Literature DB >> 9207934

Pyridazinodiazepines as a high-affinity, P2-P3 peptidomimetic class of interleukin-1 beta-converting enzyme inhibitor.

R E Dolle1, C V Prasad, C P Prouty, J M Salvino, M M Awad, S J Schmidt, D Hoyer, T M Ross, T L Graybill, G J Speier, J Uhl, B E Miller, C T Helaszek, M A Ator.   

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Year:  1997        PMID: 9207934     DOI: 10.1021/jm9701637

Source DB:  PubMed          Journal:  J Med Chem        ISSN: 0022-2623            Impact factor:   7.446


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  3 in total

Review 1.  Small Molecule Active Site Directed Tools for Studying Human Caspases.

Authors:  Marcin Poreba; Aleksandra Szalek; Paulina Kasperkiewicz; Wioletta Rut; Guy S Salvesen; Marcin Drag
Journal:  Chem Rev       Date:  2015-11-09       Impact factor: 60.622

Review 2.  Caspase substrates and inhibitors.

Authors:  Marcin Poreba; Aleksandra Strózyk; Guy S Salvesen; Marcin Drag
Journal:  Cold Spring Harb Perspect Biol       Date:  2013-08-01       Impact factor: 10.005

3.  Solid-phase synthesis of tetrahydropyridazinedione-constrained peptides.

Authors:  Chang Won Kang; Sujeewa Ranatunga; Matthew P Sarnowski; Juan R Del Valle
Journal:  Org Lett       Date:  2014-10-08       Impact factor: 6.005

  3 in total

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