Literature DB >> 20042373

Cellular basis for atrial fibrillation in an experimental model of short QT1: implications for a pharmacological approach to therapy.

Eyal Nof1, Alexander Burashnikov, Charles Antzelevitch.   

Abstract

BACKGROUND: Short QT (SQT) syndrome (SQT) 1 is an inherited sudden death syndrome often associated with atrial fibrillation (AF). We examined the cellular basis for AF in a newly developed experimental atrial model of SQT1.
METHODS: Action potentials (APs) were recorded from the pectinate muscle (PM) and crista terminalis (CT) regions of coronary-perfused canine right atrial preparations, together with a pseudoelectrocardiogram. The I(Kr) agonist PD-118057 (20 microM) was used to mimic the gain of function in I(Kr) known to underlie SQT1.
RESULTS: The I(Kr) agonist significantly abbreviated the AP duration (APD) of CT and PM and of the effective refractory period (ERP) measured in PM (n = 28). Spatial dispersion of repolarization (SDR), defined as inter-regional differences of APD, increased from 27 +/- 17 ms to 51 +/- 32 ms (P = .002; n = 28). AF could be induced by a single premature stimulus after but not before exposure to PD-118057 in 26/28 (93%) preparations. Quinidine (10 microM), which prolonged APD and ERP, but not lidocaine (20 microM) or E-4031 (5 microM), which prolonged only ERP or APD, respectively, was effective in preventing the PD-118057-mediated AF. In the presence of PD-118057, isoproterenol (100 nM) further abbreviated both APD and ERP and facilitated induction of sustained AF in five of six preparations.
CONCLUSIONS: The I(Kr) agonist recapitulates the electrophysiologic and arrhythmic manifestations of SQT1. Abbreviation of APD and ERP and amplification of SDR predispose to the development of AF by creating the substrate for reentry. Quinidine, but not E-4031 or lidocaine, was effective in preventing AF in this setting.

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Year:  2009        PMID: 20042373      PMCID: PMC2826201          DOI: 10.1016/j.hrthm.2009.10.017

Source DB:  PubMed          Journal:  Heart Rhythm        ISSN: 1547-5271            Impact factor:   6.343


  39 in total

1.  Catheter ablation of long-lasting persistent atrial fibrillation: critical structures for termination.

Authors:  Michel Haïssaguerre; Prashanthan Sanders; Mélèze Hocini; Yoshihide Takahashi; Martin Rotter; Frederic Sacher; Thomas Rostock; Li-Fern Hsu; Pierre Bordachar; Sylvain Reuter; Raymond Roudaut; Jacques Clémenty; Pierre Jaïs
Journal:  J Cardiovasc Electrophysiol       Date:  2005-11

2.  How Do Atrial-Selective Drugs Differ From Antiarrhythmic Drugs Currently Used in the Treatment of Atrial Fibrillation?

Authors:  Alexander Burashnikov; Charles Antzelevitch
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3.  Ionic mechanisms of electrical remodeling in human atrial fibrillation.

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4.  Ionic mechanisms of regional action potential heterogeneity in the canine right atrium.

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5.  Further insights into the effect of quinidine in short QT syndrome caused by a mutation in HERG.

Authors:  Christian Wolpert; Rainer Schimpf; Carla Giustetto; Charles Antzelevitch; Jonathan Cordeiro; Robert Dumaine; Ramon Brugada; Kui Hong; Urs Bauersfeld; Fiorenzo Gaita; Martin Borggrefe
Journal:  J Cardiovasc Electrophysiol       Date:  2005-01

6.  The pharmacological response of ischemia-related atrial fibrillation in dogs: evidence for substrate-specific efficacy.

Authors:  Lena Rivard; Hani Sinno; Akiko Shiroshita-Takeshita; Gernot Schram; Tack-Ki Leung; Stanley Nattel
Journal:  Cardiovasc Res       Date:  2007-01-27       Impact factor: 10.787

7.  Disopyramide is an effective inhibitor of mutant HERG K+ channels involved in variant 1 short QT syndrome.

Authors:  Mark J McPate; Rona S Duncan; Harry J Witchel; Jules C Hancox
Journal:  J Mol Cell Cardiol       Date:  2006-07-12       Impact factor: 5.000

8.  Transmembrane action potential heterogeneity in the canine isolated arterially perfused right atrium: effect of IKr and IKur/Ito block.

