Literature DB >> 21919140

Targeting histone lysine demethylases by truncating the histone 3 tail to obtain selective substrate-based inhibitors.

Brian Lohse1, Anders L Nielsen, Jan B L Kristensen, Charlotte Helgstrand, Paul A C Cloos, Lars Olsen, Michael Gajhede, Rasmus P Clausen, Jesper L Kristensen.   

Abstract

Mesh：

Substances：

Year:  2011        PMID： 21919140     DOI： 10.1002/anie.201101849

Source DB:  PubMed          Journal:  Angew Chem Int Ed Engl        ISSN： 1433-7851            Impact factor:   15.336


× No keyword cloud information.
  11 in total

Review 1.  Small molecule epigenetic inhibitors targeted to histone lysine methyltransferases and demethylases.

Authors:  Zhanxin Wang; Dinshaw J Patel
Journal:  Q Rev Biophys       Date:  2013-09-02       Impact factor: 5.318

Review 2.  The role of histone demethylases in cancer therapy.

Authors:  Inga Hoffmann; Martin Roatsch; Martin L Schmitt; Luca Carlino; Martin Pippel; Wolfgang Sippl; Manfred Jung
Journal:  Mol Oncol       Date:  2012-08-07       Impact factor: 6.603

Review 3.  Recent Advances with KDM4 Inhibitors and Potential Applications.

Authors:  Qiong Wu; Brandon Young; Yan Wang; Andrew M Davidoff; Zoran Rankovic; Jun Yang
Journal:  J Med Chem       Date:  2022-07-15       Impact factor: 8.039

Review 4.  Histone Modifications and Cancer.

Authors:  James E Audia; Robert M Campbell
Journal:  Cold Spring Harb Perspect Biol       Date:  2016-04-01       Impact factor: 10.005

5.  Quantitative analysis of histone demethylase probes using fluorescence polarization.

Authors:  Wenqing Xu; Jessica D Podoll; Xuan Dong; Anthony Tumber; Udo Oppermann; Xiang Wang
Journal:  J Med Chem       Date:  2013-06-13       Impact factor: 7.446

6.  Development of substrate-selective probes for affinity pulldown of histone demethylases.

Authors:  Laura J Marholz; Le Chang; William M Old; Xiang Wang
Journal:  ACS Chem Biol       Date:  2014-10-29       Impact factor: 5.100

Review 7.  Targeting histone lysine demethylases - progress, challenges, and the future.

Authors:  Cyrille C Thinnes; Katherine S England; Akane Kawamura; Rasheduzzaman Chowdhury; Christopher J Schofield; Richard J Hopkinson
Journal:  Biochim Biophys Acta       Date:  2014-05-21

8.  Posttranslational modifications of the histone 3 tail and their impact on the activity of histone lysine demethylases in vitro.

Authors:  Brian Lohse; Charlotte Helgstrand; Jan B L Kristensen; Ulrike Leurs; Paul A C Cloos; Jesper L Kristensen; Rasmus P Clausen
Journal:  PLoS One       Date:  2013-07-02       Impact factor: 3.240

9.  Identification of the KDM2/7 histone lysine demethylase subfamily inhibitor and its antiproliferative activity.

Authors:  Takayoshi Suzuki; Hiroki Ozasa; Yukihiro Itoh; Peng Zhan; Hideyuki Sawada; Koshiki Mino; Louise Walport; Rei Ohkubo; Akane Kawamura; Masato Yonezawa; Yuichi Tsukada; Anthony Tumber; Hidehiko Nakagawa; Makoto Hasegawa; Ryuzo Sasaki; Tamio Mizukami; Christopher J Schofield; Naoki Miyata
Journal:  J Med Chem       Date:  2013-09-05       Impact factor: 7.446

10.  Substrate- and cofactor-independent inhibition of histone demethylase KDM4C.

Authors:  Ulrike Leurs; Brian Lohse; Kasper D Rand; Shonoi Ming; Erik S Riise; Philip A Cole; Jesper L Kristensen; Rasmus P Clausen
Journal:  ACS Chem Biol       Date:  2014-07-17       Impact factor: 5.100
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.