Literature DB >> 27159573

Concurrent nuclear ERG and MYC protein overexpression defines a subset of locally advanced prostate cancer: Potential opportunities for synergistic targeted therapeutics.

Aaron M Udager1, Angelo M DeMarzo2, Yang Shi3,4, Jessica L Hicks2, Xuhong Cao4, Javed Siddiqui4, Hui Jiang3, Arul M Chinnaiyan1,4,5,6,7, Rohit Mehra1,4,6.   

Abstract

BACKGROUND: Recurrent ERG gene fusions, the most common genetic alterations in prostate cancer, drive overexpression of the nuclear transcription factor ERG, and are early clonal events in prostate cancer progression. The nuclear transcription factor MYC is also frequently overexpressed in prostate cancer and may play a role in tumor initiation and/or progression. The relationship between nuclear ERG and MYC protein overexpression in prostate cancer, as well as the clinicopathologic characteristics and prognosis of ERG-positive/MYC high tumors, is not well understood.
METHODS: Immunohistochemistry (IHC) for ERG and MYC was performed on formalin-fixed, paraffin-embedded tissue from prostate cancer tissue microarrays (TMAs), and nuclear staining was scored semi-quantitatively (IHC product score range = 0-300). Correlation between nuclear ERG and MYC protein expression and association with clinicopathologic parameters and biochemical recurrence after radical prostatectomy was assessed.
RESULTS: 29.1% of all tumor nodules showed concurrent nuclear ERG and MYC protein overexpression (i.e., ERG-positive/MYC high), including 35.0% of secondary nodules. Overall, there was weak positive correlation between ERG and MYC expression across all tumor nodules (rpb  = 0.149, P = 0.045), although this correlation was strongest in secondary nodules (rpb  = 0.520, P = 0.019). In radical prostatectomy specimens, ERG-positive/MYC high tumors were positively associated with the presence of extraprostatic extension (EPE), relative to all other ERG/MYC expression subgroups, however, there was no significant association between concurrent nuclear ERG and MYC protein overexpression and time to biochemical recurrence.
CONCLUSIONS: Concurrent nuclear ERG and MYC protein overexpression is common in prostate cancer and defines a subset of locally advanced tumors. Recent data indicates that BET bromodomain proteins regulate ERG gene fusion and MYC gene expression in prostate cancer, suggesting possible synergistic targeted therapeutics in ERG-positive/MYC high tumors. Prostate 76:845-853, 2016.
© 2016 Wiley Periodicals, Inc. © 2016 Wiley Periodicals, Inc.

Entities:  

Keywords:  BET bromodomain; ERG; MYC; immunohistochemistry (IHC); prostate cancer

Mesh:

Substances:

Year:  2016        PMID: 27159573      PMCID: PMC4975940          DOI: 10.1002/pros.23175

Source DB:  PubMed          Journal:  Prostate        ISSN: 0270-4137            Impact factor:   4.104


  28 in total

Review 1.  Targeting bromodomains: epigenetic readers of lysine acetylation.

Authors:  Panagis Filippakopoulos; Stefan Knapp
Journal:  Nat Rev Drug Discov       Date:  2014-04-22       Impact factor: 84.694

2.  ERG expression is associated with increased risk of biochemical relapse following radical prostatectomy in early onset prostate cancer.

Authors:  K-C Huang; M Dolph; B Donnelly; T A Bismar
Journal:  Clin Transl Oncol       Date:  2014-05-06       Impact factor: 3.405

Review 3.  Targeting BET bromodomains for cancer treatment.

Authors:  Marie Jung; Kathy A Gelato; Amaury Fernández-Montalván; Stephan Siegel; Bernard Haendler
Journal:  Epigenomics       Date:  2015       Impact factor: 4.778

4.  ERG status is unrelated to PSA recurrence in radically operated prostate cancer in the absence of antihormonal therapy.

Authors:  Sarah Minner; Malaika Enodien; Hüseyin Sirma; Andreas M Luebke; Antje Krohn; Pascale S Mayer; Ronald Simon; Pierre Tennstedt; Julia Müller; Laura Scholz; Jan C Brase; Alvin Y Liu; Hartmut Schlüter; Klaus Pantel; Udo Schumacher; Carsten Bokemeyer; Thomas Steuber; Markus Graefen; Guido Sauter; Thorsten Schlomm
Journal:  Clin Cancer Res       Date:  2011-07-26       Impact factor: 12.531

5.  An immunohistochemical signature comprising PTEN, MYC, and Ki67 predicts progression in prostate cancer patients receiving adjuvant docetaxel after prostatectomy.

