Literature DB >> 20127371

EC(50) of remifentanil to prevent withdrawal movement associated with injection of rocuronium.

Ji Young Yoon1, Hae Kyu Kim, Jae Young Kwon, Sang Wook Shin, Kyung Hoon Kim, Won Sung Kim, Tae Kyun Kim.   

Abstract

PURPOSE: Various strategies have been studied to reduce the discomfort of rocuronium injection. This study was designed to determine the effect-site target concentration (Ce) of remifentanil at which there was a 50% probability of preventing movement from pain in response to the injection of rocuronium (EC(50)).
METHODS: Anesthesia was induced with a propofol target-controlled infusion (TCI, Marsh model) and remifentanil TCI (Minto model). Effect-site target concentration of propofol was 3 microg/ml. Ce of remifentanil for the first patient started at 2.0 ng/ml. Ce of remifentanil for each subsequent patient was determined by the response of the previous patient by the Dixon up-and-down method with an interval of 0.5 ng/ml. After both drugs reached target concentration, rocuronium 0.8 mg/kg was administered, and the pain response was observed.
RESULTS: The EC(50) of remifentanil was 1.5 +/- 0.45 ng/ml by Dixon's up-and-down method. From probit analysis, the EC(50) of remifentanil was 1.37 ng/ml (95% confidence limits, 0.69-2.15 ng/ml), and the EC(95) was 3.19 ng/ml (95% confidence limits, 2.31-11.24 ng/ml).
CONCLUSION: The EC(50) of remifentanil to blunt the withdrawal responses to rocuronium injection was 1.37-1.5 ng/ml during 3 microg/ml propofol TCI anesthesia.

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Year:  2010        PMID: 20127371     DOI: 10.1007/s00540-010-0868-7

Source DB:  PubMed          Journal:  J Anesth        ISSN: 0913-8668            Impact factor:   2.078


  20 in total

1.  The prevention of pain from injection of rocuronium by ondansetron, lidocaine, tramadol, and fentanyl.

Authors:  Dilek Memiş; Alparslan Turan; Beyhan Karamanlioğlu; Necdet Süt; Zafer Pamukçu
Journal:  Anesth Analg       Date:  2002-06       Impact factor: 5.108

2.  Low and moderate remifentanil infusion rates do not alter target-controlled infusion propofol concentrations necessary to maintain anesthesia as assessed by bispectral index monitoring.

Authors:  Lars P Wang; Peter McLoughlin; Michael J Paech; Irina Kurowski; Emma L Brandon
Journal:  Anesth Analg       Date:  2007-02       Impact factor: 5.108

3.  Efficient analysis of experimental observations.

Authors:  W J Dixon
Journal:  Annu Rev Pharmacol Toxicol       Date:  1980       Impact factor: 13.820

4.  The use of lidocaine for preventing the withdrawal associated with the injection of rocuronium in children and adolescents.

Authors:  Y Shevchenko; J C Jocson; V A McRae; S A Stayer; R E Schwartz; M Rehman; D K Choudhry
Journal:  Anesth Analg       Date:  1999-04       Impact factor: 5.108

5.  Influence of age and gender on the pharmacokinetics and pharmacodynamics of remifentanil. I. Model development.

Authors:  C F Minto; T W Schnider; T D Egan; E Youngs; H J Lemmens; P L Gambus; V Billard; J F Hoke; K H Moore; D J Hermann; K T Muir; J W Mandema; S L Shafer
Journal:  Anesthesiology       Date:  1997-01       Impact factor: 7.892

6.  Dilution of rocuronium to 0.5 mg/mL with 0.9% NaCl eliminates the pain during intravenous injection in awake patients.

Authors:  Bahattin Tuncali; Ayse Karci; Binnur Erdalkiran Tuncali; Omur Mavioglu; Cimen Gulben Olguner; Selin Ayhan; Zahide Elar
Journal:  Anesth Analg       Date:  2004-09       Impact factor: 5.108

7.  Requirements for target-controlled infusion of propofol to insert the laryngeal mask airway.

Authors:  I N Taylor; G N Kenny
Journal:  Anaesthesia       Date:  1998-03       Impact factor: 6.955

8.  Remifentanil versus alfentanil: comparative pharmacokinetics and pharmacodynamics in healthy adult male volunteers.

Authors:  T D Egan; C F Minto; D J Hermann; J Barr; K T Muir; S L Shafer
Journal:  Anesthesiology       Date:  1996-04       Impact factor: 7.892

9.  Injection pain of rocuronium and vecuronium is evoked by direct activation of nociceptive nerve endings.

Authors:  J A Blunk; F Seifert; M Schmelz; P W Reeh; W Koppert
Journal:  Eur J Anaesthesiol       Date:  2003-03       Impact factor: 4.330

10.  Determination of the pharmacodynamic interaction of propofol and remifentanil during esophagogastroduodenoscopy in children.

Authors:  David R Drover; Catherine Litalien; Vinit Wellis; Steven L Shafer; Gregory B Hammer
Journal:  Anesthesiology       Date:  2004-06       Impact factor: 7.892

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  3 in total

1.  The effect of gender on EC(50) of remifentanil to prevent pain during injection of microemulsion propofol.

Authors:  Bo-Won Lee; Sang-Hun Kim; Keum-Young So
Journal:  Korean J Anesthesiol       Date:  2012-12-14

Review 2.  Pharmacological and non-pharmacological interventions for reducing rocuronium bromide induced pain on injection in children and adults.

Authors:  Hemanshu Prabhakar; Gyaninder Pal Singh; Zulfiqar Ali; Mani Kalaivani; Martha A Smith
Journal:  Cochrane Database Syst Rev       Date:  2016-02-12

3.  EC50 and EC95 of remifentanil to prevent rocuronium-induced withdrawal movements in children.

Authors:  Hye Jin Park; Hyoseok Kang; Eu-Gene Kim; Juyoun Choi; Jeong Sung Seo
Journal:  Korean J Anesthesiol       Date:  2014-06-26
  3 in total

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