Literature DB >> 28696317

Quinolines block every step of malaria heme crystal growth.

David J Sullivan1,2.   

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Year:  2017        PMID： 28696317      PMCID： PMC5530708          DOI： 10.1073/pnas.1708153114

Source DB:  PubMed          Journal:  Proc Natl Acad Sci U S A        ISSN： 0027-8424            Impact factor:   11.205


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  24 in total

1.  Oriented nucleation of hemozoin at the digestive vacuole membrane in Plasmodium falciparum.

Authors:  Sergey Kapishnikov; Allon Weiner; Eyal Shimoni; Peter Guttmann; Gerd Schneider; Noa Dahan-Pasternak; Ron Dzikowski; Leslie Leiserowitz; Michael Elbaum
Journal:  Proc Natl Acad Sci U S A       Date:  2012-06-28       Impact factor: 11.205

2.  Inhibition by chloroquine of a novel haem polymerase enzyme activity in malaria trophozoites.

Authors:  A F Slater; A Cerami
Journal:  Nature       Date:  1992-01-09       Impact factor: 49.962

3.  Ultrastructural and real-time microscopic changes in P. falciparum-infected red blood cells following treatment with antimalarial drugs.

Authors:  Navakanit Sachanonta; Kesinee Chotivanich; Urai Chaisri; Gareth D H Turner; David J P Ferguson; Nicholas P J Day; Emsri Pongponratn
Journal:  Ultrastruct Pathol       Date:  2011-10       Impact factor: 1.094

4.  Structure-function relationships in aminoquinolines: effect of amino and chloro groups on quinoline-hematin complex formation, inhibition of beta-hematin formation, and antiplasmodial activity.

Authors:  T J Egan; R Hunter; C H Kaschula; H M Marques; A Misplon; J Walden
Journal:  J Med Chem       Date:  2000-01-27       Impact factor: 7.446

5.  Aligned hemozoin crystals in curved clusters in malarial red blood cells revealed by nanoprobe X-ray Fe fluorescence and diffraction.

Authors:  Sergey Kapishnikov; Trine Berthing; Lars Hviid; Martin Dierolf; Andreas Menzel; Franz Pfeiffer; Jens Als-Nielsen; Leslie Leiserowitz
Journal:  Proc Natl Acad Sci U S A       Date:  2012-06-25       Impact factor: 11.205

6.  The structure of malaria pigment beta-haematin.

Authors:  S Pagola; P W Stephens; D S Bohle; A D Kosar; S K Madsen
Journal:  Nature       Date:  2000-03-16       Impact factor: 49.962

7.  The hydroxyl functionality and a rigid proximal N are required for forming a novel non-covalent quinine-heme complex.

Authors:  John N Alumasa; Alexander P Gorka; Leah B Casabianca; Erica Comstock; Angel C de Dios; Paul D Roepe
Journal:  J Inorg Biochem       Date:  2010-09-22       Impact factor: 4.155

Review 8.  Quinoline drug-heme interactions and implications for antimalarial cytostatic versus cytocidal activities.

Authors:  Alexander P Gorka; Angel de Dios; Paul D Roepe
Journal:  J Med Chem       Date:  2013-04-29       Impact factor: 7.446

9.  Zinc protoporphyrin IX binds heme crystals to inhibit the process of crystallization in Plasmodium falciparum.

Authors:  Jayasree K Iyer; Lirong Shi; Anuraj H Shankar; David J Sullivan
Journal:  Mol Med       Date:  2003 May-Aug       Impact factor: 6.354

10.  Hemin lyses malaria parasites.

Authors:  A U Orjih; H S Banyal; R Chevli; C D Fitch
Journal:  Science       Date:  1981-11-06       Impact factor: 47.728
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  11 in total

1.  Insights into structural and physicochemical properties required for β-hematin inhibition of privileged triarylimidazoles.

Authors:  Clinton G L Veale; Janeeka Jayram; Shivani Naidoo; Dustin Laming; Tarryn Swart; Tania Olivier; Matthew P Akerman; Katherine A de Villiers; Heinrich C Hoppe; Vineet Jeena
Journal:  RSC Med Chem       Date:  2019-12-16

Review 2.  Malaria parasite plasmepsins: More than just plain old degradative pepsins.

Authors:  Armiyaw S Nasamu; Alexander J Polino; Eva S Istvan; Daniel E Goldberg
Journal:  J Biol Chem       Date:  2020-05-04       Impact factor: 5.157

3.  Superacid-promoted synthesis of quinoline derivatives.

Authors:  Hein Vuong; Michael R Stentzel; Douglas A Klumpp
Journal:  Tetrahedron Lett       Date:  2020-01-14       Impact factor: 2.415

4.  Antimalarial Natural Products.

Authors:  David G I Kingston; Maria Belen Cassera
Journal:  Prog Chem Org Nat Prod       Date:  2022

5.  Novel Antimalarial Tetrazoles and Amides Active against the Hemoglobin Degradation Pathway in Plasmodium falciparum.

Authors:  Aloysus Lawong; Suraksha Gahalawat; John Okombo; Josefine Striepen; Tomas Yeo; Sachel Mok; Ioanna Deni; Jessica L Bridgford; Hanspeter Niederstrasser; Anwu Zhou; Bruce Posner; Sergio Wittlin; Francisco Javier Gamo; Benigno Crespo; Alisje Churchyard; Jake Baum; Nimisha Mittal; Elizabeth Winzeler; Benoît Laleu; Michael J Palmer; Susan A Charman; David A Fidock; Joseph M Ready; Margaret A Phillips
Journal:  J Med Chem       Date:  2021-02-23       Impact factor: 7.446

6.  Physicochemical Profiling and Comparison of Research Antiplasmodials and Advanced Stage Antimalarials with Oral Drugs.

Authors:  Amritansh Bhanot; Sandeep Sundriyal
Journal:  ACS Omega       Date:  2021-02-25

Review 7.  Structural Insights into Transporter-Mediated Drug Resistance in Infectious Diseases.

Authors:  Jonathan Kim; Rosemary J Cater; Brendon C Choy; Filippo Mancia
Journal:  J Mol Biol       Date:  2021-04-20       Impact factor: 6.151

8.  Structure and drug resistance of the Plasmodium falciparum transporter PfCRT.

Authors:  Jonathan Kim; Yong Zi Tan; Kathryn J Wicht; Satchal K Erramilli; Satish K Dhingra; John Okombo; Jeremie Vendome; Laura M Hagenah; Sabrina I Giacometti; Audrey L Warren; Kamil Nosol; Paul D Roepe; Clinton S Potter; Bridget Carragher; Anthony A Kossiakoff; Matthias Quick; David A Fidock; Filippo Mancia
Journal:  Nature       Date:  2019-11-27       Impact factor: 49.962

Review 9.  Chloroquine and hydroxychloroquine in the treatment of COVID-19: the never-ending story.

Authors:  Amin Gasmi; Massimiliano Peana; Sadaf Noor; Roman Lysiuk; Alain Menzel; Asma Gasmi Benahmed; Geir Bjørklund
Journal:  Appl Microbiol Biotechnol       Date:  2021-01-30       Impact factor: 4.813

Review 10.  Repurposing Chloroquine Against Multiple Diseases With Special Attention to SARS-CoV-2 and Associated Toxicity.

Authors:  Siya Kamat; Madhuree Kumari
Journal:  Front Pharmacol       Date:  2021-04-12       Impact factor: 5.810
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