Literature DB >> 1475316

Thiazolo[3,2-a]pyrimidine derivatives as calcium antagonists.

A Balkan1, S Uma, M Ertan, W Wiegrebe.   

Abstract

Some new thiazolo[3,2-a]pyrimidine derivatives were prepared refluxing 2-thioxo-1,2,3,4-tetrahydropyrimidine derivatives with phenacyl bromide in glacial acetic acid. Calcium antagonistic activities of these compounds were evaluated in K(+)-depolarized rat aorta, using nifedipine as reference compound.

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Year:  1992        PMID： 1475316

Source DB:  PubMed          Journal:  Pharmazie        ISSN： 0031-7144            Impact factor:   1.267


  5 in total

1.  A rapid access to novel and diverse 3-oxothiazolo[3,2-c]pyrimidine-8-carboxylates using multicomponent Mannich cyclisation reactions.

Authors:  Muhammet Yıldırım; Derya Çelikel
Journal:  Mol Divers       Date:  2014-08-24       Impact factor: 2.943

2.  Crystal structures of two 6-(2-hy-droxy-benzo-yl)-5H-thia-zolo[3,2-a]pyrimidin-5-ones.

Authors:  Ligia R Gomes; John Nicolson Low; Fernando Cagide; Fernanda Borges
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2015-06-13

3.  Synthesis, Antibacterial and Antitubercular Activities of Some 5H-Thiazolo[3,2-a]pyrimidin-5-ones and Sulfonic Acid Derivatives.

Authors:  Dong Cai; Zhi-Hua Zhang; Yu Chen; Xin-Jia Yan; Liang-Jing Zou; Ya-Xin Wang; Xue-Qi Liu
Journal:  Molecules       Date:  2015-09-10       Impact factor: 4.411

4.  Herbicidal properties of antihypertensive drugs: calcium channel blockers.

Authors:  Hannan Safiyyah Tan Sian Hui Abdullah; Poh Wai Chia; Dzolkhifli Omar; Tse Seng Chuah
Journal:  Sci Rep       Date:  2021-07-09       Impact factor: 4.379

Review 5.  Design and synthesis of some substituted thiazolo[3,2-a]pyrimidine derivatives of potential biological activities.

Authors:  Samia G Abdel Moty; Mostafa A Hussein; Salah A Abdel Aziz; Mahrous A Abou-Salim
Journal:  Saudi Pharm J       Date:  2013-12-28       Impact factor: 4.330
  5 in total

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