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78 in total

Review 1. Target-oriented and diversity-oriented organic synthesis in drug discovery.

Authors: S L Schreiber
Journal: Science Date: 2000-03-17 Impact factor: 47.728

2. A Convergent, Enantioselective Total Synthesis of Streptogramin Antibiotic (-)-Madumycin II.

Authors: Arun K. Ghosh; Wenming Liu
Journal: J Org Chem Date: 1997-11-14 Impact factor: 4.354

3. Counterions of BINAP-Pt(II) and -Pd(II) complexes: novel catalysts for highly enantioselective Diels-Alder reaction.

Authors: A K Ghosh; H Matsuda
Journal: Org Lett Date: 1999-12-30 Impact factor: 6.005

4. Structure-based design of potent and selective cell-permeable inhibitors of human beta-secretase (BACE-1).

Authors: Shawn J Stachel; Craig A Coburn; Thomas G Steele; Kristen G Jones; Elizabeth F Loutzenhiser; Alison R Gregro; Hemaka A Rajapakse; Ming-Tain Lai; Ming-Chih Crouthamel; Min Xu; Katherine Tugusheva; Janet E Lineberger; Beth L Pietrak; Amy S Espeseth; Xiao-Ping Shi; Elizabeth Chen-Dodson; M Katharine Holloway; Sanjeev Munshi; Adam J Simon; Lawrence Kuo; Joseph P Vacca
Journal: J Med Chem Date: 2004-12-16 Impact factor: 7.446

5. Potent inhibition of HIV-1 replication by novel non-peptidyl small molecule inhibitors of protease dimerization.

Authors: Yasuhiro Koh; Shintaro Matsumi; Debananda Das; Masayuki Amano; David A Davis; Jianfeng Li; Sofiya Leschenko; Abigail Baldridge; Tatsuo Shioda; Robert Yarchoan; Arun K Ghosh; Hiroaki Mitsuya
Journal: J Biol Chem Date: 2007-07-17 Impact factor: 5.157

6. Potent HIV protease inhibitors incorporating high-affinity P2-ligands and (R)-(hydroxyethylamino)sulfonamide isostere.

Authors: A K Ghosh; J F Kincaid; W Cho; D E Walters; K Krishnan; K A Hussain; Y Koo; H Cho; C Rudall; L Holland; J Buthod
Journal: Bioorg Med Chem Lett Date: 1998-03-17 Impact factor: 2.823

7. Kinetic characterization and cross-resistance patterns of HIV-1 protease mutants selected under drug pressure.

Authors: S V Gulnik; L I Suvorov; B Liu; B Yu; B Anderson; H Mitsuya; J W Erickson
Journal: Biochemistry Date: 1995-07-25 Impact factor: 3.162

8. Enantioselective total synthesis of (+)-amphidinolide t1.

Authors: Arun K Ghosh; Chunfeng Liu
Journal: J Am Chem Soc Date: 2003-03-05 Impact factor: 15.419

Review 9. Beta-secretase as a therapeutic target for inhibitor drugs.

Authors: Arun K Ghosh; Lin Hong; Jordan Tang
Journal: Curr Med Chem Date: 2002-06 Impact factor: 4.530

Review 10. Memapsin 2 (beta-secretase) inhibitors: drug development.

Authors: Arun K Ghosh; Nagaswamy Kumaragurubaran; Ling Hong; Gerald Koelsh; Jordan Tang
Journal: Curr Alzheimer Res Date: 2008-04 Impact factor: 3.498

12 in total

Review 1. Recent Progress in the Development of HIV-1 Protease Inhibitors for the Treatment of HIV/AIDS.

Authors: Arun K Ghosh; Heather L Osswald; Gary Prato
Journal: J Med Chem Date: 2016-01-22 Impact factor: 7.446

2. Facile and rapid route for the synthesis of novel conformationally constrained norstatine analogs via PADAM-cyclization methodology.

Authors: Arthur Y Shaw; Federico Medda; Christopher Hulme
Journal: Tetrahedron Lett Date: 2012-03-14 Impact factor: 2.415

3. Substituent effects on P2-cyclopentyltetrahydrofuranyl urethanes: design, synthesis, and X-ray studies of potent HIV-1 protease inhibitors.

Authors: Arun K Ghosh; Bruno D Chapsal; Melinda Steffey; Johnson Agniswamy; Yuan-Fang Wang; Masayuki Amano; Irene T Weber; Hiroaki Mitsuya
Journal: Bioorg Med Chem Lett Date: 2012-02-02 Impact factor: 2.823

4. Design of substituted bis-Tetrahydrofuran (bis-THF)-derived Potent HIV-1 Protease Inhibitors, Protein-ligand X-ray Structure, and Convenient Syntheses of bis-THF and Substituted bis-THF Ligands.

Authors: Arun K Ghosh; Cuthbert D Martyr; Melinda Steffey; Yuan-Fang Wang; Johnson Agniswamy; Masayuki Amano; Irene T Weber; Hiroaki Mitsuya
Journal: ACS Med Chem Lett Date: 2011-04-14 Impact factor: 4.345

5. Cu(II)-catalyzed olefin migration and Prins cyclization: highly diastereoselective synthesis of substituted tetrahydropyrans.

Authors: Arun K Ghosh; Daniel R Nicponski
Journal: Org Lett Date: 2011-07-28 Impact factor: 6.005

6. Nature Inspired Molecular Design: Stereoselective Synthesis of Bicyclic and Polycyclic Ethers for Potent HIV-1 Protease Inhibitors.

Authors: Arun K Ghosh; Margherita Brindisi
Journal: Asian J Org Chem Date: 2018-06-08 Impact factor: 3.319

7. Structure-based design, synthesis, X-ray studies, and biological evaluation of novel HIV-1 protease inhibitors containing isophthalamide-derived P2-ligands.

Authors: Arun K Ghosh; Jun Takayama; Luke A Kassekert; Jean-Rene Ella-Menye; Sofiya Yashchuk; Johnson Agniswamy; Yuan-Fang Wang; Manabu Aoki; Masayuki Amano; Irene T Weber; Hiroaki Mitsuya
Journal: Bioorg Med Chem Lett Date: 2015-05-30 Impact factor: 2.823

8. Capturing the essence of organic synthesis: from bioactive natural products to designed molecules in today's medicine.

Authors: Arun K Ghosh
Journal: J Org Chem Date: 2010-10-11 Impact factor: 4.354

9. Design of novel HIV-1 protease inhibitors incorporating isophthalamide-derived P2-P3 ligands: Synthesis, biological evaluation and X-ray structural studies of inhibitor-HIV-1 protease complex.

Authors: Arun K Ghosh; Margherita Brindisi; Prasanth R Nyalapatla; Jun Takayama; Jean-Rene Ella-Menye; Sofiya Yashchuk; Johnson Agniswamy; Yuan-Fang Wang; Manabu Aoki; Masayuki Amano; Irene T Weber; Hiroaki Mitsuya
Journal: Bioorg Med Chem Date: 2017-04-09 Impact factor: 3.641

10. HIV-1 Protease: Structural Perspectives on Drug Resistance.

Authors: Irene T Weber; Johnson Agniswamy
Journal: Viruses Date: 2009-12-03 Impact factor: 5.048