Literature DB >> 1513184

Adenosine A1 and A2 receptors: structure--function relationships.

P J van Galen1, G L Stiles, G Michaels, K A Jacobson.   

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Year:  1992        PMID： 1513184      PMCID： PMC3448285          DOI： 10.1002/med.2610120502

Source DB:  PubMed          Journal:  Med Res Rev        ISSN： 0198-6325            Impact factor:   12.944


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  166 in total

Review 1.  Structure and function of A1 adenosine receptors.

Authors:  J Linden
Journal:  FASEB J       Date:  1991-09       Impact factor: 5.191

2.  Adenosine receptors and beyond: molecular mechanisms of physiological regulation.

Authors:  G L Stiles
Journal:  Clin Res       Date:  1990-01

3.  A model for the antagonist binding site on the adenosine A1 receptor, based on steric, electrostatic, and hydrophobic properties.

Authors:  P J van Galen; H W van Vlijmen; A P IJzerman; W Soudijn
Journal:  J Med Chem       Date:  1990-06       Impact factor: 7.446

4.  Agonist photoaffinity labeling of A1 adenosine receptors: persistent activation reveals spare receptors.

Authors:  M J Lohse; K N Klotz; U Schwabe
Journal:  Mol Pharmacol       Date:  1986-10       Impact factor: 4.436

5.  Mechanism of A2 adenosine receptor activation. I. Blockade of A2 adenosine receptors by photoaffinity labeling.

Authors:  M J Lohse; K N Klotz; U Schwabe
Journal:  Mol Pharmacol       Date:  1991-04       Impact factor: 4.436

6.  Sleep improvement in dogs after oral administration of mioflazine, a nucleoside transport inhibitor.

Authors:  A Wauquier; H Van Belle; W A Van den Broeck; P A Janssen
Journal:  Psychopharmacology (Berl)       Date:  1987       Impact factor: 4.530

7.  Model for the structure of bacteriorhodopsin based on high-resolution electron cryo-microscopy.

Authors:  R Henderson; J M Baldwin; T A Ceska; F Zemlin; E Beckmann; K H Downing
Journal:  J Mol Biol       Date:  1990-06-20       Impact factor: 5.469

8.  Effects of 8-phenyl and 8-cycloalkyl substituents on the activity of mono-, di-, and trisubstituted alkylxanthines with substitution at the 1-, 3-, and 7-positions.

Authors:  M T Shamim; D Ukena; W L Padgett; J W Daly
Journal:  J Med Chem       Date:  1989-06       Impact factor: 7.446

9.  Guanine nucleotide and cation regulation of the binding of [3H]cyclohexyladenosine and [3H]diethylphenylxanthine to adenosine A1 receptors in brain membranes.

Authors:  R R Goodman; M J Cooper; M Gavish; S H Snyder
Journal:  Mol Pharmacol       Date:  1982-03       Impact factor: 4.436

10.  Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors.

Authors:  K A Jacobson; S Barone; U Kammula; G L Stiles
Journal:  J Med Chem       Date:  1989-05       Impact factor: 7.446
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  41 in total

1.  Substitution of a mutant alpha2a-adrenergic receptor via "hit and run" gene targeting reveals the role of this subtype in sedative, analgesic, and anesthetic-sparing responses in vivo.

Authors:  P P Lakhlani; L B MacMillan; T Z Guo; B A McCool; D M Lovinger; M Maze; L E Limbird
Journal:  Proc Natl Acad Sci U S A       Date:  1997-09-02       Impact factor: 11.205

2.  Immunological identification of A2 adenosine receptors by two antipeptide antibody preparations.

Authors:  T M Palmer; K A Jacobson; G L Stiles
Journal:  Mol Pharmacol       Date:  1992-09       Impact factor: 4.436

3.  Molecular modeling of adenosine receptors. I. The ligand binding site on the A1 receptor.

Authors:  A P IJzerman; P J Van Galen; K A Jacobson
Journal:  Drug Des Discov       Date:  1992

4.  Chemical modification and irreversible inhibition of striatal A2a adenosine receptors.

Authors:  K A Jacobson; G L Stiles; X D Ji
Journal:  Mol Pharmacol       Date:  1992-07       Impact factor: 4.436

5.  Thermodynamic in vitro studies as a method to investigate the pharmacodynamic behavior of adenosine A1 receptor ligands.

Authors:  A Dalpiaz; A Scatturin; B Pavan; K Varani; A P IJzerman; P Andrea Borea
Journal:  Pharm Res       Date:  1999-07       Impact factor: 4.200

6.  Adenosine receptor-induced second messenger production in adult guinea-pig cerebellum.

Authors:  F Hernández; D A Kendall; S P Alexander
Journal:  Br J Pharmacol       Date:  1993-11       Impact factor: 8.739

7.  Coupling of a transfected human brain A1 adenosine receptor in CHO-K1 cells to calcium mobilisation via a pertussis toxin-sensitive mechanism.

Authors:  P A Iredale; S P Alexander; S J Hill
Journal:  Br J Pharmacol       Date:  1994-04       Impact factor: 8.739

8.  Stimulation of human umbilical vein endothelial cell proliferation by A2-adenosine and beta 2-adrenoceptors.

Authors:  V Sexl; G Mancusi; S Baumgartner-Parzer; W Schütz; M Freissmuth
Journal:  Br J Pharmacol       Date:  1995-04       Impact factor: 8.739

9.  Structure-activity relationships of 8-styrylxanthines as A2-selective adenosine antagonists.

Authors:  K A Jacobson; C Gallo-Rodriguez; N Melman; B Fischer; M Maillard; A van Bergen; P J van Galen; Y Karton
Journal:  J Med Chem       Date:  1993-05-14       Impact factor: 7.446

Review 10.  Adenosine receptors and asthma in humans.

Authors:  C N Wilson
Journal:  Br J Pharmacol       Date:  2008-10       Impact factor: 8.739
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