Literature DB >> 25560207

Intratesticular, intraperitoneal, and oral administration of thienopyrimidine derivatives increases the testosterone level in male rats.

K V Derkach1, D V Dar'in, P S Lobanov, A O Shpakov.   

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Year:  2015        PMID： 25560207     DOI： 10.1134/S0012496614060040

Source DB:  PubMed          Journal:  Dokl Biol Sci        ISSN： 0012-4966


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  10 in total

1.  The first orally active low molecular weight agonists for the LH receptor: thienopyr(im)idines with therapeutic potential for ovulation induction.

Authors:  N C R van Straten; G G Schoonus-Gerritsma; R G van Someren; J Draaijer; A E P Adang; C M Timmers; R G J M Hanssen; C A A van Boeckel
Journal:  Chembiochem       Date:  2002-10-04       Impact factor: 3.164

2.  Determination of different putative allosteric binding pockets at the lutropin receptor by using diverse drug-like low molecular weight ligands.

Authors:  Laura H Heitman; Gunnar Kleinau; Johannes Brussee; Gerd Krause; Adriaan P Ijzerman
Journal:  Mol Cell Endocrinol       Date:  2012-01-18       Impact factor: 4.102

Review 3.  [Low-molecular regulators of polypeptide hormones receptors containing LGR repeats].

Authors:  A O Shpakov; E A Shpakova
Journal:  Biomed Khim       Date:  2010 May-Jun

4.  Does gonadotropin receptor complex have an amplifying role in cAMP/testosterone production in Leydig cells?

Authors:  E S Browne; V K Bhalla
Journal:  J Androl       Date:  1991 Mar-Apr

Review 5.  [Structural-functional organization of polypeptide hormones receptors containing LRR-repeats and their interaction with heterotrimeric G proteins].

Authors:  A O Shpakov
Journal:  Tsitologiia       Date:  2009

6.  The stimulating influence of thienopyrimidine compounds on the adenylyl cyclase signaling systems in the rat testes.

Authors:  A O Shpakov; D V Dar'in; K V Derkach; P S Lobanov
Journal:  Dokl Biochem Biophys       Date:  2014-07-04       Impact factor: 0.788

7.  [Activation of adenylyl cyclase in rats testes and ovaries using thienopyrimidine derivatives].

Authors:  A O Shpakov; K V Derkach; D V Dar'in; P S Lobanov
Journal:  Tsitologiia       Date:  2014

8.  [3H]Org 43553, the first low-molecular-weight agonistic and allosteric radioligand for the human luteinizing hormone receptor.

Authors:  Laura H Heitman; Julia Oosterom; Kimberly M Bonger; Cornelis M Timmers; Peter H G Wiegerinck; Adriaan P Ijzerman
Journal:  Mol Pharmacol       Date:  2007-11-07       Impact factor: 4.436

Review 9.  G protein-coupled receptors of the hypothalamic-pituitary-gonadal axis: a case for Gnrh, LH, FSH, and GPR54 receptor ligands.

Authors:  Laura H Heitman; Adriaan P Ijzerman
Journal:  Med Res Rev       Date:  2008-11       Impact factor: 12.944

Review 10.  Structure-function relationships of the luteinizing hormone receptor.

Authors:  David Puett; Yongsheng Li; Krassimira Angelova; Geneva Demars; Thomas P Meehan; Francesca Fanelli; Prema Narayan
Journal:  Ann N Y Acad Sci       Date:  2005-12       Impact factor: 5.691
  10 in total

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