Literature DB >> 8576904

Nonpeptide angiotensin II receptor antagonists: the next generation in antihypertensive therapy.

R R Wexler1, W J Greenlee, J D Irvin, M R Goldberg, K Prendergast, R D Smith, P B Timmermans.   

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Year:  1996        PMID： 8576904     DOI： 10.1021/jm9504722

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  21 in total

1.  An efficient synthesis of a rationally designed 1,5 disubstituted imidazole AT(1) angiotensin II receptor antagonist: reorientation of imidazole pharmacophore groups in losartan reserves high receptor affinity and confirms docking studies.

Authors:  George Agelis; Panagiota Roumelioti; Amalia Resvani; Serdar Durdagi; Maria-Eleni Androutsou; Konstantinos Kelaidonis; Demetrios Vlahakos; Thomas Mavromoustakos; John Matsoukas
Journal:  J Comput Aided Mol Des       Date:  2010-07-10       Impact factor: 3.686

2.  Thermal analysis study of antihypertensive drugs telmisartan and cilazapril.

Authors:  Refaat Ahmed Saber; Ali Kamal Attia; Waheed Mohamed Salem
Journal:  Adv Pharm Bull       Date:  2014-02-07

Review 3.  Comparative safety and tolerability of angiotensin II receptor antagonists.

Authors:  L Mazzolai; M Burnier
Journal:  Drug Saf       Date:  1999-07       Impact factor: 5.606

4.  LAT1 activity of carboxylic acid bioisosteres: Evaluation of hydroxamic acids as substrates.

Authors:  Arik A Zur; Huan-Chieh Chien; Evan Augustyn; Andrew Flint; Nathan Heeren; Karissa Finke; Christopher Hernandez; Logan Hansen; Sydney Miller; Lawrence Lin; Kathleen M Giacomini; Claire Colas; Avner Schlessinger; Allen A Thomas
Journal:  Bioorg Med Chem Lett       Date:  2016-09-03       Impact factor: 2.823

5.  Efficient and improved synthesis of Telmisartan.

Authors:  A Sanjeev Kumar; Samir Ghosh; G N Mehta
Journal:  Beilstein J Org Chem       Date:  2010-03-11       Impact factor: 2.883

6.  Scaffold Morphing Identifies 3-Pyridyl Azetidine Ureas as Inhibitors of Nicotinamide Phosphoribosyltransferase (NAMPT).

Authors:  Daniel S Palacios; Erik L Meredith; Toshio Kawanami; Christopher M Adams; Xin Chen; Veronique Darsigny; Mark Palermo; Daniel Baird; Elizabeth L George; Chantale Guy; Jeffrey Hewett; Laryssa Tierney; Sachin Thigale; Louis Wang; Wilhelm A Weihofen
Journal:  ACS Med Chem Lett       Date:  2019-10-10       Impact factor: 4.345

7.  Design, synthesis, and evaluation of 5-sulfamoyl benzimidazole derivatives as novel angiotensin II receptor antagonists.

Authors:  Navneet Kaur; Amardeep Kaur; Yogita Bansal; Dhvanit I Shah; Gulshan Bansal; Manjeet Singh
Journal:  Bioorg Med Chem       Date:  2008-10-29       Impact factor: 3.641

Review 8.  Carboxylic acid (bio)isosteres in drug design.

Authors:  Carlo Ballatore; Donna M Huryn; Amos B Smith
Journal:  ChemMedChem       Date:  2013-01-29       Impact factor: 3.466

9.  α-Amino Acid-Isosteric α-Amino Tetrazoles.

Authors:  Ting Zhao; Katarzyna Kurpiewska; Justyna Kalinowska-Tłuścik; Eberhardt Herdtweck; Alexander Dömling
Journal:  Chemistry       Date:  2016-01-28       Impact factor: 5.236

10.  Transforming Suzuki-Miyaura cross-couplings of MIDA boronates into a green technology: no organic solvents.

Authors:  Nicholas A Isley; Fabrice Gallou; Bruce H Lipshutz
Journal:  J Am Chem Soc       Date:  2013-11-13       Impact factor: 15.419
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