Literature DB >> 1738138

Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.

K A Jacobson1, P J van Galen, M Williams.   

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Year:  1992        PMID： 1738138      PMCID： PMC3476067          DOI： 10.1021/jm00081a001

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  132 in total

1.  RDC8 codes for an adenosine A2 receptor with physiological constitutive activity.

Authors:  C Maenhaut; J Van Sande; F Libert; M Abramowicz; M Parmentier; J J Vanderhaegen; J E Dumont; G Vassart; S Schiffmann
Journal:  Biochem Biophys Res Commun       Date:  1990-12-31       Impact factor: 3.575

2.  The physiological activity of adenine compounds with especial reference to their action upon the mammalian heart.

Authors:  A N Drury; A Szent-Györgyi
Journal:  J Physiol       Date:  1929-11-25       Impact factor: 5.182

Review 3.  Receptor triggering and receptor regulation: structure-activity relationships from the receptor's point of view.

Authors:  M D Hollenberg
Journal:  J Med Chem       Date:  1990-05       Impact factor: 7.446

4.  Imidazodiazepinediones: a new class of adenosine receptor antagonists.

Authors:  J W Daly; I Hide; P K Bridson
Journal:  J Med Chem       Date:  1990-10       Impact factor: 7.446

5.  Allosteric enhancement of adenosine A1 receptor binding and function by 2-amino-3-benzoylthiophenes.

Authors:  R F Bruns; J H Fergus
Journal:  Mol Pharmacol       Date:  1990-12       Impact factor: 4.436

6.  The adenosine/neutrophil paradox resolved: human neutrophils possess both A1 and A2 receptors that promote chemotaxis and inhibit O2 generation, respectively.

Authors:  B N Cronstein; L Daguma; D Nichols; A J Hutchison; M Williams
Journal:  J Clin Invest       Date:  1990-04       Impact factor: 14.808

7.  Interaction of amiloride and its analogues with adenosine A1 receptors in calf brain.

Authors:  A Garritsen; A P Ijzerman; M W Beukers; E J Cragoe; W Soudijn
Journal:  Biochem Pharmacol       Date:  1990-08-15       Impact factor: 5.858

8.  A1 adenosine-receptor antagonists activate chloride efflux from cystic fibrosis cells.

Authors:  O Eidelman; C Guay-Broder; P J van Galen; K A Jacobson; C Fox; R J Turner; Z I Cabantchik; H B Pollard
Journal:  Proc Natl Acad Sci U S A       Date:  1992-06-15       Impact factor: 11.205

9.  Binding of the A1-selective adenosine antagonist 8-cyclopentyl-1,3-dipropylxanthine to rat brain membranes.

Authors:  R F Bruns; J H Fergus; E W Badger; J A Bristol; L A Santay; J D Hartman; S J Hays; C C Huang
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1987-01       Impact factor: 3.000

Review 10.  Adenosine A1 and A2 receptors: structure--function relationships.

Authors:  P J van Galen; G L Stiles; G Michaels; K A Jacobson
Journal:  Med Res Rev       Date:  1992-09       Impact factor: 12.944
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  76 in total

Review 1.  A(2A) adenosine receptors in human peripheral blood cells.

Authors:  S Gessi; K Varani; S Merighi; E Ongini; P A Borea
Journal:  Br J Pharmacol       Date:  2000-01       Impact factor: 8.739

2.  A(2A) adenosine receptor deficiency attenuates brain injury induced by transient focal ischemia in mice.

Authors:  J F Chen; Z Huang; J Ma; J Zhu; R Moratalla; D Standaert; M A Moskowitz; J S Fink; M A Schwarzschild
Journal:  J Neurosci       Date:  1999-11-01       Impact factor: 6.167

3.  CoMFA-based comparison of two models of binding site on adenosine A1 receptor.

Authors:  I Doytchinova
Journal:  J Comput Aided Mol Des       Date:  2001-01       Impact factor: 3.686

4.  Orally active adenosine A(1) receptor agonists with antinociceptive effects in mice.

Authors:  Ilia Korboukh; Emily A Hull-Ryde; Joseph E Rittiner; Amarjit S Randhawa; Jennifer Coleman; Brendan J Fitzpatrick; Vincent Setola; William P Janzen; Stephen V Frye; Mark J Zylka; Jian Jin
Journal:  J Med Chem       Date:  2012-07-16       Impact factor: 7.446

Review 5.  Xanthines as adenosine receptor antagonists.

Authors:  Christa E Müller; Kenneth A Jacobson
Journal:  Handb Exp Pharmacol       Date:  2011

6.  Mutagenesis reveals structure-activity parallels between human A2A adenosine receptors and biogenic amine G protein-coupled receptors.

Authors:  Q Jiang; B X Lee; M Glashofer; A M van Rhee; K A Jacobson
Journal:  J Med Chem       Date:  1997-08-01       Impact factor: 7.446

7.  Adenosine receptor-induced second messenger production in adult guinea-pig cerebellum.

Authors:  F Hernández; D A Kendall; S P Alexander
Journal:  Br J Pharmacol       Date:  1993-11       Impact factor: 8.739

8.  Selective ligands for rat A3 adenosine receptors: structure-activity relationships of 1,3-dialkylxanthine 7-riboside derivatives.

Authors:  H O Kim; X D Ji; N Melman; M E Olah; G L Stiles; K A Jacobson
Journal:  J Med Chem       Date:  1994-11-11       Impact factor: 7.446

9.  Enhancement of adenosine A1 receptor functions by benzoylthiophenes in guinea pig tissues in vitro.

Authors:  E Leung; L K Walsh; L A Flippin; E J Kim; D A Lazar; C S Seran; E H Wong; R M Eglen
Journal:  Naunyn Schmiedebergs Arch Pharmacol       Date:  1995-08       Impact factor: 3.000

10.  Coupling of a transfected human brain A1 adenosine receptor in CHO-K1 cells to calcium mobilisation via a pertussis toxin-sensitive mechanism.

Authors:  P A Iredale; S P Alexander; S J Hill
Journal:  Br J Pharmacol       Date:  1994-04       Impact factor: 8.739
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