date:  2021-04-02       Impact factor: 39.397

Review 8.  Defining and Targeting BRAF Mutations in Solid Tumors.

Authors:  Briana R Halle; Douglas B Johnson
Journal:  Curr Treat Options Oncol       Date:  2021-02-27

Review 9.  Current management of melanoma patients with nodal metastases.

Authors:  Dale Han; Alexander C J van Akkooi; Richard J Straker; Adrienne B Shannon; Giorgos C Karakousis; Lin Wang; Kevin B Kim; Douglas Reintgen
Journal:  Clin Exp Metastasis       Date:  2021-05-07       Impact factor: 4.510

10.  BRAF-MEK inhibitors as steroid-sparing bridge prior to checkpoint blockade therapy in symptomatic intracranial melanoma.

Authors:  Karam Khaddour; Tanner M Johanns; George Ansstas
Journal:  Melanoma Manag       Date:  2021-02-15
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