Literature DB >> 30247579

Effect of fluconazole prophylaxis on Candida fluconazole susceptibility in premature infants.

Julie Autmizguine1,2,3, P Brian Smith4,5, Kristi Prather5, Catherine Bendel6, Girija Natarajan7, Margarita Bidegain4, David A Kaufman8, David J Burchfield9, Ashley S Ross10, Paresh Pandit11, Wiley A Schell12, Jamie Gao5, Daniel K Benjamin4,5.   

Abstract

Objectives: Extremely premature infants are at high risk of developing invasive candidiasis; fluconazole prophylaxis is safe and effective for reducing invasive candidiasis in this population but further study is needed. We sought to better understand the effect of prophylactic fluconazole on a selection of fluconazole-resistant Candida species.
Methods: We evaluated the susceptibility to fluconazole of Candida isolates from premature infants (<750 g birth weight) enrolled in a multicentre, randomized, placebo-controlled trial of fluconazole prophylaxis. Candida species were isolated through surveillance cultures at baseline (study day 0-7), period 1 (study day 8-28) and period 2 (study day 29-49). Fluconazole MICs were determined for all Candida isolates.
Results: Three hundred and sixty-one infants received fluconazole (n = 188) or placebo (n = 173). After the baseline period, Candida colonization was significantly lower in the fluconazole group compared with placebo during periods 1 (5% versus 27%; P < 0.001) and 2 (3% versus 27%; P < 0.001). After the baseline period, two infants (1%) were colonized with at least one fluconazole-resistant Candida in each group. Median fluconazole MIC was similar in both treatment groups at baseline and period 1. However, in period 2, median MIC was higher in the fluconazole group compared with placebo (1.00 versus 0.50 mg/L, P = 0.01). There was no emergence of resistance observed and no patients developed invasive candidiasis with a resistant Candida isolate. Conclusions: Fluconazole prophylaxis decreased Candida albicans and 'non-albicans' Candida colonization and was associated with a slightly higher fluconazole MIC for colonizing Candida isolates.

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Year:  2018        PMID: 30247579      PMCID: PMC6927883          DOI: 10.1093/jac/dky353

Source DB:  PubMed          Journal:  J Antimicrob Chemother        ISSN: 0305-7453            Impact factor:   5.790


  23 in total

Review 1.  Progress in antifungal susceptibility testing of Candida spp. by use of Clinical and Laboratory Standards Institute broth microdilution methods, 2010 to 2012.

Authors:  M A Pfaller; D J Diekema
Journal:  J Clin Microbiol       Date:  2012-06-27       Impact factor: 5.948

2.  Neonatal candidiasis among extremely low birth weight infants: risk factors, mortality rates, and neurodevelopmental outcomes at 18 to 22 months.

Authors:  Daniel K Benjamin; Barbara J Stoll; Avory A Fanaroff; Scott A McDonald; William Oh; Rosemary D Higgins; Shahnaz Duara; Kenneth Poole; Abbot Laptook; Ronald Goldberg
Journal:  Pediatrics       Date:  2006-01       Impact factor: 7.124

3.  In vivo fluconazole pharmacodynamics and resistance development in a previously susceptible Candida albicans population examined by microbiologic and transcriptional profiling.

Authors:  D Andes; A Lepak; J Nett; L Lincoln; K Marchillo
Journal:  Antimicrob Agents Chemother       Date:  2006-07       Impact factor: 5.191

4.  Fluconazole for prophylaxis against candidal rectal colonization in the very low birth weight infant.

Authors:  S D Kicklighter; S C Springer; T Cox; T C Hulsey; R B Turner
Journal:  Pediatrics       Date:  2001-02       Impact factor: 7.124

5.  Emergence of fluconazole resistance in a Candida parapsilosis strain that caused infections in a neonatal intensive care unit.

Authors:  Emmi Sarvikivi; Outi Lyytikäinen; David R Soll; Claude Pujol; Michael A Pfaller; Malcolm Richardson; Pirkko Koukila-Kähkölä; Päivi Luukkainen; Harri Saxén
Journal:  J Clin Microbiol       Date:  2005-06       Impact factor: 5.948

6.  Twice weekly fluconazole prophylaxis for prevention of invasive Candida infection in high-risk infants of <1000 grams birth weight.

Authors:  David Kaufman; Robert Boyle; Kevin C Hazen; James T Patrie; Melinda Robinson; Leigh B Grossman
Journal:  J Pediatr       Date:  2005-08       Impact factor: 4.406

7.  A multicenter, randomized trial of prophylactic fluconazole in preterm neonates.

Authors:  Paolo Manzoni; Ilaria Stolfi; Lorenza Pugni; Lidia Decembrino; Cristiana Magnani; Gennaro Vetrano; Elisabetta Tridapalli; Giuseppina Corona; Chiara Giovannozzi; Daniele Farina; Riccardo Arisio; Franco Merletti; Milena Maule; Fabio Mosca; Roberto Pedicino; Mauro Stronati; Michael Mostert; Giovanna Gomirato
Journal:  N Engl J Med       Date:  2007-06-14       Impact factor: 91.245

8.  Routine use of fluconazole prophylaxis in a neonatal intensive care unit does not select natively fluconazole-resistant Candida subspecies.

