Literature DB >> 20160926

A Simple Method for the Conversion of Carboxylic Acids into Thioacids with Lawesson's Reagent.

Yu Rao1, Xuechen Li, Pavel Nagorny, Joji Hayashida, Samuel J Danishefsky.   

Abstract

A one-step protocol for the conversion of carboxylic acids to thioesters, using Lawesson's Reagent, has been developed.

Entities:  

Year:  2009        PMID： 20160926      PMCID： PMC2762222          DOI： 10.1016/j.tetlet.2009.09.080

Source DB:  PubMed          Journal:  Tetrahedron Lett        ISSN： 0040-4039            Impact factor:   2.415


  18 in total

1.  Mechanism of thio acid/azide amidation.

Authors:  Robert V Kolakowski; Ning Shangguan; Ronald R Sauers; Lawrence J Williams
Journal:  J Am Chem Soc       Date:  2006-05-03       Impact factor: 15.419

2.  Use of Lawesson's reagent in organic syntheses.

Authors:  Turan Ozturk; Erdal Ertas; Olcay Mert
Journal:  Chem Rev       Date:  2007-09-15       Impact factor: 60.622

3.  Chemical synthesis of alpha-inhibin-92 by the thiocarboxyl segment coupling method.

Authors:  J Blake; D Yamashiro; K Ramasharma; C H Li
Journal:  Int J Pept Protein Res       Date:  1986-11

4.  Coupling reactions of hindered isonitriles and hindered alkyl thioacids: Mechanistic studies.

Authors:  Jennifer L Stockdill; Xiangyang Wu; Samuel J Danishefsky
Journal:  Tetrahedron Lett       Date:  2009-09-09       Impact factor: 2.415

5.  Thio-mediated synthesis of derivatized N-linked glycopeptides using isonitrile chemistry.

Authors:  Xiangyang Wu; Yu Yuan; Xuechen Li; Samuel J Danishefsky
Journal:  Tetrahedron Lett       Date:  2009-08-12       Impact factor: 2.415

6.  New segment synthesis of alpha-inhibin-92 by the acyl disulfide method.

Authors:  D Yamashiro; C H Li
Journal:  Int J Pept Protein Res       Date:  1988-03

7.  Resin-bound sulfonyl azides: efficient loading and activation strategy for the preparation of the N-acyl sulfonamide linker.

Authors:  Remco Merkx; Matthijs J van Haren; Dirk T S Rijkers; Rob M J Liskamp
Journal:  J Org Chem       Date:  2007-05-12       Impact factor: 4.354

8.  Thio acid/azide amidation: an improved route to N-acyl sulfonamides.

Authors:  Kristin N Barlett; Robert V Kolakowski; Sreenivas Katukojvala; Lawrence J Williams
Journal:  Org Lett       Date:  2006-03-02       Impact factor: 6.005

9.  Toward fully synthetic homogeneous beta-human follicle-stimulating hormone (beta-hFSH) with a biantennary N-linked dodecasaccharide. synthesis of beta-hFSH with chitobiose units at the natural linkage sites.

Authors:  Pavel Nagorny; Bernhard Fasching; Xuechen Li; Gong Chen; Baptiste Aussedat; Samuel J Danishefsky
Journal:  J Am Chem Soc       Date:  2009-04-29       Impact factor: 15.419

10.  Amino acid and peptide synthesis and functionalization by the reaction of thioacids with 2,4-dinitrobenzenesulfonamides.

Authors:  David Crich; Kasinath Sana; Songpo Guo
Journal:  Org Lett       Date:  2007-09-27       Impact factor: 6.005
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  8 in total

1.  Dihydro-3-(triphenylphosphoranylidene)-2,5-thiophendione: A Convenient Synthon for the Preparation of Substituted 1,4-Thiazepin-5-ones and Piperidinones via the Intermediacy of Thioacids.

Authors:  David Crich; Md Yeajur Rahaman
Journal:  Tetrahedron       Date:  2010-08-14       Impact factor: 2.457

2.  Total synthesis of cyclosporine: access to N-methylated peptides via isonitrile coupling reactions.

Authors:  Xiangyang Wu; Jennifer L Stockdill; Ping Wang; Samuel J Danishefsky
Journal:  J Am Chem Soc       Date:  2010-03-31       Impact factor: 15.419

3.  Biomimetic Stereoselective Sulfa-Michael Addition Leads to Platensimycin and Platencin Sulfur Analogues against Methicillin-Resistant Staphylococcus aureus.

Authors:  Lin Qiu; Kai Tian; Zhongqing Wen; Youchao Deng; Dingding Kang; Haoyu Liang; Xiangcheng Zhu; Ben Shen; Yanwen Duan; Yong Huang
Journal:  J Nat Prod       Date:  2018-02-01       Impact factor: 4.050

4.  Esterase-Sensitive Prodrugs with Tunable Release Rates and Direct Generation of Hydrogen Sulfide.

Authors:  Yueqin Zheng; Bingchen Yu; Kaili Ji; Zhixiang Pan; Vayou Chittavong; Binghe Wang
Journal:  Angew Chem Int Ed Engl       Date:  2016-01-28       Impact factor: 15.336

5.  Migrastatin analogues inhibit canine mammary cancer cell migration and invasion.

Authors:  Kinga Majchrzak; Daniele Lo Re; Małgorzata Gajewska; Małgorzata Bulkowska; Agata Homa; Karol Pawłowski; Tomasz Motyl; Paul V Murphy; Magdalena Król
Journal:  PLoS One       Date:  2013-10-08       Impact factor: 3.240

Review 6.  The Therapeutic Potential of Migrastatin-Core Analogs for the Treatment of Metastatic Cancer.

Authors:  Ernest Giralt; Daniele Lo Re
Journal:  Molecules       Date:  2017-02-09       Impact factor: 4.411

Review 7.  Trends in H2S-Donors Chemistry and Their Effects in Cardiovascular Diseases.

Authors:  Angela Corvino; Francesco Frecentese; Elisa Magli; Elisa Perissutti; Vincenzo Santagada; Antonia Scognamiglio; Giuseppe Caliendo; Ferdinando Fiorino; Beatrice Severino
Journal:  Antioxidants (Basel)       Date:  2021-03-11

Review 8.  H2S Donors and Their Use in Medicinal Chemistry.

Authors:  Elisa Magli; Elisa Perissutti; Vincenzo Santagada; Giuseppe Caliendo; Angela Corvino; Gianluca Esposito; Giovanna Esposito; Ferdinando Fiorino; Marco Migliaccio; Antonia Scognamiglio; Beatrice Severino; Rosa Sparaco; Francesco Frecentese
Journal:  Biomolecules       Date:  2021-12-18
  8 in total

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