Literature DB >> 27393274

Pharmacokinetics, Safety, and Efficacy of Chemoembolization with Doxorubicin-Loaded Tightly Calibrated Small Microspheres in Patients with Hepatocellular Carcinoma.

Katerina Malagari1, Theodoros Kiakidis2, Maria Pomoni2, Hippokratis Moschouris2, Emmanouil Emmanouil2, Themis Spiridopoulos2, Vlasios Sotirchos2, Savvas Tandeles2, Dimitrios Koundouras2, Alexios Kelekis2, Dimitrios Filippiadis2, Angelos Charokopakis2, Evanthia Bouma2, Achilles Chatziioannou2, Spyridon Dourakis3, John Koskinas3, Theodoros Karampelas4, Konstantinos Tamvakopoulos4, Nikolaos Kelekis2, Dimitrios Kelekis2.   

Abstract

PURPOSE: This study examines safety, efficacy, and pharmacokinetics of chemoembolization with loadable microspheres ≤100 μm for hepatocellular carcinoma.
MATERIALS AND METHODS: A pilot safety study was performed in 19 patients with size and dose escalation and then 52 patients were enrolled prospectively and randomly assigned to chemoembolization with TANDEM™ loaded with 150 or 100 mg of doxorubicin.
RESULTS: The mean diameter of the tumors was 7.28 ± 2.09 cm (range 4-12) and distribution dominant/multiple 51.9/48.1 %. Child A/B distribution was 32/20 (61.5/38.5 %) and etiology HBV/HCV/HBV/HCV-hemochromatosis was 61.6/9.6/9.6/15.4 %. Twenty-five patients were assigned in the low and 27 in the high loading group. There was 1.92 % thirty-day mortality due to lesion rupture. Biliary damage was seen in 3 patients (5.7 %) in the high loading. Mean maximum plasma concentration of doxorubicin C max ± SD was 284.9 ± 276.2 ng/mL for the high and 108.5 ± 77.6 ng/mL for the low loading (p < 0.001). According to m-RECIST overall objective response after two sessions reached 61.22 and 63.82 % at 6 months. Notably, complete target lesion response (CR) after the second session was observed in 28.57 % and maintained in 23.40 % at 6 months. No statistical differences in the local response rates were observed between the two loading groups. Overall survival (OS) at 6 months, 1 , 2, and 3 years was 98.08, 92.3, 88.46, and 82.6 %, respectively. OS and Progression-Free Survival did not demonstrate statistical significance between the two loading groups.
CONCLUSION: Initial evidence shows that (a) TANDEM™ achieves high rates of local response and mid-term survival, (b) high loading provides no clinical benefit and is associated with biliary toxicity.

Entities:  

Keywords:  Chemoembolization; Drug eluting beads; Hepatocellular carcinoma; Tightly calibrated microspheres

Mesh:

Substances:

Year:  2016        PMID: 27393274     DOI: 10.1007/s00270-016-1382-6

Source DB:  PubMed          Journal:  Cardiovasc Intervent Radiol        ISSN: 0174-1551            Impact factor:   2.740


  13 in total

1.  Association of Chemotherapy for Solid Tumors With Development of Therapy-Related Myelodysplastic Syndrome or Acute Myeloid Leukemia in the Modern Era.

Authors:  Lindsay M Morton; Graça M Dores; Sara J Schonfeld; Martha S Linet; Byron S Sigel; Clara J K Lam; Margaret A Tucker; Rochelle E Curtis
Journal:  JAMA Oncol       Date:  2019-03-01       Impact factor: 31.777

Review 2.  Advances in Biomaterials and Technologies for Vascular Embolization.

Authors:  Jingjie Hu; Hassan Albadawi; Brian W Chong; Amy R Deipolyi; Rahul A Sheth; Ali Khademhosseini; Rahmi Oklu
Journal:  Adv Mater       Date:  2019-06-06       Impact factor: 30.849

Review 3.  Therapy of Intermediate-Stage Hepatocellular Carcinoma: Current Evidence and Clinical Practice.

Authors:  Nathan X Chai; Julius Chapiro
Journal:  Semin Intervent Radiol       Date:  2020-12-11       Impact factor: 1.513

Review 4.  Clinical Pharmacokinetics and Pharmacodynamics of Transarterial Chemoembolization and Targeted Therapies in Hepatocellular Carcinoma.

Authors:  Anne Hulin; Jeanick Stocco; Mohamed Bouattour
Journal:  Clin Pharmacokinet       Date:  2019-08       Impact factor: 6.447

5.  Systematic Review and Pharmacokinetic Meta-analysis of Doxorubicin Exposure in Transcatheter Arterial Chemoembolization and Doxorubicin-Eluted Beads Chemoembolization for Treatment of Unresectable Hepatocellular Carcinoma.

Authors:  Mohammadreza Zarisfi; Arta Kasaeian; Anna Wen; Eleni Liapi
Journal:  Eur J Drug Metab Pharmacokinet       Date:  2022-05-11       Impact factor: 2.441

6.  Unresectable hepatocellular carcinoma treatment with doxorubicin-eluting polyethylene glycol microspheres: a single-center experience.

Authors:  Gerardo Tovar-Felice; Andrés García-Gámez; Virgilio Benito-Santamaría; David Balaguer-Paniagua; Jordi Villalba-Auñón; Jaume Sampere-Moragues
Journal:  Hepat Oncol       Date:  2021-06-04

7.  Transarterial chemoembolization with drug-eluting beads in hepatocellular carcinoma.

Authors:  Hee Chul Nam; Bohyun Jang; Myeong Jun Song
Journal:  World J Gastroenterol       Date:  2016-10-28       Impact factor: 5.742

8.  Safety and Feasibility of Chemoembolization with Doxorubicin-Loaded Small Calibrated Microspheres in Patients with Hepatocellular Carcinoma: Results of the MIRACLE I Prospective Multicenter Study.

Authors:  Götz Richter; Boris Radeleff; Christian Stroszczynski; Philippe Pereira; Thomas Helmberger; Mark Barakat; Peter Huppert
Journal:  Cardiovasc Intervent Radiol       Date:  2017-11-22       Impact factor: 2.740

9.  Initial Transarterial Chemoembolization (TACE) Using HepaSpheres 20-40 µm and Subsequent Lipiodol TACE in Patients with Hepatocellular Carcinoma > 5 cm.

Authors:  Su Min Cho; Hee Ho Chu; Jong Woo Kim; Jin Hyung Kim; Dong Il Gwon
Journal:  Life (Basel)       Date:  2021-04-18

10.  The short-term safety and efficacy of TANDEM microspheres of various sizes and doxorubicin loading concentrations for hepatocellular carcinoma treatment.

Authors:  Chia-Ying Lin; Yi-Sheng Liu; Kuang-Tse Pan; Chia-Bang Chen; Chein-Fu Hung; Chen-Te Chou
Journal:  Sci Rep       Date:  2021-06-10       Impact factor: 4.379

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