Literature DB >> 17907127

Targeted degradation of the aryl hydrocarbon receptor by the PROTAC approach: a useful chemical genetic tool.

Hyosung Lee1, Dinesh Puppala, Eun-Young Choi, Hollie Swanson, Kyung-Bo Kim.   

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Year:  2007        PMID： 17907127     DOI： 10.1002/cbic.200700438

Source DB:  PubMed          Journal:  Chembiochem        ISSN： 1439-4227            Impact factor:   3.164


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  27 in total

1.  Impact of linker length on the activity of PROTACs.

Authors:  Kedra Cyrus; Marie Wehenkel; Eun-Young Choi; Hyeong-Jun Han; Hyosung Lee; Hollie Swanson; Kyung-Bo Kim
Journal:  Mol Biosyst       Date:  2010-10-04

Review 2.  Chemical inducers of targeted protein degradation.

Authors:  Kanak Raina; Craig M Crews
Journal:  J Biol Chem       Date:  2010-02-10       Impact factor: 5.157

Review 3.  PROTACs: great opportunities for academia and industry.

Authors:  Xiuyun Sun; Hongying Gao; Yiqing Yang; Ming He; Yue Wu; Yugang Song; Yan Tong; Yu Rao
Journal:  Signal Transduct Target Ther       Date:  2019-12-24

Review 4.  PROteolysis TArgeting Chimeras (PROTACs) - Past, present and future.

Authors:  Mariell Pettersson; Craig M Crews
Journal:  Drug Discov Today Technol       Date:  2019-02-13

5.  Two-headed PROTAC: an effective new tool for targeted protein degradation.

Authors:  Kedra Cyrus; Marie Wehenkel; Eun-Young Choi; Hollie Swanson; Kyung-Bo Kim
Journal:  Chembiochem       Date:  2010-07-26       Impact factor: 3.164

6.  Evolution of Cereblon-Mediated Protein Degradation as a Therapeutic Modality.

Authors:  Philip P Chamberlain; Laura A D'Agostino; J Michael Ellis; Joshua D Hansen; Mary E Matyskiela; Joseph J McDonald; Jennifer R Riggs; Lawrence G Hamann
Journal:  ACS Med Chem Lett       Date:  2019-11-12       Impact factor: 4.345

Review 7.  Induced protein degradation: an emerging drug discovery paradigm.

Authors:  Ashton C Lai; Craig M Crews
Journal:  Nat Rev Drug Discov       Date:  2016-11-25       Impact factor: 84.694

8.  HaloPROTACS: Use of Small Molecule PROTACs to Induce Degradation of HaloTag Fusion Proteins.

Authors:  Dennis L Buckley; Kanak Raina; Nicole Darricarrere; John Hines; Jeffrey L Gustafson; Ian E Smith; Afjal H Miah; John D Harling; Craig M Crews
Journal:  ACS Chem Biol       Date:  2015-06-23       Impact factor: 5.100

9.  Inhibitor mediated protein degradation.

Authors:  Marcus J C Long; Deviprasad R Gollapalli; Lizbeth Hedstrom
Journal:  Chem Biol       Date:  2012-05-25

Review 10.  Design and Applications of Bifunctional Small Molecules: Why Two Heads Are Better Than One.

Authors:  Timothy W Corson; Nicholas Aberle; Craig M Crews
Journal:  ACS Chem Biol       Date:  2008-11-21       Impact factor: 5.100
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