Literature DB >> 20177623

Clickable bifunctional radiometal chelates for peptide labeling.

Artem Y Lebedev1, Jason P Holland, Jason S Lewis.   

Abstract

Novel synthetic methods for producing an array of chelates for use in "click"-radiolabeling of peptides are described, and their reactivity with regards to subsequent conjugation and radiolabeling is discussed.

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Year:  2010        PMID: 20177623      PMCID: PMC4958412          DOI: 10.1039/b924784j

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN: 1359-7345            Impact factor:   6.222


  15 in total

1.  "Click to chelate": synthesis and installation of metal chelates into biomolecules in a single step.

Authors:  Thomas L Mindt; Harriet Struthers; Luc Brans; Todor Anguelov; Christian Schweinsberg; Veronique Maes; Dirk Tourwé; Roger Schibli
Journal:  J Am Chem Soc       Date:  2006-11-29       Impact factor: 15.419

Review 2.  Nonnatural amino acids for site-specific protein conjugation.

Authors:  Albert J de Graaf; Marlous Kooijman; Wim E Hennink; Enrico Mastrobattista
Journal:  Bioconjug Chem       Date:  2009-07       Impact factor: 4.774

3.  Synthesis of a cross-bridged cyclam derivative for peptide conjugation and 64Cu radiolabeling.

Authors:  C Andrew Boswell; Celeste A S Regino; Kwamena E Baidoo; Karen J Wong; Ambika Bumb; Heng Xu; Diane E Milenic; James A Kelley; Christopher C Lai; Martin W Brechbiel
Journal:  Bioconjug Chem       Date:  2008-07-03       Impact factor: 4.774

4.  DOTA-D-Tyr(1)-octreotate: a somatostatin analogue for labeling with metal and halogen radionuclides for cancer imaging and therapy.

Authors:  Wen Ping Li; Jason S Lewis; Joonyoung Kim; Joseph E Bugaj; Michael A Johnson; Jack L Erion; Carolyn J Anderson
Journal:  Bioconjug Chem       Date:  2002 Jul-Aug       Impact factor: 4.774

5.  Copper-64 radiopharmaceuticals for PET imaging of cancer: advances in preclinical and clinical research.

Authors:  Carolyn J Anderson; Riccardo Ferdani
Journal:  Cancer Biother Radiopharm       Date:  2009-08       Impact factor: 3.099

6.  Preparation and biological evaluation of 64Cu-CB-TE2A-sst2-ANT, a somatostatin antagonist for PET imaging of somatostatin receptor-positive tumors.

Authors:  Thaddeus J Wadas; Martin Eiblmaier; Alexander Zheleznyak; Christopher D Sherman; Riccardo Ferdani; Kexian Liang; Samuel Achilefu; Carolyn J Anderson
Journal:  J Nucl Med       Date:  2008-10-16       Impact factor: 10.057

7.  Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloaddition.

Authors:  Qian Wang; Timothy R Chan; Robert Hilgraf; Valery V Fokin; K Barry Sharpless; M G Finn
Journal:  J Am Chem Soc       Date:  2003-03-19       Impact factor: 15.419

8.  Synthesis of novel 1,4,7,10-tetraazacyclodecane-1,4,7,10-tetraacetic acid (DOTA) derivatives for chemoselective attachment to unprotected polyfunctionalized compounds.

Authors:  Sebastian Knör; Armin Modlinger; Thorsten Poethko; Margret Schottelius; Hans-Jürgen Wester; Horst Kessler
Journal:  Chemistry       Date:  2007       Impact factor: 5.236

9.  In vivo evaluation and small-animal PET/CT of a prostate cancer mouse model using 64Cu bombesin analogs: side-by-side comparison of the CB-TE2A and DOTA chelation systems.

Authors:  Jered C Garrison; Tammy L Rold; Gary L Sieckman; Said Daibes Figueroa; Wynn A Volkert; Silvia S Jurisson; Timothy J Hoffman
Journal:  J Nucl Med       Date:  2007-07-13       Impact factor: 10.057

10.  64Cu-labeled alpha-melanocyte-stimulating hormone analog for microPET imaging of melanocortin 1 receptor expression.

