Literature DB >> 29388990

The inverse electron-demand Diels-Alder reaction as a new methodology for the synthesis of 225Ac-labelled radioimmunoconjugates.

S Poty1, R Membreno, J M Glaser, A Ragupathi, W W Scholz, B M Zeglis, J S Lewis.   

Abstract

The inverse electron-demand Diels-Alder reaction between tetrazine (Tz) and trans-cyclooctene (TCO) facilitates the efficient radiosynthesis of 225Ac-labelled radioimmunoconjugates in a two-step method, outperforming conventional approaches based on isothiocyanate couplings.

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Year:  2018        PMID： 29388990      PMCID： PMC5843558          DOI： 10.1039/c7cc09129j

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN： 1359-7345            Impact factor:   6.222


  21 in total

1.  Copper-free click chemistry with the short-lived positron emitter fluorine-18.

Authors:  Vincent Bouvet; Melinda Wuest; Frank Wuest
Journal:  Org Biomol Chem       Date:  2011-09-22       Impact factor: 3.876

2.  The traceless Staudinger ligation for indirect 18F-radiolabelling.

Authors:  Laurence Carroll; Sophie Boldon; Romain Bejot; Jane E Moore; Jérôme Declerck; Véronique Gouverneur
Journal:  Org Biomol Chem       Date:  2010-11-22       Impact factor: 3.876

Review 3.  Staudinger ligation as a method for bioconjugation.

Authors:  Sander S van Berkel; Mark B van Eldijk; Jan C M van Hest
Journal:  Angew Chem Int Ed Engl       Date:  2011-09-02       Impact factor: 15.336

4.  Efficient 1-step radiolabeling of monoclonal antibodies to high specific activity with 225Ac for α-particle radioimmunotherapy of cancer.

Authors:  William F Maguire; Michael R McDevitt; Peter M Smith-Jones; David A Scheinberg
Journal:  J Nucl Med       Date:  2014-06-30       Impact factor: 10.057

5.  Design and synthesis of 225Ac radioimmunopharmaceuticals.

Authors:  Michael R McDevitt; Dangshe Ma; Jim Simon; R Keith Frank; David A Scheinberg
Journal:  Appl Radiat Isot       Date:  2002-12       Impact factor: 1.513

6.  Tumor therapy with targeted atomic nanogenerators.

Authors:  M R McDevitt; D Ma; L T Lai; J Simon; P Borchardt; R K Frank; K Wu; V Pellegrini; M J Curcio; M Miederer; N H Bander; D A Scheinberg
Journal:  Science       Date:  2001-11-16       Impact factor: 47.728

7.  Tetrazine-trans-cyclooctene ligation for the rapid construction of integrin αvβ₃ targeted PET tracer based on a cyclic RGD peptide.

Authors:  Ramajeyam Selvaraj; Shuanglong Liu; Matthew Hassink; Chiun-Wei Huang; Li-Peng Yap; Ryan Park; Joseph M Fox; Zibo Li; Peter S Conti
Journal:  Bioorg Med Chem Lett       Date:  2011-05-04       Impact factor: 2.823

8.  Large scale accelerator production of 225Ac: Effective cross sections for 78-192MeV protons incident on 232Th targets.

Authors:  J R Griswold; D G Medvedev; J W Engle; R Copping; J M Fitzsimmons; V Radchenko; J C Cooley; M E Fassbender; D L Denton; K E Murphy; A C Owens; E R Birnbaum; K D John; F M Nortier; D W Stracener; L H Heilbronn; L F Mausner; S Mirzadeh
Journal:  Appl Radiat Isot       Date:  2016-09-28       Impact factor: 1.513

9.  Improved synthesis and biological evaluation of chelator-modified α-MSH analogs prepared by copper-free click chemistry.

Authors:  Nicholas J Baumhover; Molly E Martin; Sharavathi G Parameswarappa; Kyle C Kloepping; M Sue O'Dorisio; F Christopher Pigge; Michael K Schultz
Journal:  Bioorg Med Chem Lett       Date:  2011-08-08       Impact factor: 2.823

10.  Initial evaluation of (227)Th-p-benzyl-DOTA-rituximab for low-dose rate alpha-particle radioimmunotherapy.

Authors:  Jostein Dahle; Jørgen Borrebaek; Katrine B Melhus; Oyvind S Bruland; Gro Salberg; Dag Rune Olsen; Roy H Larsen
Journal:  Nucl Med Biol       Date:  2006-02       Impact factor: 2.408
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  13 in total

