Literature DB >> 19239229

Kinase domain mutations in cancer: implications for small molecule drug design strategies.

Jack A Bikker1, Natasja Brooijmans, Allan Wissner, Tarek S Mansour.   

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Year:  2009        PMID： 19239229     DOI： 10.1021/jm8010542

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  28 in total

1.  A computational workflow for the design of irreversible inhibitors of protein kinases.

Authors:  Alberto Del Rio; Miriam Sgobba; Marco Daniele Parenti; Gianluca Degliesposti; Rosetta Forestiero; Claudia Percivalle; Pier Franco Conte; Mauro Freccero; Giulio Rastelli
Journal:  J Comput Aided Mol Des       Date:  2010-03-21       Impact factor: 3.686

Review 2.  Role of genetic and molecular profiling in sarcomas.

Authors:  Scott M Norberg; Sujana Movva
Journal:  Curr Treat Options Oncol       Date:  2015-05

3.  An enriched structural kinase database to enable kinome-wide structure-based analyses and drug discovery.

Authors:  Natasja Brooijmans; Yu-Wei Chang; Dominick Mobilio; Rajiah A Denny; Christine Humblet
Journal:  Protein Sci       Date:  2010-04       Impact factor: 6.725

4.  Regioselective multi-component synthesis of 1H-pyrazolo[3,4-d]pyrimidine-6(7H)-thiones.

Authors:  Shirin Safaei; Iraj Mohammadpoor-Baltork; Ahmad Reza Khosropour; Majid Moghadam; Shahram Tangestaninejad; Valiollah Mirkhani
Journal:  Mol Divers       Date:  2012-08-29       Impact factor: 2.943

5.  Diamine Ligands in Copper-Catalyzed Reactions.

Authors:  David S Surry; Stephen L Buchwald
Journal:  Chem Sci       Date:  2010       Impact factor: 9.825

6.  Dialkylbiaryl Phosphines in Pd-Catalyzed Amination: A User's Guide.

Authors:  David S Surry; Stephen L Buchwald
Journal:  Chem Sci       Date:  2011       Impact factor: 9.825

7.  Synthesis and structure-activity relationship study of diaryl[d,f][1,3]diazepines as potential anti-cancer agents.

Authors:  Longjia Yan; Hui Wang; Yunpeng Chen; Zhiwei Li; Yazhong Pei
Journal:  Mol Divers       Date:  2018-01-03       Impact factor: 2.943

8.  Selective Proteolysis to Study the Global Conformation and Regulatory Mechanisms of c-Src Kinase.

Authors:  Michael P Agius; Kristin S Ko; Taylor K Johnson; Frank E Kwarcinski; Sameer Phadke; Eric J Lachacz; Matthew B Soellner
Journal:  ACS Chem Biol       Date:  2019-07-09       Impact factor: 5.100

9.  Synthesis of novel 4H-pyrimido[1,6-a]pyrimidines via a one-pot three-component condensation.

Authors:  Jinbao Xiang; Hanghang Li; Kai Yang; Lang Yi; Yongnan Xu; Qun Dang; Xu Bai
Journal:  Mol Divers       Date:  2011-12-04       Impact factor: 2.943

Review 10.  Targeted therapy in GIST: in silico modeling for prediction of resistance.

Authors:  Marco A Pierotti; Elena Tamborini; Tiziana Negri; Sabrina Pricl; Silvana Pilotti
Journal:  Nat Rev Clin Oncol       Date:  2011-03       Impact factor: 66.675
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