Authors:  Alexander Burashnikov; Sandeep Mannava; Charles Antzelevitch
Journal:  Am J Physiol Heart Circ Physiol       Date:  2004-06       Impact factor: 4.733

9.  Sudden death associated with short-QT syndrome linked to mutations in HERG.

Authors:  Ramon Brugada; Kui Hong; Robert Dumaine; Jonathan Cordeiro; Fiorenzo Gaita; Martin Borggrefe; Teresa M Menendez; Josep Brugada; Guido D Pollevick; Christian Wolpert; Elena Burashnikov; Kiyotaka Matsuo; Yue Sheng Wu; Alejandra Guerchicoff; Francesca Bianchi; Carla Giustetto; Rainer Schimpf; Pedro Brugada; Charles Antzelevitch
Journal:  Circulation       Date:  2003-12-15       Impact factor: 29.690

10.  Identification of a KCNE2 gain-of-function mutation in patients with familial atrial fibrillation.

Authors:  Yiqing Yang; Min Xia; Qingfeng Jin; Saïd Bendahhou; Jingyi Shi; Yiping Chen; Bo Liang; Jie Lin; Yi Liu; Ban Liu; Qinshu Zhou; Dongwei Zhang; Rong Wang; Ning Ma; Xiaoyan Su; Kaiya Niu; Yan Pei; Wenyuan Xu; Zhaopeng Chen; Haiying Wan; Jianmin Cui; Jacques Barhanin; Yihan Chen
Journal:  Am J Hum Genet       Date:  2004-09-13       Impact factor: 11.025

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  11 in total

Review 1.  Optical and electrical recordings from isolated coronary-perfused ventricular wedge preparations.

Authors:  José M Di Diego; Serge Sicouri; Rachel C Myles; Francis L Burton; Godfrey L Smith; Charles Antzelevitch
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2.  Overview of Basic Mechanisms of Cardiac Arrhythmia.

Authors:  Charles Antzelevitch; Alexander Burashnikov
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3.  PQ segment depression in patients with short QT syndrome: a novel marker for diagnosing short QT syndrome?

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Journal:  Heart Rhythm       Date:  2014-02-28       Impact factor: 6.343

Review 4.  Inherited cardiac arrhythmias.

Authors:  Peter J Schwartz; Michael J Ackerman; Charles Antzelevitch; Connie R Bezzina; Martin Borggrefe; Bettina F Cuneo; Arthur A M Wilde
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Review 5.  HERG1 channel agonists and cardiac arrhythmia.

Authors:  Michael C Sanguinetti
Journal:  Curr Opin Pharmacol       Date:  2013-11-27       Impact factor: 5.547

Review 6.  The role of late I Na in development of cardiac arrhythmias.

Authors:  Charles Antzelevitch; Vladislav Nesterenko; John C Shryock; Sridharan Rajamani; Yejia Song; Luiz Belardinelli
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Review 7.  Atrial Fibrillation Predictors: Importance of the Electrocardiogram.

Authors:  David M German; Muammar M Kabir; Thomas A Dewland; Charles A Henrikson; Larisa G Tereshchenko
Journal:  Ann Noninvasive Electrocardiol       Date:  2015-11-02       Impact factor: 1.468

8.  Circulating KCNH2 current-activating factor in patients with heart failure and ventricular tachyarrhythmia.

Authors:  Hiroki Sugiyama; Kazufumi Nakamura; Hiroshi Morita; Satoshi Akagi; Yoshinori Tani; Yusuke Katayama; Nobuhiro Nishii; Toru Miyoshi; Satoshi Nagase; Kunihisa Kohno; Kengo Fukushima Kusano; Tohru Ohe; Junko Kurokawa; Tetsushi Furukawa; Hiroshi Ito
Journal:  PLoS One       Date:  2011-05-19       Impact factor: 3.240

9.  The hERG K(+) channel S4 domain L532P mutation: characterization at 37°C.

Authors:  Yi H Zhang; Charlotte K Colenso; Richard B Sessions; Christopher E Dempsey; Jules C Hancox
Journal:  Biochim Biophys Acta       Date:  2011-07-14

10.  Action potential clamp characterization of the S631A hERG mutation associated with short QT syndrome.

Authors:  Andrew Butler; Yihong Zhang; Alan G Stuart; Christopher E Dempsey; Jules C Hancox
Journal:  Physiol Rep       Date:  2018-09
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