Literature DB >> 19719234

Amide isosteres of oroidin: assessment of antibiofilm activity and C. elegans toxicity.

Justin J Richards1, Samuel Reyes, Sean D Stowe, Ashley T Tucker, T Eric Ballard, Laura D Mathies, John Cavanagh, Christian Melander.   

Abstract

The synthesis and antibiofilm activities of sulfonamide, urea, and thiourea oroidin analogues are described. The most active derivative was able to selectively inhibit P. aeruginosa biofilm development and is also shown to be nontoxic upward of 1 mM to the development of C. elegans in comparison to other similar isosteric analogues and the natural product oroidin.

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Year:  2009        PMID： 19719234      PMCID： PMC2739084          DOI： 10.1021/jm900378s

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


  29 in total

Review 1.  Device-associated infections: a macroproblem that starts with microadherence.

Authors:  R O Darouiche
Journal:  Clin Infect Dis       Date:  2001-09-26       Impact factor: 9.079

Review 2.  Bacterial biofilms: a common cause of persistent infections.

Authors:  J W Costerton; P S Stewart; E P Greenberg
Journal:  Science       Date:  1999-05-21       Impact factor: 47.728

Review 3.  Biofilms as complex differentiated communities.

Authors:  P Stoodley; K Sauer; D G Davies; J W Costerton
Journal:  Annu Rev Microbiol       Date:  2002-01-30       Impact factor: 15.500

4.  Small molecule inhibitors of bacterial quorum sensing and biofilm formation.

Authors:  Grant D Geske; Rachel J Wezeman; Adam P Siegel; Helen E Blackwell
Journal:  J Am Chem Soc       Date:  2005-09-21       Impact factor: 15.419

5.  Toxicology. Transforming environmental health protection.

Authors:  Francis S Collins; George M Gray; John R Bucher
Journal:  Science       Date:  2008-02-15       Impact factor: 47.728

6.  Inhibition and dispersion of proteobacterial biofilms.

Authors:  Justin J Richards; Robert W Huigens Iii; T Eric Ballard; Anne Basso; John Cavanagh; Christian Melander
Journal:  Chem Commun (Camb)       Date:  2008-02-08       Impact factor: 6.222

Review 7.  The role of quorum sensing in the pathogenicity of the cunning aggressor Pseudomonas aeruginosa.

Authors:  Thomas Bjarnsholt; Michael Givskov
Journal:  Anal Bioanal Chem       Date:  2006-09-26       Impact factor: 4.142

8.  Differential gene expression for investigation of Escherichia coli biofilm inhibition by plant extract ursolic acid.

Authors:  Dacheng Ren; Rongjun Zuo; Andrés F González Barrios; Laura A Bedzyk; Gary R Eldridge; Mark E Pasmore; Thomas K Wood
Journal:  Appl Environ Microbiol       Date:  2005-07       Impact factor: 4.792

Review 9.  Cystic fibrosis pathogenesis and the role of biofilms in persistent infection.

Authors:  J W Costerton
Journal:  Trends Microbiol       Date:  2001-02       Impact factor: 17.079

10.  Evaluation of dihydrooroidin as an antifouling additive in marine paint.

Authors:  Christian Melander; Peter D R Moeller; T Eric Ballard; Justin J Richards; Robert W Huigens; John Cavanagh
Journal:  Int Biodeterior Biodegradation       Date:  2009-06       Impact factor: 4.320
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  16 in total

1.  Evaluation of the toxicity of 2-aminoimidazole antibiofilm agents using both cellular and model organism systems.

Authors:  Sean D Stowe; Ashley T Tucker; Richele Thompson; Amanda Piper; Justin J Richards; Steven A Rogers; Laura D Mathies; Christian Melander; John Cavanagh
Journal:  Drug Chem Toxicol       Date:  2012-01-31       Impact factor: 3.356

2.  Novel pentadecenyl tetrazole enhances susceptibility of methicillin-resistant Staphylococcus aureus biofilms to gentamicin.

Authors:  Krista M Olson; Courtney M Starks; Russell B Williams; Mark O'Neil-Johnson; Zhongping Huang; Michael Ellis; John E Reilly; Gary R Eldridge
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3.  Marine sponge alkaloids as a source of anti-bacterial adjuvants.

Authors:  Roberta J Melander; Hong-Bing Liu; Matthew D Stephens; Carole A Bewley; Christian Melander
Journal:  Bioorg Med Chem Lett       Date:  2016-11-09       Impact factor: 2.823

4.  Synergistic effects between conventional antibiotics and 2-aminoimidazole-derived antibiofilm agents.

Authors:  Steven A Rogers; Robert W Huigens; John Cavanagh; Christian Melander
Journal:  Antimicrob Agents Chemother       Date:  2010-03-08       Impact factor: 5.191

5.  5-Benzylidene-4-oxazolidinones potently inhibit biofilm formation in Methicillin-resistant Staphylococcus aureus.

Authors:  Grant A Edwards; Nataliia V Shymanska; Joshua G Pierce
Journal:  Chem Commun (Camb)       Date:  2017-06-29       Impact factor: 6.222

6.  Inhibition and breaking of advanced glycation end-products (AGEs) with bis-2-aminoimidazole derivatives.

Authors:  Mike A Richardson; Robert E Furlani; Brendan K Podell; David F Ackart; Jessica D Haugen; Roberta J Melander; Christian Melander; Randall J Basaraba
Journal:  Tetrahedron Lett       Date:  2015       Impact factor: 2.415

7.  The bromotyrosine derivative ianthelline isolated from the arctic marine sponge Stryphnus fortis inhibits marine micro- and macrobiofouling.

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Journal:  Mar Biotechnol (NY)       Date:  2014-07-23       Impact factor: 3.619

8.  Identification of BfmR, a response regulator involved in biofilm development, as a target for a 2-Aminoimidazole-based antibiofilm agent.

Authors:  Richele J Thompson; Benjamin G Bobay; Sean D Stowe; Andrew L Olson; Lingling Peng; Zhaoming Su; Luis A Actis; Christian Melander; John Cavanagh
Journal:  Biochemistry       Date:  2012-11-29       Impact factor: 3.162

Review 9.  A submarine journey: the pyrrole-imidazole alkaloids.

Authors:  Barbara Forte; Beatrice Malgesini; Claudia Piutti; Francesca Quartieri; Alessandra Scolaro; Gianluca Papeo
Journal:  Mar Drugs       Date:  2009-11-27       Impact factor: 5.118

10.  2-Aminobenzimidazoles as antibiofilm agents against Salmonella enterica serovar Typhimurium.

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Journal:  Medchemcomm       Date:  2018-08-02       Impact factor: 3.597
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