Literature DB >> 16699973

A Phase II trial of epothilone B analogue BMS-247550 (NSC #710428) ixabepilone, in patients with advanced pancreas cancer: a Southwest Oncology Group study.

Robert P Whitehead1, Sheryl McCoy, Saul E Rivkin, Howard M Gross, Marcel E Conrad, Gary C Doolittle, Robert A Wolff, J Wendall Goodwin, Shaker R Dakhil, James L Abbruzzese.   

Abstract

PURPOSE: The purpose of this Phase II multi-institutional study was to define the efficacy and toxicity of ixabepilone in patients with advance pancreatic adenocarcinoma. PATIENTS AND METHODS: Patients were required to have pancreatic adenocarcinoma and metastatic or recurrent disease that was not amenable to curative resection. Performance status was 0-1, and patients could not have had prior chemotherapy, or chemoradiation therapy for their advanced disease although prior local palliative radiation was allowed. Ixabepilone was administered iv as a 3 hour infusion every 21 days. Initially, the dose was 50 mg/m(2) but this was lowered to 40 mg/m(2) shortly after the trial opened because of concerns about neurotoxicity.
RESULTS: Sixty-two patients were registered however 2 were ineligible because they did not have recurrent or metastatic disease. For the 60 eligible patients, 22 had performance status of 0 and 38 performance status of 1. The estimated 6-month survival was 60% (95% CI 48%-72%) with a median survival of 7.2 months and an estimated time to treatment failure of 2.3 months. Out of 56 patients with measurable disease there were 5 confirmed partial responses for a confirmed response probability of 9% (95% CI 3%-20%) and 7 unconfirmed partial responses for an overall response probability of 21% (95% CI 12%-34%). Common toxicities were neutropenia/granulocytopenia, nausea and vomiting and neuropathy. There was one death, cause not determined but judged "possibly" related to treatment.
CONCLUSION: Ixabepilone shows encouraging activity in patients with advanced pancreatic cancer and should be investigated further in this disease.

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Year:  2006        PMID: 16699973     DOI: 10.1007/s10637-006-8440-x

Source DB:  PubMed          Journal:  Invest New Drugs        ISSN: 0167-6997            Impact factor:   3.850


  13 in total

1.  BMS-247550: a novel epothilone analog with a mode of action similar to paclitaxel but possessing superior antitumor efficacy.

Authors:  F Y Lee; R Borzilleri; C R Fairchild; S H Kim; B H Long; C Reventos-Suarez; G D Vite; W C Rose; R A Kramer
Journal:  Clin Cancer Res       Date:  2001-05       Impact factor: 12.531

2.  New guidelines to evaluate the response to treatment in solid tumors. European Organization for Research and Treatment of Cancer, National Cancer Institute of the United States, National Cancer Institute of Canada.

Authors:  P Therasse; S G Arbuck; E A Eisenhauer; J Wanders; R S Kaplan; L Rubinstein; J Verweij; M Van Glabbeke; A T van Oosterom; M C Christian; S G Gwyther
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3.  Phase II trial of paclitaxel and granulocyte colony-stimulating factor in patients with pancreatic carcinoma: a Southwest Oncology Group study.

Authors:  R P Whitehead; J Jacobson; T D Brown; S A Taylor; G R Weiss; J S Macdonald
Journal:  J Clin Oncol       Date:  1997-06       Impact factor: 44.544

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Authors:  John S Macdonald; Sheryl McCoy; Robert P Whitehead; Syma Iqbal; James L Wade; Jeffrey K Giguere; James L Abbruzzese
Journal:  Invest New Drugs       Date:  2005-10       Impact factor: 3.850

5.  An investigational new drug treatment program for patients with gemcitabine: results for over 3000 patients with pancreatic carcinoma.

Authors:  A M Storniolo; N H Enas; C A Brown; M Voi; M L Rothenberg; R Schilsky
Journal:  Cancer       Date:  1999-03-15       Impact factor: 6.860

6.  Phase II trial of gemcitabine (2,2'-difluorodeoxycytidine) in patients with adenocarcinoma of the pancreas.

Authors:  E S Casper; M R Green; D P Kelsen; R T Heelan; T D Brown; C D Flombaum; B Trochanowski; P G Tarassoff
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7.  Phase I clinical and pharmacokinetic study of BMS-247550, a novel derivative of epothilone B, in solid tumors.

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Authors:  Henry Q Xiong; Arthur Rosenberg; Albert LoBuglio; William Schmidt; Robert A Wolff; John Deutsch; Michael Needle; James L Abbruzzese
Journal:  J Clin Oncol       Date:  2004-07-01       Impact factor: 44.544

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Authors:  Caio M Rocha Lima; Mark R Green; Robert Rotche; Wilson H Miller; G Mark Jeffrey; Laura A Cisar; Adele Morganti; Nicoletta Orlando; Gabriela Gruia; Langdon L Miller
Journal:  J Clin Oncol       Date:  2004-09-15       Impact factor: 44.544

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  18 in total

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Journal:  Invest New Drugs       Date:  2011-11-10       Impact factor: 3.850

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Authors:  Gregory Friberg; Hedy Lee Kindler
Journal:  Curr Oncol Rep       Date:  2005-05       Impact factor: 5.075

Review 3.  Chemotherapy-induced peripheral neuropathy: clinical features, diagnosis, prevention and treatment strategies.

Authors:  Gerardo Gutiérrez-Gutiérrez; María Sereno; Ambrosio Miralles; Enrique Casado-Sáenz; Eduardo Gutiérrez-Rivas
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4.  Phase II trials of dolastatin-10 in advanced pancreaticobiliary cancers.

Authors:  Hedy L Kindler; Peter K Tothy; Robert Wolff; Richard A McCormack; James L Abbruzzese; Sridhar Mani; Kurombi T Wade-Oliver; Everett E Vokes
Journal:  Invest New Drugs       Date:  2005-10       Impact factor: 3.850

5.  A Phase II trial of epothilone B analogue BMS-247550 (NSC #710428) ixabepilone, in patients with advanced pancreas cancer: a Southwest Oncology Group study.

Authors:  Robert P Whitehead; Sheryl McCoy; Saul E Rivkin; Howard M Gross; Marcel E Conrad; Gary C Doolittle; Robert A Wolff; J Wendall Goodwin; Shaker R Dakhil; James L Abbruzzese
Journal:  Invest New Drugs       Date:  2006-11       Impact factor: 3.850

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7.  Ixabepilone (ixempra), a therapeutic option for locally advanced or metastatic breast cancer.

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8.  Phase I trial of ixabepilone administered as three oral doses each separated by 6 hours every 3 weeks in patients with advanced solid tumors.

Authors:  Pamela L Kunz; Aiwu R He; A Dimitrios Colevas; Michael J Pishvaian; Jimmy J Hwang; Pamela L Clemens; Marianne Messina; Remigiusz Kaleta; Fernanda Abrahao; Branimir I Sikic; John L Marshall
Journal:  Invest New Drugs       Date:  2012-02-14       Impact factor: 3.850

9.  Ixabepilone: a new chemotherapeutic option for refractory metastatic breast cancer.

Authors:  Shannon Puhalla; Adam Brufsky
Journal:  Biologics       Date:  2008-09

10.  Novel microtubule-targeting agents - the epothilones.

Authors:  Kit L Cheng; Thomas Bradley; Daniel R Budman
Journal:  Biologics       Date:  2008-12
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