Authors:  Paolo Manzoni; Marialisa Leonessa; Paolo Galletto; Maria Agnese Latino; Riccardo Arisio; Milena Maule; Giovanni Agriesti; Luca Gastaldo; Elena Gallo; Michael Mostert; Daniele Farina
Journal:  Pediatr Infect Dis J       Date:  2008-08       Impact factor: 2.129

9.  Effect of fluconazole prophylaxis on candidiasis and mortality in premature infants: a randomized clinical trial.

Authors:  Daniel K Benjamin; Mark L Hudak; Shahnaz Duara; David A Randolph; Margarita Bidegain; Gratias T Mundakel; Girija Natarajan; David J Burchfield; Robert D White; Karen E Shattuck; Natalie Neu; Catherine M Bendel; M Roger Kim; Neil N Finer; Dan L Stewart; Antonio C Arrieta; Kelly C Wade; David A Kaufman; Paolo Manzoni; Kristi O Prather; Daniela Testoni; Katherine Y Berezny; P Brian Smith
Journal:  JAMA       Date:  2014-05-07       Impact factor: 157.335

10.  Efficacy and safety of fluconazole prophylaxis in extremely low birth weight infants: multicenter pre-post cohort study.

Authors:  Juyoung Lee; Han-Suk Kim; Seung Han Shin; Chang Won Choi; Ee-Kyung Kim; Eun Hwa Choi; Beyong Il Kim; Jung-Hwan Choi
Journal:  BMC Pediatr       Date:  2016-05-16       Impact factor: 2.125

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  12 in total

1.  A New Variant of Mutational and Polymorphic Signatures in the ERG11 Gene of Fluconazole-Resistant Candida albicans.

Authors:  Arome Solomon Odiba; Olanrewaju Ayodeji Durojaye; Ifeoma Maureen Ezeonu; Anthony Christian Mgbeahuruike; Bennett Chima Nwanguma
Journal:  Infect Drug Resist       Date:  2022-06-17       Impact factor: 4.177

Review 2.  Review of Fluconazole Treatment and Prophylaxis for Invasive Candidiasis in Neonates.

Authors:  Chi D Hornik; Deborah S Bondi; Nicole M Greene; M Petrea Cober; Barnabas John
Journal:  J Pediatr Pharmacol Ther       Date:  2021-02-15

3.  Physiologically-Based Pharmacokinetic Modeling of Fluconazole Using Plasma and Cerebrospinal Fluid Samples From Preterm and Term Infants.

Authors:  Jacqueline G Gerhart; Kevin M Watt; Andrea Edginton; Kelly C Wade; Sara N Salerno; Daniel K Benjamin; P Brian Smith; Christoph P Hornik; Michael Cohen-Wolkowiez; Shahnaz Duara; Ashley Ross; Karen Shattuck; Dan L Stewart; Natalie Neu; Daniel Gonzalez
Journal:  CPT Pharmacometrics Syst Pharmacol       Date:  2019-05-22

Review 4.  Therapeutic Drug Monitoring Is a Feasible Tool to Personalize Drug Administration in Neonates Using New Techniques: An Overview on the Pharmacokinetics and Pharmacodynamics in Neonatal Age.

Authors:  Domenico Umberto De Rose; Sara Cairoli; Marco Dionisi; Alessandra Santisi; Luca Massenzi; Bianca Maria Goffredo; Carlo Dionisi-Vici; Andrea Dotta; Cinzia Auriti
Journal:  Int J Mol Sci       Date:  2020-08-17       Impact factor: 5.923

5.  Breakpoints for the Classification of Anti-Candida Compounds in Antifungal Screening.

Authors:  Danielle da Nóbrega Alves; Alana Rodrigues Ferreira; Allana Brunna Sucupira Duarte; Ana Karoline Vieira Melo; Damião Pergentino de Sousa; Ricardo Dias de Castro
Journal:  Biomed Res Int       Date:  2021-04-06       Impact factor: 3.411

6.  Mucosal Bacteria Modulate Candida albicans Virulence in Oropharyngeal Candidiasis.

Authors:  M Bertolini; R Vazquez Munoz; L Archambault; S Shah; J G S Souza; R C Costa; A Thompson; Y Zhou; T Sobue; A Dongari-Bagtzoglou
Journal:  mBio       Date:  2021-08-17       Impact factor: 7.867

Review 7.  Fungicide effects on human fungal pathogens: Cross-resistance to medical drugs and beyond.

Authors:  Rafael W Bastos; Luana Rossato; Gustavo H Goldman; Daniel A Santos
Journal:  PLoS Pathog       Date:  2021-12-09       Impact factor: 6.823

8.  Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols.

Authors:  Nicolas Lebouvier; Fabrice Pagniez; Young Min Na; Da Shi; Patricia Pinson; Mathieu Marchivie; Jean Guillon; Tarek Hakki; Rita Bernhardt; Sook Wah Yee; Claire Simons; Marie-Pierre Lézé; Rolf W Hartmann; Angélique Mularoni; Guillaume Le Baut; Isabelle Krimm; Ruben Abagyan; Patrice Le Pape; Marc Le Borgne
Journal:  Pharmaceuticals (Basel)       Date:  2020-08-08

Review 9.  Plant-Derived Substances in the Fight Against Infections Caused by Candida Species.

Authors:  Ibeth Guevara-Lora; Grazyna Bras; Justyna Karkowska-Kuleta; Miriam González-González; Kinga Ceballos; Wiktoria Sidlo; Maria Rapala-Kozik
Journal:  Int J Mol Sci       Date:  2020-08-25       Impact factor: 5.923

Review 10.  Invasive Candida Infections in Neonates after Major Surgery: Current Evidence and New Directions.

Authors:  Domenico Umberto De Rose; Alessandra Santisi; Maria Paola Ronchetti; Ludovica Martini; Lisa Serafini; Pasqua Betta; Marzia Maino; Francesco Cavigioli; Ilaria Cocchi; Lorenza Pugni; Elvira Bonanno; Chryssoula Tzialla; Mario Giuffrè; Jenny Bua; Benedetta Della Torre; Giovanna Nardella; Danila Mazzeo; Paolo Manzoni; Andrea Dotta; Pietro Bagolan; Cinzia Auriti
Journal:  Pathogens       Date:  2021-03-09
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