Literature DB >> 26213141

Phase II study of an AKT inhibitor MK2206 in patients with relapsed or refractory lymphoma.

Yasuhiro Oki1, Michelle Fanale1, Jorge Romaguera1, Luis Fayad1, Nathan Fowler1, Amanda Copeland1, Felipe Samaniego1, Larry W Kwak1, Sattva Neelapu1, Michael Wang1, Lei Feng2, Anas Younes1.   

Abstract

We conducted a phase II study of the AKT inhibitor, MK2206 in patients with relapsed or refractory lymphoma of any histology excluding Burkitt lymphoma or lymphoblastic lymphoma. MK-2206 was administered orally at 200 mg once weekly in 28-d cycles up to 12 cycles in the absence of progression or significant toxicity. The dose was adjusted based on tolerance. A total of 59 patients were enrolled. The final doses patients received were 300 mg (n = 33), 250 mg (n = 2), 200 mg (n = 16) and 135 mg (n = 8). Based on intent-to-treat analysis, objective response was observed in 8 (14%) patients (2 complete response and 6 partial response), with median response duration of 5·8 months. The overall response rate was 20% in 25 patients with classical Hodgkin lymphoma. Rash was the most common toxicity (any grade 53%, Grade 3 in 15%) and was observed in a dose-dependent manner. The correlative cytokine analysis showed paradoxical increase in several cytokines, which may be explained by negative feedback mechanism induced by the on-target effect of AKT inhibitor. Our data demonstrate that MK2206 has a favourable safety profile with a modest activity in patients with relapsed Hodgkin lymphoma. The future studies should explore mechanism-based combinations (clinicaltrials.gov NCT01258998).
© 2015 John Wiley & Sons Ltd.

Entities:  

Keywords:  AKT; clinical trials; lymphoma; target therapy

Mesh:

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Year:  2015        PMID: 26213141      PMCID: PMC5278973          DOI: 10.1111/bjh.13603

Source DB:  PubMed          Journal:  Br J Haematol        ISSN: 0007-1048            Impact factor:   6.998


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