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Literature DB >> 20575134

Cross-linked peptoid-based dimerization inhibitors of HIV-1 protease.

Song-Gil Lee¹, Jean Chmielewski.

Abstract

Entities: Chemical Disease Gene Species

Mesh：

Substances：

Year: 2010 PMID： 20575134 PMCID： PMC4441096 DOI： 10.1002/cbic.201000248

Source DB: PubMed Journal: Chembiochem ISSN： 1439-4227 Impact factor: 3.164

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20 in total

Review 1. Novel strategies for targeting the dimerization interface of HIV protease with cross-linked interfacial peptides.

Authors: Michael J Bowman; Jean Chmielewski
Journal: Biopolymers Date: 2002 Impact factor: 2.505

Review 2. Targeting protein-protein interactions by rational design: mimicry of protein surfaces.

Authors: Steven Fletcher; Andrew D Hamilton
Journal: J R Soc Interface Date: 2006-04-22 Impact factor: 4.118

3. Dissociative inhibition of dimeric enzymes. Kinetic characterization of the inhibition of HIV-1 protease by its COOH-terminal tetrapeptide.

Authors: Z Y Zhang; R A Poorman; L L Maggiora; R L Heinrikson; F J Kézdy
Journal: J Biol Chem Date: 1991-08-25 Impact factor: 5.157

Review 4. Peptoid architectures: elaboration, actuation, and application.

Authors: Barney Yoo; Kent Kirshenbaum
Journal: Curr Opin Chem Biol Date: 2008-09-09 Impact factor: 8.822

5. Examples of peptide-peptoid hybrid serine protease inhibitors based on the trypsin inhibitor SFTI-1 with complete protease resistance at the P1-P1' reactive site.

Authors: Maciej Stawikowski; Roma Stawikowska; Anna Jaśkiewicz; Ewa Zabłotna; Krzysztof Rolka
Journal: Chembiochem Date: 2005-06 Impact factor: 3.164

6. A simple, continuous fluorometric assay for HIV protease.

Authors: M V Toth; G R Marshall
Journal: Int J Pept Protein Res Date: 1990-12

Review 7. HIV-1 protease inhibitors. A review for clinicians.

Authors: S G Deeks; M Smith; M Holodniy; J O Kahn
Journal: JAMA Date: 1997-01-08 Impact factor: 56.272

8. Sequence-specific polypeptoids: a diverse family of heteropolymers with stable secondary structure.

Authors: K Kirshenbaum; A E Barron; R A Goldsmith; P Armand; E K Bradley; K T Truong; K A Dill; F E Cohen; R N Zuckermann
Journal: Proc Natl Acad Sci U S A Date: 1998-04-14 Impact factor: 11.205

9. Crucial amides for dimerization inhibitors of HIV-1 protease.

Authors: Michael J Bowman; Jean Chmielewski
Journal: Bioorg Med Chem Lett Date: 2004-03-22 Impact factor: 2.823

10. Cross-resistance analysis of human immunodeficiency virus type 1 variants individually selected for resistance to five different protease inhibitors.

Authors: M Tisdale; R E Myers; B Maschera; N R Parry; N M Oliver; E D Blair
Journal: Antimicrob Agents Chemother Date: 1995-08 Impact factor: 5.191

6 in total

1. Synthetic, structural mimetics of the β-hairpin flap of HIV-1 protease inhibit enzyme function.

Authors: Jay Chauhan; Shen-En Chen; Katherine J Fenstermacher; Aurash Naser-Tavakolian; Tali Reingewertz; Rosene Salmo; Christian Lee; Emori Williams; Mithun Raje; Eric Sundberg; Jeffrey J DeStefano; Ernesto Freire; Steven Fletcher
Journal: Bioorg Med Chem Date: 2015-09-07 Impact factor: 3.641