Authors:  Zhen Cheng; Zhengming Xiong; Murugesan Subbarayan; Xiaoyuan Chen; Sanjiv Sam Gambhir
Journal:  Bioconjug Chem       Date:  2007-03-10       Impact factor: 4.774

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  17 in total

1.  Cu(I)-assisted click chemistry strategy for conjugation of non-protected cross-bridged macrocyclic chelators to tumour-targeting peptides.

Authors:  Zhengxin Cai; Barbara T Y Li; Edward H Wong; Gary R Weisman; Carolyn J Anderson
Journal:  Dalton Trans       Date:  2015-03-07       Impact factor: 4.390

2.  A practical guide to the construction of radiometallated bioconjugates for positron emission tomography.

Authors:  Brian M Zeglis; Jason S Lewis
Journal:  Dalton Trans       Date:  2011-03-25       Impact factor: 4.390

3.  Synthesis of a DOTA--biotin conjugate for radionuclide chelation via Cu-free click chemistry.

Authors:  Michael K Schultz; Sharavathi G Parameswarappa; F Christopher Pigge
Journal:  Org Lett       Date:  2010-05-21       Impact factor: 6.005

4.  Copper-Free Click for PET: Rapid 1,3-Dipolar Cycloadditions with a Fluorine-18 Cyclooctyne.

Authors:  Richard D Carpenter; Sven H Hausner; Julie L Sutcliffe
Journal:  ACS Med Chem Lett       Date:  2011-10-07       Impact factor: 4.345

5.  Universal Molecular Scaffold for Facile Construction of Multivalent and Multimodal Imaging Probes.

Authors:  Yongkang Gai; Guangya Xiang; Xiang Ma; Wenqi Hui; Qin Ouyang; Lingyi Sun; Jiule Ding; Jing Sheng; Dexing Zeng
Journal:  Bioconjug Chem       Date:  2016-02-24       Impact factor: 4.774

6.  Improved synthesis and biological evaluation of chelator-modified α-MSH analogs prepared by copper-free click chemistry.

Authors:  Nicholas J Baumhover; Molly E Martin; Sharavathi G Parameswarappa; Kyle C Kloepping; M Sue O'Dorisio; F Christopher Pigge; Michael K Schultz
Journal:  Bioorg Med Chem Lett       Date:  2011-08-08       Impact factor: 2.823

7.  Synthesis and biological evaluation of water-soluble progesterone-conjugated probes for magnetic resonance imaging of hormone related cancers.

Authors:  Preeti A Sukerkar; Keith W MacRenaris; Taryn R Townsend; Roshan A Ahmed; Joanna E Burdette; Thomas J Meade
Journal:  Bioconjug Chem       Date:  2011-10-05       Impact factor: 4.774

Review 8.  Click Chemistry and Radiochemistry: The First 10 Years.

Authors:  Jan-Philip Meyer; Pierre Adumeau; Jason S Lewis; Brian M Zeglis
Journal:  Bioconjug Chem       Date:  2016-11-22       Impact factor: 4.774

9.  H(2)azapa: a versatile acyclic multifunctional chelator for (67)Ga, (64)Cu, (111)In, and (177)Lu.

Authors:  Gwendolyn A Bailey; Eric W Price; Brian M Zeglis; Cara L Ferreira; Eszter Boros; Michael J Lacasse; Brian O Patrick; Jason S Lewis; Michael J Adam; Chris Orvig
Journal:  Inorg Chem       Date:  2012-10-29       Impact factor: 5.165

10.  New cross-bridged cyclam derivative CB-TE1K1P, an improved bifunctional chelator for copper radionuclides.

Authors:  Dexing Zeng; Qin Ouyang; Zhengxin Cai; Xiang-Qun Xie; Carolyn J Anderson
Journal:  Chem Commun (Camb)       Date:  2014-01-04       Impact factor: 6.222

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