Literature DB >> 21103523

The traceless Staudinger ligation for indirect 18F-radiolabelling.

Laurence Carroll1, Sophie Boldon, Romain Bejot, Jane E Moore, Jérôme Declerck, Véronique Gouverneur.   

Abstract

The Staudinger ligation of phosphine-substituted thioesters with (18)F-fluoroethylazide has been successfully applied to access (18)F-labelled molecules in radiochemical yields superior to 95%; the first fluorous variant of a Staudinger radio-ligation has been validated.

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Year:  2010        PMID： 21103523     DOI： 10.1039/c0ob00564a

Source DB:  PubMed          Journal:  Org Biomol Chem        ISSN： 1477-0520            Impact factor:   3.876


  9 in total

Review 1.  18 F-Labeling of Sensitive Biomolecules for Positron Emission Tomography.

Authors:  Hema S Krishnan; Longle Ma; Neil Vasdev; Steven H Liang
Journal:  Chemistry       Date:  2017-09-01       Impact factor: 5.236

Review 2.  Fluorine-18 patents (2009-2015). Part 2: new radiochemistry.

Authors:  Andrew V Mossine; Stephen Thompson; Allen F Brooks; Alexandra R Sowa; Jason M Miller; Peter Jh Scott
Journal:  Pharm Pat Anal       Date:  2016-09

3.  Light-Activated Staudinger-Bertozzi Ligation within Living Animals.

Authors:  Lisa Shah; Scott T Laughlin; Isaac S Carrico
Journal:  J Am Chem Soc       Date:  2016-04-13       Impact factor: 15.419

Review 4.  Click Chemistry and Radiochemistry: The First 10 Years.

Authors:  Jan-Philip Meyer; Pierre Adumeau; Jason S Lewis; Brian M Zeglis
Journal:  Bioconjug Chem       Date:  2016-11-22       Impact factor: 4.774

Review 5.  The growing impact of bioorthogonal click chemistry on the development of radiopharmaceuticals.

Authors:  Dexing Zeng; Brian M Zeglis; Jason S Lewis; Carolyn J Anderson
Journal:  J Nucl Med       Date:  2013-04-24       Impact factor: 10.057

6.  The inverse electron-demand Diels-Alder reaction as a new methodology for the synthesis of 225Ac-labelled radioimmunoconjugates.

Authors:  S Poty; R Membreno; J M Glaser; A Ragupathi; W W Scholz; B M Zeglis; J S Lewis
Journal:  Chem Commun (Camb)       Date:  2018-03-08       Impact factor: 6.222

7.  Towards in vivo imaging of cancer sialylation.

Authors:  Ivan Martinez-Duncker; Roberta Salinas-Marin; Carlos Martinez-Duncker
Journal:  Int J Mol Imaging       Date:  2011-09-19

Review 8.  18F-labelled intermediates for radiosynthesis by modular build-up reactions: newer developments.

Authors:  Johannes Ermert
Journal:  Biomed Res Int       Date:  2014-06-23       Impact factor: 3.411

Review 9.  Fluorine-18 radiochemistry, labeling strategies and synthetic routes.

Authors:  Orit Jacobson; Dale O Kiesewetter; Xiaoyuan Chen
Journal:  Bioconjug Chem       Date:  2014-12-12       Impact factor: 4.774
  9 in total

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