Literature DB >> 24104417

Novel thrombin and factor Xa inhibitors: challenges to reversal of their anticoagulation effects.

Sean Yates1, Ravi Sarode.   

Abstract

PURPOSE OF REVIEW: Warfarin has been the sole oral anticoagulant used in the management of thromboembolic disorders for over 60 years. Target-specific oral anticoagulants (TSOAs) have recently emerged as alternatives to warfarin, because they do not require laboratory monitoring. Nevertheless, with the rising use of TSOAs, there is growing concern among clinicians regarding management of bleeding in patients taking them. Unlike warfarin, there is no antidote or reversal agent for TSOAs. This review summarizes recent developments and attempts to provide a systematic approach to patients on TSOAs presenting with bleeding complications. RECENT
FINDINGS: Currently, data involving clinical management of TSOAs are limited and primarily based on ex-vivo or animal models using hemostatic agents with uncertain implications in bleeding patients. There is a pressing need for randomized clinical trials evaluating the safety and efficacy of hemostatic agents.
SUMMARY: Without evidence-based guidelines for TSOA management, appropriate patient care requires an understanding of TSOA pharmacology, their effect on coagulation tests and, hence, a correct interpretation of test results, as well as a systematic approach to bleeding complications.

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Year:  2013        PMID: 24104417     DOI: 10.1097/MOH.0b013e328365a164

Source DB:  PubMed          Journal:  Curr Opin Hematol        ISSN: 1065-6251            Impact factor:   3.284


  6 in total

1.  Allosteric inhibition of factor XIa. Sulfated non-saccharide glycosaminoglycan mimetics as promising anticoagulants.

Authors:  Rami A Al-Horani; David Gailani; Umesh R Desai
Journal:  Thromb Res       Date:  2015-04-22       Impact factor: 3.944

2.  Therapeutic Plasma Exchange for Urgent Rivaroxaban Reversal.

Authors:  Varun Kumar; Joseph Allencherril; Arthur Bracey; Alice J Chen; Wilson W Lam
Journal:  Tex Heart Inst J       Date:  2018-04-07

Review 3.  Hematoma Expansion Following Intracerebral Hemorrhage: Mechanisms Targeting the Coagulation Cascade and Platelet Activation.

Authors:  Sherrefa R Burchell; Jiping Tang; John H Zhang
Journal:  Curr Drug Targets       Date:  2017       Impact factor: 3.465

4.  Plasma Exchange for Urgent Apixaban Reversal in a Case of Hemorrhagic Tamponade after Pacemaker Implantation.

Authors:  Wilson W Lam; Meredith A Reyes; John J Seger
Journal:  Tex Heart Inst J       Date:  2015-08-01

5.  Designing allosteric inhibitors of factor XIa. Lessons from the interactions of sulfated pentagalloylglucopyranosides.

Authors:  Rami A Al-Horani; Umesh R Desai
Journal:  J Med Chem       Date:  2014-05-29       Impact factor: 7.446

6.  Influence of ABCB1 Gene Polymorphism on Rivaroxaban Blood Concentration and Hemorrhagic Events in Patients With Atrial Fibrillation.

Authors:  Yan Wang; Min Chen; Hui Chen; Fang Wang
Journal:  Front Pharmacol       Date:  2021-04-14       Impact factor: 5.810

  6 in total

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