Literature DB >> 15047563

Antimalarial and antileishmanial activities of aroyl-pyrrolyl-hydroxyamides, a new class of histone deacetylase inhibitors.

Antonello Mai, Ilaria Cerbara, Sergio Valente, Silvio Massa, Larry A Walker, Babu L Tekwani.   

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Year:  2004        PMID: 15047563      PMCID: PMC375343          DOI: 10.1128/AAC.48.4.1435-1436.2004

Source DB:  PubMed          Journal:  Antimicrob Agents Chemother        ISSN: 0066-4804            Impact factor:   5.191


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  9 in total

Review 1.  Chromatin remodelling during the life cycle of trypanosomatids.

Authors:  S I Belli
Journal:  Int J Parasitol       Date:  2000-05       Impact factor: 3.981

2.  Pentamidine isethionate as treatment and secondary prophylaxis for disseminated cutaneous leishmaniasis during HIV infection: case report.

Authors:  L Calza; G Marinacci; R Manfredi; V Colangeli; L Fortunato; F Chiodo
Journal:  J Chemother       Date:  2001-12       Impact factor: 1.714

3.  Anti-malarial effect of histone deacetylation inhibitors and mammalian tumour cytodifferentiating agents.

Authors:  K T Andrews; A Walduck; M J Kelso; D P Fairlie; A Saul; P G Parsons
Journal:  Int J Parasitol       Date:  2000-05       Impact factor: 3.981

Review 4.  Chemotherapy of leishmaniasis.

Authors:  Simon L Croft; Vanessa Yardley
Journal:  Curr Pharm Des       Date:  2002       Impact factor: 3.116

5.  Apicidin: a novel antiprotozoal agent that inhibits parasite histone deacetylase.

Authors:  S J Darkin-Rattray; A M Gurnett; R W Myers; P M Dulski; T M Crumley; J J Allocco; C Cannova; P T Meinke; S L Colletti; M A Bednarek; S B Singh; M A Goetz; A W Dombrowski; J D Polishook; D M Schmatz
Journal:  Proc Natl Acad Sci U S A       Date:  1996-11-12       Impact factor: 11.205

6.  Binding mode analysis of 3-(4-benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: a new synthetic histone deacetylase inhibitor inducing histone hyperacetylation, growth inhibition, and terminal cell differentiation.

Authors:  Antonello Mai; Silvio Massa; Rino Ragno; Monica Esposito; Gianluca Sbardella; Giuseppina Nocca; Roberto Scatena; Florian Jesacher; Peter Loidl; Gerald Brosch
Journal:  J Med Chem       Date:  2002-04-25       Impact factor: 7.446

7.  3-(4-Aroyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-alkylamides as a new class of synthetic histone deacetylase inhibitors. 1. Design, synthesis, biological evaluation, and binding mode studies performed through three different docking procedures.

Authors:  Antonello Mai; Silvio Massa; Rino Ragno; Ilaria Cerbara; Florian Jesacher; Peter Loidl; Gerald Brosch
Journal:  J Med Chem       Date:  2003-02-13       Impact factor: 7.446

8.  Parasite lactate dehydrogenase as an assay for Plasmodium falciparum drug sensitivity.

Authors:  M T Makler; J M Ries; J A Williams; J E Bancroft; R C Piper; B L Gibbins; D J Hinrichs
Journal:  Am J Trop Med Hyg       Date:  1993-06       Impact factor: 2.345

9.  Cytotoxicity of T-2 toxin and its metabolites determined with the neutral red cell viability assay.

Authors:  H Babich; E Borenfreund
Journal:  Appl Environ Microbiol       Date:  1991-07       Impact factor: 4.792

  9 in total
  15 in total

Review 1.  Macrocyclic histone deacetylase inhibitors.

Authors:  Sandra C Mwakwari; Vishal Patil; William Guerrant; Adegboyega K Oyelere
Journal:  Curr Top Med Chem       Date:  2010       Impact factor: 3.295

Review 2.  Epigenetics in Plasmodium: what do we really know?

Authors:  Catherine J Merrick; Manoj T Duraisingh
Journal:  Eukaryot Cell       Date:  2010-06-18

Review 3.  Bromodomains in Protozoan Parasites: Evolution, Function, and Opportunities for Drug Development.

Authors:  Victoria Jeffers; Chunlin Yang; Sherri Huang; William J Sullivan
Journal:  Microbiol Mol Biol Rev       Date:  2017-01-11       Impact factor: 11.056

4.  Cytotoxic effect of curcumin on malaria parasite Plasmodium falciparum: inhibition of histone acetylation and generation of reactive oxygen species.

Authors:  Long Cui; Jun Miao; Liwang Cui
Journal:  Antimicrob Agents Chemother       Date:  2006-12-04       Impact factor: 5.191

5.  Introducing histone modification in trypanosomes.

Authors:  David Horn
Journal:  Trends Parasitol       Date:  2007-04-11

Review 6.  Leishmaniasis treatment--a challenge that remains: a review.

Authors:  Dilvani O Santos; Carlos E R Coutinho; Maria F Madeira; Carolina G Bottino; Rodrigo T Vieira; Samara B Nascimento; Alice Bernardino; Saulo C Bourguignon; Suzana Corte-Real; Rosa T Pinho; Carlos Rangel Rodrigues; Helena C Castro
Journal:  Parasitol Res       Date:  2008-06       Impact factor: 2.289

7.  Potent antimalarial activity of histone deacetylase inhibitor analogues.

Authors:  K T Andrews; T N Tran; A J Lucke; P Kahnberg; G T Le; G M Boyle; D L Gardiner; T S Skinner-Adams; D P Fairlie
Journal:  Antimicrob Agents Chemother       Date:  2008-01-22       Impact factor: 5.191

8.  Novel inhibitor of Plasmodium histone deacetylase that cures P. berghei-infected mice.

Authors:  S Agbor-Enoh; C Seudieu; E Davidson; A Dritschilo; M Jung
Journal:  Antimicrob Agents Chemother       Date:  2009-02-17       Impact factor: 5.191

9.  An apicomplexan ankyrin-repeat histone deacetylase with relatives in photosynthetic eukaryotes.

Authors:  S Dean Rider; Guan Zhu
Journal:  Int J Parasitol       Date:  2008-12-24       Impact factor: 3.981

10.  A kernel for open source drug discovery in tropical diseases.

Authors:  Leticia Ortí; Rodrigo J Carbajo; Ursula Pieper; Narayanan Eswar; Stephen M Maurer; Arti K Rai; Ginger Taylor; Matthew H Todd; Antonio Pineda-Lucena; Andrej Sali; Marc A Marti-Renom
Journal:  PLoS Negl Trop Dis       Date:  2009-04-21
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