Authors:  Emmanuel S Antonarakis; Daniel Keizman; Zhe Zhang; Bora Gurel; Tamara L Lotan; Jessica L Hicks; Helen L Fedor; Michael A Carducci; Angelo M De Marzo; Mario A Eisenberger
Journal:  Cancer       Date:  2012-06-06       Impact factor: 6.860

6.  Therapeutic targeting of BET bromodomain proteins in castration-resistant prostate cancer.

Authors:  Irfan A Asangani; Vijaya L Dommeti; Xiaoju Wang; Rohit Malik; Marcin Cieslik; Rendong Yang; June Escara-Wilke; Kari Wilder-Romans; Sudheer Dhanireddy; Carl Engelke; Mathew K Iyer; Xiaojun Jing; Yi-Mi Wu; Xuhong Cao; Zhaohui S Qin; Shaomeng Wang; Felix Y Feng; Arul M Chinnaiyan
Journal:  Nature       Date:  2014-04-23       Impact factor: 49.962

7.  TMPRSS2-ERG fusion, a common genomic alteration in prostate cancer activates C-MYC and abrogates prostate epithelial differentiation.

Authors:  C Sun; A Dobi; A Mohamed; H Li; R L Thangapazham; B Furusato; S Shaheduzzaman; S-H Tan; G Vaidyanathan; E Whitman; D J Hawksworth; Y Chen; M Nau; V Patel; M Vahey; J S Gutkind; T Sreenath; G Petrovics; I A Sesterhenn; D G McLeod; S Srivastava
Journal:  Oncogene       Date:  2008-06-09       Impact factor: 9.867

8.  Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia.

Authors:  Mark A Dawson; Rab K Prinjha; Antje Dittmann; George Giotopoulos; Marcus Bantscheff; Wai-In Chan; Samuel C Robson; Chun-wa Chung; Carsten Hopf; Mikhail M Savitski; Carola Huthmacher; Emma Gudgin; Dave Lugo; Soren Beinke; Trevor D Chapman; Emma J Roberts; Peter E Soden; Kurt R Auger; Olivier Mirguet; Konstanze Doehner; Ruud Delwel; Alan K Burnett; Phillip Jeffrey; Gerard Drewes; Kevin Lee; Brian J P Huntly; Tony Kouzarides
Journal:  Nature       Date:  2011-10-02       Impact factor: 49.962

9.  Inhibition of BET bromodomain proteins as a therapeutic approach in prostate cancer.

Authors:  Anastasia Wyce; Yan Degenhardt; Yuchen Bai; BaoChau Le; Susan Korenchuk; Ming-Chih Crouthame; Charles F McHugh; Robert Vessella; Caretha L Creasy; Peter J Tummino; Olena Barbash
Journal:  Oncotarget       Date:  2013-12

10.  A novel RNA in situ hybridization assay for the long noncoding RNA SChLAP1 predicts poor clinical outcome after radical prostatectomy in clinically localized prostate cancer.

Authors:  Rohit Mehra; Yang Shi; Aaron M Udager; John R Prensner; Anirban Sahu; Matthew K Iyer; Javed Siddiqui; Xuhong Cao; John Wei; Hui Jiang; Felix Y Feng; Arul M Chinnaiyan
Journal:  Neoplasia       Date:  2014-12       Impact factor: 5.715

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  4 in total

1.  MYC Overexpression at the Protein and mRNA Level and Cancer Outcomes among Men Treated with Radical Prostatectomy for Prostate Cancer.

Authors:  Andreas Pettersson; Travis Gerke; Kathryn L Penney; Rosina T Lis; Edward C Stack; Nelma Pértega-Gomes; Giorgia Zadra; Svitlana Tyekucheva; Edward L Giovannucci; Lorelei A Mucci; Massimo Loda
Journal:  Cancer Epidemiol Biomarkers Prev       Date:  2017-11-15       Impact factor: 4.254

2.  Leveraging artificial intelligence to predict ERG gene fusion status in prostate cancer.

Authors:  Vipulkumar Dadhania; Daniel Gonzalez; Mustafa Yousif; Jerome Cheng; Todd M Morgan; Daniel E Spratt; Zachery R Reichert; Rahul Mannan; Xiaoming Wang; Anya Chinnaiyan; Xuhong Cao; Saravana M Dhanasekaran; Arul M Chinnaiyan; Liron Pantanowitz; Rohit Mehra
Journal:  BMC Cancer       Date:  2022-05-05       Impact factor: 4.638

3.  cMYC expression in thyroid follicular cell-derived carcinomas: a role in thyroid tumorigenesis.

Authors:  Hany I Sakr; Deborah J Chute; Christian Nasr; Charles D Sturgis
Journal:  Diagn Pathol       Date:  2017-10-03       Impact factor: 2.644

4.  The Role of Immunohistochemical Analysis as a Tool for the Diagnosis, Prognostic Evaluation and Treatment of Prostate Cancer: A Systematic Review of the Literature.

Authors:  Arie Carneiro; Álan Roger Gomes Barbosa; Lucas Seiti Takemura; Paulo Priante Kayano; Natasha Kouvaleski Saviano Moran; Carolina Ko Chen; Marcelo Langer Wroclawski; Gustavo Caserta Lemos; Isabela Werneck da Cunha; Marcos Takeo Obara; Marcos Tobias-Machado; Adam G Sowalsky; Bianca Bianco
Journal:  Front Oncol       Date:  2018-09-18       Impact factor: 6.244

  4 in total

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