1.  Leveraging Bioorthogonal Click Chemistry to Improve 225Ac-Radioimmunotherapy of Pancreatic Ductal Adenocarcinoma.

Authors:  Sophie Poty; Lukas M Carter; Komal Mandleywala; Rosemery Membreno; Dalya Abdel-Atti; Ashwin Ragupathi; Wolfgang W Scholz; Brian M Zeglis; Jason S Lewis
Journal:  Clin Cancer Res       Date:  2018-10-23       Impact factor: 12.531

Review 2.  Overview of the Most Promising Radionuclides for Targeted Alpha Therapy: The "Hopeful Eight".

Authors:  Romain Eychenne; Michel Chérel; Férid Haddad; François Guérard; Jean-François Gestin
Journal:  Pharmaceutics       Date:  2021-06-18       Impact factor: 6.321

3.  Multifunctional Clickable Reagents for Rapid Bioorthogonal Astatination and Radio-Crosslinking.

Authors:  Christoph Denk; Martin Wilkovitsch; Emma Aneheim; Matthias M Herth; Holger Jensen; Sture Lindegren; Hannes Mikula
Journal:  Chempluschem       Date:  2019-04-04       Impact factor: 2.863

Review 4.  Development of Targeted Alpha Particle Therapy for Solid Tumors.

Authors:  Narges K Tafreshi; Michael L Doligalski; Christopher J Tichacek; Darpan N Pandya; Mikalai M Budzevich; Ghassan El-Haddad; Nikhil I Khushalani; Eduardo G Moros; Mark L McLaughlin; Thaddeus J Wadas; David L Morse
Journal:  Molecules       Date:  2019-11-26       Impact factor: 4.411

5.  A suitable time point for quantifying the radiochemical purity of 225Ac-labeled radiopharmaceuticals.

Authors:  James M Kelly; Alejandro Amor-Coarasa; Elizabeth Sweeney; Justin J Wilson; Patrick W Causey; John W Babich
Journal:  EJNMMI Radiopharm Chem       Date:  2021-12-20

6.  Evaluation of polydentate picolinic acid chelating ligands and an α-melanocyte-stimulating hormone derivative for targeted alpha therapy using ISOL-produced 225Ac.

Authors:  Caterina F Ramogida; Andrew K H Robertson; Una Jermilova; Chengcheng Zhang; Hua Yang; Peter Kunz; Jens Lassen; Ivica Bratanovic; Victoria Brown; Lily Southcott; Cristina Rodríguez-Rodríguez; Valery Radchenko; François Bénard; Chris Orvig; Paul Schaffer
Journal:  EJNMMI Radiopharm Chem       Date:  2019-08-06

Review 7.  Recent Advances in Bioorthogonal Click Chemistry for Efficient Synthesis of Radiotracers and Radiopharmaceuticals.

Authors:  Sajid Mushtaq; Seong-Jae Yun; Jongho Jeon
Journal:  Molecules       Date:  2019-10-02       Impact factor: 4.411

8.  89Zr-PET imaging of DNA double-strand breaks for the early monitoring of response following α- and β-particle radioimmunotherapy in a mouse model of pancreatic ductal adenocarcinoma.

Authors:  Sophie Poty; Komal Mandleywala; Edward O'Neill; James C Knight; Bart Cornelissen; Jason S Lewis
Journal:  Theranostics       Date:  2020-04-27       Impact factor: 11.556

9.  Delivery of polymeric nanostars for molecular imaging and endoradiotherapy through the enhanced permeability and retention (EPR) effect.

Authors:  Jeroen A C M Goos; Andrew Cho; Lukas M Carter; Thomas R Dilling; Maria Davydova; Komal Mandleywala; Simon Puttick; Abhishek Gupta; William S Price; John F Quinn; Michael R Whittaker; Jason S Lewis; Thomas P Davis
Journal:  Theranostics       Date:  2020-01-01       Impact factor: 11.556

10.  A Cleavable C2-Symmetric trans-Cyclooctene Enables Fast and Complete Bioorthogonal Disassembly of Molecular Probes.

Authors:  Martin Wilkovitsch; Maximilian Haider; Barbara Sohr; Barbara Herrmann; Jenna Klubnick; Ralph Weissleder; Jonathan C T Carlson; Hannes Mikula
Journal:  J Am Chem Soc       Date:  2020-10-29       Impact factor: 15.419
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