Literature DB >> 22941286

Natural products possessing protein tyrosine phosphatase 1B (PTP1B) inhibitory activity found in the last decades.

Cheng-Shi Jiang1, Lin-fu Liang, Yue-wei Guo.   

Abstract

This article provides an overview of approximately 300 secondary metabolites with inhibitory activity against protein tyrosine phosphatase 1B (PTP1B), which were isolated from various natural sources or derived from synthetic process in the last decades. The structure-activity relationship and the selectivity of some compounds against other protein phosphatases were also discussed. Potential pharmaceutical applications of several PTP1B inhibitors were presented.

Entities:  

Mesh：

Substances：

Year:  2012        PMID： 22941286      PMCID： PMC4002712          DOI： 10.1038/aps.2012.90

Source DB:  PubMed          Journal:  Acta Pharmacol Sin        ISSN： 1671-4083            Impact factor:   6.150


  134 in total

1.  Inhibition of PTP1B by metabolites from Micromucor ramannianus var. angulisporus CRM000232.

Authors:  Hyuncheol Oh; Beom Seok Kim; Eun Young Bae; Min Soo Kim; Bo Yeon Kim; Hyang Burm Lee; Chang-Jin Kim; Jong Seog Ahn
Journal:  J Antibiot (Tokyo)       Date:  2004-08       Impact factor: 2.649

2.  Water-soluble constituents of the root barks of Fraxinus rhynchophylla (Chinese drug Qinpi).

Authors:  Kai Xiao; Qing-Hong Song; Shu-Wei Zhang; Li-Jiang Xuan
Journal:  J Asian Nat Prod Res       Date:  2008 Jan-Feb       Impact factor: 1.569

3.  Solution-phase and solid-phase syntheses of enzyme inhibitor RK-682 and antibiotic agglomerins.

Authors:  Rainer Schobert; Carsten Jagusch
Journal:  J Org Chem       Date:  2005-07-22       Impact factor: 4.354

4.  Synthesis and biological evaluation of oleanolic acid derivatives as inhibitors of protein tyrosine phosphatase 1B.

Authors:  Shan Qian; Haijiao Li; Yin Chen; Weiyu Zhang; Shengyong Yang; Yong Wu
Journal:  J Nat Prod       Date:  2010-10-21       Impact factor: 4.050

5.  Novel and therapeutic effect of caffeic acid and caffeic acid phenyl ester on hepatocarcinoma cells: complete regression of hepatoma growth and metastasis by dual mechanism.

Authors:  Tae-Wook Chung; Sung-Kwon Moon; Young-Chae Chang; Jeong-Heon Ko; Young-Choon Lee; Gun Cho; Soo-Hyun Kim; Jong-Guk Kim; Cheorl-Ho Kim
Journal:  FASEB J       Date:  2004-11       Impact factor: 5.191

6.  Novel synthesis of flavonoids of Scutellaria baicalensis Georgi.

Authors:  Wen-Hsin Huang; Pei-Yu Chien; Ching-Huey Yang; An-Rong Lee
Journal:  Chem Pharm Bull (Tokyo)       Date:  2003-03       Impact factor: 1.645

7.  Cellular effects of small molecule PTP1B inhibitors on insulin signaling.

Authors:  Laiping Xie; Seung-Yub Lee; Jannik N Andersen; Steve Waters; Kui Shen; Xiao-Ling Guo; Niels Peter H Moller; Jerrold M Olefsky; David S Lawrence; Zhong-Yin Zhang
Journal:  Biochemistry       Date:  2003-11-11       Impact factor: 3.162

8.  Synthesis and antimicrobial activities of halogenated bis(hydroxyphenyl)methanes.

Authors:  Ki-Bong Oh; Ji Hye Lee; Jong Wook Lee; Kyung-Mi Yoon; Soon-Chun Chung; Heung Bae Jeon; Jongheon Shin; Hyi-Seung Lee
Journal:  Bioorg Med Chem Lett       Date:  2008-11-27       Impact factor: 2.823

Review 9.  Dietary fats and prevention of type 2 diabetes.

