Literature DB >> 10508044

Potentiation of artemisinin activity against chloroquine-resistant Plasmodium falciparum strains by using heme models.

F Benoit-Vical1, A Robert, B Meunier.   

Abstract

The influence of different metalloporphyrin derivatives on the antimalarial activity of artemisinin was studied with two chloroquine-resistant strains of Plasmodium falciparum (FcB1-Colombia and FcM29-Cameroon) cultured in human erythrocytes. This potentiation study indicates that the manganese complex of meso-tetrakis(4-sulfonatophenyl)porphyrin has a significant synergistic effect on the activity of artemisinin against both Plasmodium strains.

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Year:  1999        PMID： 10508044      PMCID： PMC89520          DOI： 10.1128/AAC.43.10.2555

Source DB:  PubMed          Journal:  Antimicrob Agents Chemother        ISSN： 0066-4804            Impact factor:   5.191


  13 in total

1.  In vitro antimalarial activity of vegetal extracts used in West African traditional medicine.

Authors:  F Benoit; A Valentin; Y Pelissier; F Diafouka; C Marion; D Kone-Bamba; M Kone; M Mallie; A Yapo; J M Bastide
Journal:  Am J Trop Med Hyg       Date:  1996-01       Impact factor: 2.345

2.  Bisbenzylisoquinolines as modulators of chloroquine resistance in Plasmodium falciparum and multidrug resistance in tumor cells.

Authors:  F Frappier; A Jossang; J Soudon; F Calvo; P Rasoanaivo; S Ratsimamanga-Urverg; J Saez; J Schrevel; P Grellier
Journal:  Antimicrob Agents Chemother       Date:  1996-06       Impact factor: 5.191

3.  Mechanism-based design, synthesis, and in vitro antimalarial testing of new 4-methylated trioxanes structurally related to artemisinin: the importance of a carbon-centered radical for antimalarial activity.

Authors:  G H Posner; C H Oh; D Wang; L Gerena; W K Milhous; S R Meshnick; W Asawamahasadka
Journal:  J Med Chem       Date:  1994-04-29       Impact factor: 7.446

4.  Free radicals and antioxidants.

Authors:  S R Meshnick
Journal:  Lancet       Date:  1994-11-19       Impact factor: 79.321

5.  The antimalarial action on Plasmodium falciparum of qinghaosu and artesunate in combination with agents which modulate oxidant stress.

Authors:  S R Krungkrai; Y Yuthavong
Journal:  Trans R Soc Trop Med Hyg       Date:  1987       Impact factor: 2.184

Review 6.  Artemisinin and the antimalarial endoperoxides: from herbal remedy to targeted chemotherapy.

Authors:  S R Meshnick; T E Taylor; S Kamchonwongpaisan
Journal:  Microbiol Rev       Date:  1996-06

7.  The interaction of artemisinin with malarial hemozoin.

Authors:  Y L Hong; Y Z Yang; S R Meshnick
Journal:  Mol Biochem Parasitol       Date:  1994-01       Impact factor: 1.759

8.  Reversal of chloroquine resistance in Plasmodium falciparum by verapamil.

Authors:  S K Martin; A M Oduola; W K Milhous
Journal:  Science       Date:  1987-02-20       Impact factor: 47.728

Review 9.  Qinghaosu (artemisinin): an antimalarial drug from China.

Authors:  D L Klayman
Journal:  Science       Date:  1985-05-31       Impact factor: 47.728

10.  In vitro antimalarial activity of penduline, a bisbenzylisoquinoline from Isopyrum thalictroides.

Authors:  A Valentin; F Benoit-Vical; C Moulis; E Stanislas; M Mallié; I Fouraste; J M Bastide
Journal:  Antimicrob Agents Chemother       Date:  1997-10       Impact factor: 5.191
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  4 in total

1.  In vitro and in vivo potentiation of artemisinin and synthetic endoperoxide antimalarial drugs by metalloporphyrins.

Authors:  F Benoit-Vical; A Robert; B Meunier
Journal:  Antimicrob Agents Chemother       Date:  2000-10       Impact factor: 5.191

2.  Trioxaquines are new antimalarial agents active on all erythrocytic forms, including gametocytes.

Authors:  Françoise Benoit-Vical; Joël Lelièvre; Antoine Berry; Caroline Deymier; Odile Dechy-Cabaret; Jérôme Cazelles; Christophe Loup; Anne Robert; Jean-François Magnaval; Bernard Meunier
Journal:  Antimicrob Agents Chemother       Date:  2007-01-22       Impact factor: 5.191

3.  Mechanistic Investigation of the Specific Anticancer Property of Artemisinin and Its Combination with Aminolevulinic Acid for Enhanced Anticolorectal Cancer Activity.

Authors:  Jigang Wang; Jianbin Zhang; Yin Shi; Chengchao Xu; Chongjing Zhang; Yin Kwan Wong; Yew Mun Lee; Sanjeev Krishna; Yingke He; Teck Kwang Lim; Weiying Sim; Zi-Chun Hua; Han-Ming Shen; Qingsong Lin
Journal:  ACS Cent Sci       Date:  2017-06-28       Impact factor: 14.553

Review 4.  Oxidative stress in malaria.

Authors:  Sandro Percário; Danilo R Moreira; Bruno A Q Gomes; Michelli E S Ferreira; Ana Carolina M Gonçalves; Paula S O C Laurindo; Thyago C Vilhena; Maria F Dolabela; Michael D Green
Journal:  Int J Mol Sci       Date:  2012-12-03       Impact factor: 5.923
  4 in total

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