Literature DB >> 1590691

In vitro activities of chloroquine in combination with chlorpromazine or prochlorperazine against isolates of Plasmodium falciparum.

L K Basco1, J Le Bras.   

Abstract

The combinations of chloroquine plus chlorpromazine and chloroquine plus prochlorperazine were evaluated in vitro for potentiation against isolates of Plasmodium falciparum. Potentiation was observed against all chloroquine-resistant isolates. There was no potentiation against 8 of 10 chloroquine-susceptible isolates. The results indicated that the phenothiazines can potentiate chloroquine action against resistant parasites found in natural conditions.

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Year:  1992        PMID： 1590691      PMCID： PMC189259          DOI： 10.1128/AAC.36.1.209

Source DB:  PubMed          Journal:  Antimicrob Agents Chemother        ISSN： 0066-4804            Impact factor:   5.191


  10 in total

1.  Reversal of chloroquine resistance with desipramine in isolates of Plasmodium falciparum from Central and West Africa.

Authors:  L K Basco; J Le Bras
Journal:  Trans R Soc Trop Med Hyg       Date:  1990 Jul-Aug       Impact factor: 2.184

2.  Tricyclic antidepressant plasma level monitoring: intraindividual variability in everyday practice.

Authors:  S Vandel; G Bertschy; S Nezeloff; B Bonin; R Volmat
Journal:  Eur J Clin Pharmacol       Date:  1990       Impact factor: 2.953

3.  Reversal of chloroquine resistance with cyproheptadine in 'wild' strains of Plasmodium falciparum.

Authors:  L K Basco; J Le Bras
Journal:  Trans R Soc Trop Med Hyg       Date:  1991 Mar-Apr       Impact factor: 2.184

4.  Field study of cyproheptadine/chloroquine synergism in falciparum malaria.

Authors:  A Björkman; M Willcox; C M Kihamia; L F Mahikwano; P A Howard; A Häkansson; D Warhurst
Journal:  Lancet       Date:  1990-07-07       Impact factor: 79.321

5.  Antihistaminic drugs that reverse chloroquine resistance in Plasmodium falciparum.

Authors:  W Peters; R Ekong; B L Robinson; D C Warhurst; X Q Pan
Journal:  Lancet       Date:  1989-08-05       Impact factor: 79.321

6.  Plasmodium falciparum: modulation by calcium antagonists of resistance to chloroquine, desethylchloroquine, quinine, and quinidine in vitro.

Authors:  D E Kyle; A M Oduola; S K Martin; W K Milhous
Journal:  Trans R Soc Trop Med Hyg       Date:  1990 Jul-Aug       Impact factor: 2.184

7.  Reversal of chloroquine resistance in malaria parasite Plasmodium falciparum by desipramine.

Authors:  A J Bitonti; A Sjoerdsma; P P McCann; D E Kyle; A M Oduola; R N Rossan; W K Milhous; D E Davidson
Journal:  Science       Date:  1988-12-02       Impact factor: 47.728

Review 8.  Plasma level monitoring of antipsychotic drugs. Clinical utility.

Authors:  S G Dahl
Journal:  Clin Pharmacokinet       Date:  1986 Jan-Feb       Impact factor: 6.447

9.  Reversal of chloroquine resistance in Plasmodium falciparum by verapamil.

Authors:  S K Martin; A M Oduola; W K Milhous
Journal:  Science       Date:  1987-02-20       Impact factor: 47.728

10.  In vitro study of drug sensitivity of Plasmodium falciparum: evaluation of a new semi-micro test.

Authors:  J Le Bras; P Deloron
Journal:  Am J Trop Med Hyg       Date:  1983-05       Impact factor: 2.345
  10 in total
  9 in total

1.  Role of the neurotransmitter reuptake-blocking activity of antidepressants in reversing chloroquine resistance in vitro in Plasmodium falciparum.

Authors:  D Taylor; J C Walden; A H Robins; P J Smith
Journal:  Antimicrob Agents Chemother       Date:  2000-10       Impact factor: 5.191

2.  Assessment of three in vitro tests and an in vivo test for chloroquine resistance in Plasmodium falciparum clinical isolates.

Authors:  J Bickii; L K Basco; P Ringwald
Journal:  J Clin Microbiol       Date:  1998-01       Impact factor: 5.948

3.  Searching for new antimalarial therapeutics amongst known drugs.

Authors:  Jennifer L Weisman; Ally P Liou; Anang A Shelat; Fred E Cohen; R Kiplin Guy; Joseph L DeRisi
Journal:  Chem Biol Drug Des       Date:  2006-06       Impact factor: 2.817

4.  Nonylphenolethoxylates as malarial chloroquine resistance reversal agents.

Authors:  I Crandall; J Charuk; K C Kain
Journal:  Antimicrob Agents Chemother       Date:  2000-09       Impact factor: 5.191

Review 5.  Thioridazine: resurrection as an antimicrobial agent?

Authors:  H K R Thanacoody
Journal:  Br J Clin Pharmacol       Date:  2007-08-31       Impact factor: 4.335

6.  Reversal of mefloquine and quinine resistance in Plasmodium falciparum with NP30.

Authors:  Michelle Ciach; Kathleen Zong; Kevin C Kain; Ian Crandall
Journal:  Antimicrob Agents Chemother       Date:  2003-08       Impact factor: 5.191

Review 7.  A bibliometric review of drug repurposing.

Authors:  Nancy C Baker; Sean Ekins; Antony J Williams; Alexander Tropsha
Journal:  Drug Discov Today       Date:  2018-01-09       Impact factor: 7.851

8.  Evidence for the contribution of the hemozoin synthesis pathway of the murine Plasmodium yoelii to the resistance to artemisinin-related drugs.

Authors:  Benoit Witkowski; Joel Lelièvre; Marie-Laure Nicolau-Travers; Xavier Iriart; Patrice Njomnang Soh; Fatima Bousejra-Elgarah; Bernard Meunier; Antoine Berry; Françoise Benoit-Vical
Journal:  PLoS One       Date:  2012-03-05       Impact factor: 3.240

9.  Plasmodium falciparum and Plasmodium vivax Demonstrate Contrasting Chloroquine Resistance Reversal Phenotypes.

Authors:  Grennady Wirjanata; Irene Handayuni; Pak Prayoga; Leo Leonardo; Dwi Apriyanti; Leily Trianty; Ruland Wandosa; Basbak Gobay; Enny Kenangalem; Jeanne Rini Poespoprodjo; Rintis Noviyanti; Dennis E Kyle; Qin Cheng; Ric N Price; Jutta Marfurt
Journal:  Antimicrob Agents Chemother       Date:  2017-07-25       Impact factor: 5.191
  9 in total

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