Authors:  Ulf Risérus; Walter C Willett; Frank B Hu
Journal:  Prog Lipid Res       Date:  2008-11-07       Impact factor: 16.195

10.  Synthesis of (+)-nocardione A--use of formal radical cyclization onto a benzene ring.

Authors:  Derrick L J Clive; Stephen P Fletcher
Journal:  Chem Commun (Camb)       Date:  2003-10-07       Impact factor: 6.222
View more
  36 in total

1.  Biphenyl ether derivatives with protein tyrosine phosphatase 1B inhibitory activity from the freshwater fungus Phoma sp.

Authors:  Deiske A Sumilat; Hiroyuki Yamazaki; Syu-Ichi Kanno; Ryo Saito; Yuta Watanabe; Michio Namikoshi
Journal:  J Antibiot (Tokyo)       Date:  2017-01-11       Impact factor: 2.649

2.  A 2,4'-linked tetrahydroxanthone dimer with protein tyrosine phosphatase 1B inhibitory activity from the Okinawan freshwater Aspergillus sp.

Authors:  Henki Rotinsulu; Hiroyuki Yamazaki; Tomohito Miura; Satomi Chiba; Defny S Wewengkang; Deiske A Sumilat; Michio Namikoshi
Journal:  J Antibiot (Tokyo)       Date:  2017-06-28       Impact factor: 2.649

3.  Protein tyrosine phosphatase 1B inhibitory properties of seco-cucurbitane triterpenes obtained from fruiting bodies of Russula lepida.

Authors:  Wilmar Maarisit; Hiroyuki Yamazaki; Syu-Ichi Kanno; Ayako Tomizawa; Jong-Soo Lee; Michio Namikoshi
Journal:  J Nat Med       Date:  2016-11-19       Impact factor: 2.343

4.  Cladosporamide A, a new protein tyrosine phosphatase 1B inhibitor, produced by an Indonesian marine sponge-derived Cladosporium sp.

Authors:  Henki Rotinsulu; Hiroyuki Yamazaki; Shino Sugai; Natsuki Iwakura; Defny S Wewengkang; Deiske A Sumilat; Michio Namikoshi
Journal:  J Nat Med       Date:  2018-03-05       Impact factor: 2.343

Review 5.  Covalent inhibition of protein tyrosine phosphatases.

Authors:  Kasi Viswanatharaju Ruddraraju; Zhong-Yin Zhang
Journal:  Mol Biosyst       Date:  2017-06-27

6.  Trichoketides A and B, two new protein tyrosine phosphatase 1B inhibitors from the marine-derived fungus Trichoderma sp.

Authors:  Hiroyuki Yamazaki; Ryo Saito; Ohgi Takahashi; Ryota Kirikoshi; Kengo Toraiwa; Kohei Iwasaki; Yuta Izumikawa; Wataru Nakayama; Michio Namikoshi
Journal:  J Antibiot (Tokyo)       Date:  2015-04-22       Impact factor: 2.649

Review 7.  Chemical and Biological Aspects of Extracts from Medicinal Plants with Antidiabetic Effects.

Authors:  Lucas F Gushiken; Fernando P Beserra; Ariane L Rozza; Patrícia L Bérgamo; Danilo A Bérgamo; Cláudia H Pellizzon
Journal:  Rev Diabet Stud       Date:  2016-08-10

8.  PAIN-less identification and evaluation of small molecule inhibitors against protein tyrosine phosphatase 1B.

Authors:  Hamid R Nasiri; Philipp Mracek; Steffen K Grimm; Janine Gastaldello; Adrian Kolodzik; Dirk Ullmann
Journal:  Medchemcomm       Date:  2017-04-07       Impact factor: 3.597

9.  Design, synthesis and antimicrobial activity of usnic acid derivatives.

Authors:  Kartsev Victor; Lichitsky Boris; Geronikaki Athina; Petrou Anthi; Smiljkovic Marija; Kostic Marina; Radanovic Oliver; Soković Marina
Journal:  Medchemcomm       Date:  2018-04-11       Impact factor: 3.597

Review 10.  Phytochemicals as Potential Epidrugs in Type 2 Diabetes Mellitus.

Authors:  Karina Ramírez-Alarcón; Montserrat Victoriano; Lorena Mardones; Marcelo Villagran; Ahmed Al-Harrasi; Ahmed Al-Rawahi; Natália Cruz-Martins; Javad Sharifi-Rad; Miquel Martorell
Journal:  Front Endocrinol (Lausanne)       Date:  2021-06-01       Impact factor: 5.555
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.