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16 in total

Review 1. Bioactivation of Selective Estrogen Receptor Modulators (SERMs).

Authors: Tamara S Dowers; Zhi-Hui Qin; Gregory R J Thatcher; Judy L Bolton
Journal: Chem Res Toxicol Date: 2006-09 Impact factor: 3.739

2. Metalloradical approach to 2H-chromenes.

Authors: Nanda D Paul; Sutanuva Mandal; Matthias Otte; Xin Cui; X Peter Zhang; Bas de Bruin
Journal: J Am Chem Soc Date: 2014-01-08 Impact factor: 15.419

3. Enantioselective copper-catalyzed alkynylation of benzopyranyl oxocarbenium ions.

Authors: Harathi D Srinivas; Prantik Maity; Glenn P A Yap; Mary P Watson
Journal: J Org Chem Date: 2015-04-07 Impact factor: 4.354

4. Nickel-catalyzed cross-coupling of chromene acetals and boronic acids.

Authors: Thomas J A Graham; Abigail G Doyle
Journal: Org Lett Date: 2012-03-02 Impact factor: 6.005

5. Construction of a database for the evaluation and the clinical management of patients with breast cancer treated with antiestrogens and/or aromatase inhibitors.

Authors: Francesca Giusti; Silva Ottanelli; Laura Masi; Antonietta Amedei; Maria Luisa Brandi; Alberto Falchetti
Journal: Clin Cases Miner Bone Metab Date: 2011-01

6. Flexible small molecular anti-estrogens with N,N-dialkylated-2,5-diethoxy-4-morpholinoaniline scaffold targets multiple estrogen receptor conformations.

Authors: Bethany K Asare; Emmanuel Yawson; Rajendram V Rajnarayanan
Journal: Cell Cycle Date: 2017-07-19 Impact factor: 4.534

(S)-(+)-4-[7-(2,2-dimethyl-1-oxopropoxy)-4-methyl-2-[4-[2-(1-piperidinyl)-ethoxy]phenyl]-2H-1-benzopyran-3-yl]-phenyl 2,2-dimethylpropanoate (EM-800): a highly potent, specific, and orally active nonsteroidal antiestrogen.

Review 1. Bioactivation of Selective Estrogen Receptor Modulators (SERMs).

2. Metalloradical approach to 2H-chromenes.

3. Enantioselective copper-catalyzed alkynylation of benzopyranyl oxocarbenium ions.

4. Nickel-catalyzed cross-coupling of chromene acetals and boronic acids.

5. Construction of a database for the evaluation and the clinical management of patients with breast cancer treated with antiestrogens and/or aromatase inhibitors.

6. Flexible small molecular anti-estrogens with N,N-dialkylated-2,5-diethoxy-4-morpholinoaniline scaffold targets multiple estrogen receptor conformations.

7. Application of screening methods, shape signatures and engineered biosensors in early drug discovery process.

8. Synthesis of 3,4-disubstituted 2H-benzopyrans through C-C bond formation via electrophilic cyclization.

9. Pharmacophore mapping of flavone derivatives for aromatase inhibition.

10. Identification of xenoestrogens in food additives by an integrated in silico and in vitro approach.