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107 in total

1. Discovery and synthesis of namalide reveals a new anabaenopeptin scaffold and peptidase inhibitor.

Authors: Pradeep Cheruku; Alberto Plaza; Gianluigi Lauro; Jessica Keffer; John R Lloyd; Giuseppe Bifulco; Carole A Bewley
Journal: J Med Chem Date: 2012-01-05 Impact factor: 7.446

Review 2. Macrocyclic histone deacetylase inhibitors.

Authors: Sandra C Mwakwari; Vishal Patil; William Guerrant; Adegboyega K Oyelere
Journal: Curr Top Med Chem Date: 2010 Impact factor: 3.295

3. Largazole and analogues with modified metal-binding motifs targeting histone deacetylases: synthesis and biological evaluation.

Authors: Pravin Bhansali; Christin L Hanigan; Robert A Casero; L M Viranga Tillekeratne
Journal: J Med Chem Date: 2011-10-10 Impact factor: 7.446

4. Largazole is a Brain-Penetrant Class I HDAC Inhibitor with Extended Applicability to Glioblastoma and CNS Diseases.

Authors: Fatma H Al-Awadhi; Lilibeth A Salvador-Reyes; Lobna A Elsadek; Ranjala Ratnayake; Qi-Yin Chen; Hendrik Luesch
Journal: ACS Chem Neurosci Date: 2020-06-19 Impact factor: 4.418

Review 5. Discovery and mechanism of natural products as modulators of histone acetylation.

Authors: Lilibeth A Salvador; Hendrik Luesch
Journal: Curr Drug Targets Date: 2012-07 Impact factor: 3.465

Review 6. Biologically active secondary metabolites from marine cyanobacteria.

Authors: Joshawna K Nunnery; Emily Mevers; William H Gerwick
Journal: Curr Opin Biotechnol Date: 2010-10-26 Impact factor: 9.740

7. Design, synthesis, biological evaluation, and structural characterization of potent histone deacetylase inhibitors based on cyclic alpha/beta-tetrapeptide architectures.

Authors: Ana Montero; John M Beierle; Christian A Olsen; M Reza Ghadiri
Journal: J Am Chem Soc Date: 2009-03-04 Impact factor: 15.419

8. Synthesis and histone deacetylase inhibitory activity of largazole analogs: alteration of the zinc-binding domain and macrocyclic scaffold.

Authors: Albert A Bowers; Nathan West; Tenaya L Newkirk; Annie E Troutman-Youngman; Stuart L Schreiber; Olaf Wiest; James E Bradner; Robert M Williams
Journal: Org Lett Date: 2009-03-19 Impact factor: 6.005

Review 9. Structural determinants of affinity and selectivity in the binding of inhibitors to histone deacetylase 6.

Authors: Jeremy D Osko; David W Christianson
Journal: Bioorg Med Chem Lett Date: 2020-02-11 Impact factor: 2.823

10. Enantioselective total synthesis of (+)-largazole, a potent inhibitor of histone deacetylase.

Authors: Arun K Ghosh; Sarang Kulkarni
Journal: Org Lett Date: 2008-07-29 Impact factor: 6.005