Literature DB >> 22093758

Synthesis and biological activity of dihydroimidazole and 3,4-dihydrobenzo[4,5]imidazo[1,2-a][1,3,5]triazins.

Ahmed M Soliman1, Shaaban K Mohamed, Mahmoud A A El Remaily, H Abdel-Ghany.   

Abstract

Reaction of 2-guanidinobenzimidazole with halogenated active methylenes and ketones gave dihydroimidazole and 3,4-dihydrobenzo[4,5]imidazo [1,2-a][1,3,5]triazin derivatives in very good yield. The anti-bacterial evaluation of the newly synthesized products against broad spectrum of bacteria was performed. Most of products showed high inhibitory effect. All compounds have been characterized based on IR, (1)H NMR, (13)C NMR and Mass spectra.
Copyright © 2011 Elsevier Masson SAS. All rights reserved.

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Year:  2011        PMID： 22093758     DOI： 10.1016/j.ejmech.2011.10.034

Source DB:  PubMed          Journal:  Eur J Med Chem        ISSN： 0223-5234            Impact factor:   6.514


  9 in total

Review 1.  Nitrogen-Containing Heterocyclic Compounds Obtained from Monoterpenes or Their Derivatives: Synthesis and Properties.

Authors:  Vladimir V Chernyshov; Irina I Popadyuk; Olga I Yarovaya; Nariman F Salakhutdinov
Journal:  Top Curr Chem (Cham)       Date:  2022-08-11

2.  2-(4-Isobutyl-phen-yl)-N'-[(3Z)-2-oxoindolin-3-yl-idene]propano-hydrazide.

Authors:  Shaaban K Mohamed; Mehmet Akkurt; Mustafa R Albayati; Kuldip Singh; Herman Potgieter
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-03-28

3.  2-Anilino-3-(2-hy-droxy-prop-yl)-4-methyl-1,3-thia-zol-3-ium chloride.

Authors:  Shaaban K Mohamed; Mehmet Akkurt; Muhammad N Tahir; Antar A Abdelhamid; Ali N Khalilov
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-05-26

4.  2-Amino-6-(dimethyl-amino)pyridine-3,5-dicarbonitrile.

Authors:  Shaaban K Mohamed; Ahmed M Soliman; Eman M M Abdel-Raheem; Sohail Saeed; Wing-Tak Wong
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-04-25

5.  2-(Piperidin-1-yl)-6-(1H-pyrrol-1-yl)pyridine-3,5-dicarbonitrile.

Authors:  Peter N Horton; Shaaban K Mohamed; Ahmed M Soliman; Eman M M Abdel-Raheem; Mehmet Akkurt
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-03-03

6.  Synthesis and Toxicological Effect of Some New Pyrrole Derivatives as Prospective Insecticidal Agents against the Cotton Leafworm, Spodoptera littoralis (Boisduval).

Authors:  Antar A Abdelhamid; Kaoud S M Salama; Ahmed M Elsayed; Mohamed A Gad; Mahmoud Abd El Aleem Ali Ali El-Remaily
Journal:  ACS Omega       Date:  2022-01-25

7.  4-(1-Allyl-4,5-diphenyl-1H-imidazol-2-yl)-N,N-dimethyl-aniline.

Authors:  Mehmet Akkurt; Frank R Fronczek; Shaaban K Mohamed; Avtandil H Talybov; Adel A E Marzouk; Antar A Abdelhamid
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2013-03-09

8.  2-Eth-oxy-4-(4-methyl-phen-yl)-6-phenyl-pyridine-3-carbonitrile.

Authors:  Shaaban K Mohamed; Mehmet Akkurt; Antar A Abdelhamid; Kuldip Singh; Mahoud A A El-Remaily
Journal:  Acta Crystallogr Sect E Struct Rep Online       Date:  2012-07-18

9.  Green Method for the Synthetic Ugi Reaction by Twin Screw Extrusion without a Solvent and Catalyst.

Authors:  Mahmoud Abd El Aleem Ali Ali El-Remaily; Ahmed M M Soliman; Omar M Elhady
Journal:  ACS Omega       Date:  2020-03-12
  9 in total

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