Literature DB >> 22717269

Pharmacokinetics of the etonogestrel contraceptive implant in obese women.

Sara Mornar1, Lingtak-Neander Chan, Stephanie Mistretta, Amy Neustadt, Summer Martins, Melissa Gilliam.   

Abstract

OBJECTIVE: We sought to examine the pharmacokinetics and acceptability of the etonogestrel contraceptive implant in obese women. STUDY
DESIGN: We developed and validated a plasma etonogestrel concentration assay and enrolled 13 obese (body mass index ≥30) women and 4 normal-weight (body mass index <25) women, who ensured comparability with historical controls. Etonogestrel concentrations were measured at 50-hour intervals through 300 hours postinsertion, then at 3 and 6 months to establish a pharmacokinetic curve.
RESULTS: All obese participants were African American, while all normal-weight participants were white. Across time, the plasma etonogestrel concentrations in obese women were lower than published values for normal-weight women and 31-63% lower than in the normal-weight study cohort, although these differences were not statistically significant. The implant device was found highly acceptable among obese women.
CONCLUSION: Obese women have lower plasma etonogestrel concentration than normal-weight women in the first 6 months after implant insertion. These findings should not be interpreted as decreased contraceptive effectiveness without additional considerations.
Copyright © 2012 Mosby, Inc. All rights reserved.

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Year:  2012        PMID: 22717269     DOI: 10.1016/j.ajog.2012.05.002

Source DB:  PubMed          Journal:  Am J Obstet Gynecol        ISSN: 0002-9378            Impact factor:   8.661


  15 in total

1.  Prolonged use of the etonogestrel implant and levonorgestrel intrauterine device: 2 years beyond Food and Drug Administration-approved duration.

Authors:  Colleen McNicholas; Erin Swor; Leping Wan; Jeffrey F Peipert
Journal:  Am J Obstet Gynecol       Date:  2017-01-29       Impact factor: 8.661

Review 2.  Contraception and the obese woman.

Authors:  Elizabeth Reifsnider; Nonie Mendias; Yolanda Davila; Jennie Bever Babendure
Journal:  J Am Assoc Nurse Pract       Date:  2013-02-27       Impact factor: 1.165

Review 3.  Hormonal Contraception and HIV-1 Acquisition: Biological Mechanisms.

Authors:  Janet P Hapgood; Charu Kaushic; Zdenek Hel
Journal:  Endocr Rev       Date:  2018-02-01       Impact factor: 19.871

Review 4.  Obesity and contraception.

Authors:  Sheila K Mody; Michelle Han
Journal:  Clin Obstet Gynecol       Date:  2014-09       Impact factor: 2.190

5.  Efavirenz decreases etonogestrel exposure: a pharmacokinetic evaluation of implantable contraception with antiretroviral therapy.

Authors:  Catherine A Chappell; Mohammed Lamorde; Shadia Nakalema; Beatrice A Chen; Hope Mackline; Sharon A Riddler; Susan E Cohn; Kristin M Darin; Sharon L Achilles; Kimberly K Scarsi
Journal:  AIDS       Date:  2017-09-10       Impact factor: 4.177

Review 6.  A Review of the Toxicologic Implications of Obesity.

Authors:  Matthew Zuckerman; Howard A Greller; Kavita M Babu
Journal:  J Med Toxicol       Date:  2015-09

Review 7.  Obesity and hormonal contraceptive efficacy.

Authors:  Jennifer A Robinson; Anne E Burke
Journal:  Womens Health (Lond)       Date:  2013-09

8.  Superoxide dismutase 1 overexpression in mice abolishes maternal diabetes-induced endoplasmic reticulum stress in diabetic embryopathy.

Authors:  Fang Wang; E Albert Reece; Peixin Yang
Journal:  Am J Obstet Gynecol       Date:  2013-06-20       Impact factor: 8.661

9.  Relationship between patient characteristics and serum etonogestrel concentrations in contraceptive implant users.

Authors:  Aaron Lazorwitz; Christina L Aquilante; Jeanelle Sheeder; Maryam Guiahi; Stephanie Teal
Journal:  Contraception       Date:  2019-04-10       Impact factor: 3.375

Review 10.  Clarification of contraceptive drug pharmacokinetics in obesity.

Authors:  William J Jusko
Journal:  Contraception       Date:  2016-08-16       Impact factor: 3.375

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